Search Results - "Jass, Paul A."

Use of N-trifluoroacetyl-protected amino acid chlorides in peptide coupling reactions with virtually complete preservation of stereochemistry by Jass, Paul A, Rosso, Victor W, Racha, Saibaba, Soundararajan, Nachimuthu, Venit, John J, Rusowicz, Andrew, Swaminathan, Shankar, Livshitz, Julia, Delaney, Edward J

“…The use of protected amino acid chlorides for peptide coupling reactions has long been avoided due to the extensive racemization that commonly occurs during…”
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Total synthesis of (+)-breynolide by Williams, David R, Jass, Paul A, Tse, H. L. Allan, Gaston, Ricky D

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1,3-Dipolar cycloaddition annulations to the thieno[2,3-d]pyridazine, thieno[3,2-c]pyridine, and thieno[2,3-d]pyrimidine ring systems by New, James S, Christopher, William L, Jass, Paul A

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Regio- and stereoselective ring opening of epoxide with cyanoguanidine dianions, a facile synthesis of the KATP opener BMS-180448 by Chen, Bang-Chi, Quinlan, Sandra L, Reid, J.Gregory, Jass, Paul A, Robinson, Tonya P, Early, William A, Delaney, Edward J, Humora, Michael J, Madding, Gary D, Venit, John J, Winter, William J

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Process Development of 5-Fluoro-3-[3-[4-(5-methoxy-4-pyrimidinyl)-1- piperazinyl]propyl]-1H-indole Dihydrochloride by Anderson, Neal G, Ary, Thomas D, Berg, James L, Bernot, Peter J, Chan, Yeung Y, Chen, Chien-Kuang, Davies, Merrill L, DiMarco, John D, Dennis, Ronald D, Deshpande, Rajan P, Do, Hoang D, Droghini, Roberto, Early, William A, Gougoutas, Jack Z, Grosso, John A, Harris, John C, Haas, Oscar W, Jass, Paul A, Kim, Daniel H, Kodersha, Gus A, Kotnis, Atul S, LaJeunesse, Jean, Lust, David A, Madding, Gary D, Modi, Sandeep P, Moniot, Jerome L, Nguyen, Andrew, Palaniswamy, Venkatapuram, Phillipson, Douglas W, Simpson, James H, Thoraval, Dominique, Thurston, David A, Tse, Kai, Polomski, Robert E, Wedding, Donald L, Winter, William J

“…5-Fluoro-3-[3-[4-(5-methoxy-4-pyrimidinyl)-1-piperazinyl]propyl]-1H-indole dihydrochloride (1) facilitates 5-HT neurotransmission and was an antidepressant…”
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Regio- and stereoselective ring opening of epoxide with cyanoguanidine dianions, a facile synthesis of the K ATP opener BMS-180448 by Chen, Bang-Chi, Quinlan, Sandra L, Reid, J.Gregory, Jass, Paul A, Robinson, Tonya P, Early, William A, Delaney, Edward J, Humora, Michael J, Madding, Gary D, Venit, John J, Winter, William J

“…BMS-180448, (3S,4R)- 2, was prepared in 63% yield via a facile method which involved a new regio- and stereoselective ring opening of epoxide (3S,4S)- 12 with…”
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Process Development of 5-Fluoro-3-[3-[4-(5-methoxy-4-pyrimidinyl)-1- piperazinyl]propyl]-1 H -indole Dihydrochloride by Anderson, Neal G., Ary, Thomas D., Berg, James L., Bernot, Peter J., Chan, Yeung Y., Chen, Chien-Kuang, Davies, Merrill L., DiMarco, John D., Dennis, Ronald D., Deshpande, Rajan P., Do, Hoang D., Droghini, Roberto, Early, William A., Gougoutas, Jack Z., Grosso, John A., Harris, John C., Haas, Oscar W., Jass, Paul A., Kim, Daniel H., Kodersha, Gus A., Kotnis, Atul S., LaJeunesse, Jean, Lust, David A., Madding, Gary D., Modi, Sandeep P., Moniot, Jerome L., Nguyen, Andrew, Palaniswamy, Venkatapuram, Phillipson, Douglas W., Simpson, James H., Thoraval, Dominique, Thurston, David A., Tse, Kai, Polomski, Robert E., Wedding, Donald L., Winter, William J.

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