Search Results - "JARD, S"

Characterization of SR 121463A, a highly potent and selective, orally active vasopressin V2 receptor antagonist by Serradeil-Le Gal, C, Lacour, C, Valette, G, Garcia, G, Foulon, L, Galindo, G, Bankir, L, Pouzet, B, Guillon, G, Barberis, C, Chicot, D, Jard, S, Vilain, P, Garcia, C, Marty, E, Raufaste, D, Brossard, G, Nisato, D, Maffrand, J P, Le Fur, G

“…SR 121463A, a potent and selective, orally active, nonpeptide vasopressin V2 receptor antagonist, has been characterized in several in vitro and in vivo…”
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Mechanisms of action of vasopressin and vasopressin antagonists by Jard, S

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Tyr115 is the key residue for determining agonist selectivity in the V1a vasopressin receptor by Chini, B., Mouillac, B., Ala, Y., Balestre, M.N., Trumpp‐Kallmeyer, S., Hoflack, J., Elands, J., Hibert, M., Manning, M., Jard, S.

“…Using a three‐dimensional model of G protein‐coupled receptors (GPCR), we have previously succeeded in docking the neurohypophysial hormone…”
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Biochemical and pharmacological properties of SR 49059, a new, potent, nonpeptide antagonist of rat and human vasopressin V1a receptors by SERRADEIL-LE GAL, C, WAGNON, J, GUILLON, G, CANTAU, B, BARBERIS, C, TRUEBA, M, ALA, Y, JARD, S, GARCIA, C, LACOUR, C, GUIRAUDOU, P, CHRISTOPHE, P, VILLANOVA, G, NISATO, D, MAFFRAND, J. P, LE FUR, G

“…SR 49059, a new potent and selective orally active, nonpeptide vasopressin (AVP) antagonist has been characterized in several in vitro and in vivo models. SR…”
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Localization and pharmacological characterization of high affinity binding sites for vasopressin and oxytocin in the rat brain by light microscopic autoradiography by Tribollet, E, Barberis, C, Jard, S, Dubois-Dauphin, M, Dreifuss, J J

“…Sites which bind tritiated vasopressin (AVP) with high affinity were detected in the brain of male, adult rats, by light microscopic autoradiography. Their…”
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Oxytocin receptors in the central nervous system. Distribution, development, and species differences by Tribollet, E, Dubois-Dauphin, M, Dreifuss, J J, Barberis, C, Jard, S

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Tyr115 is the key residue for determining agonist selectivity in the V1a vasopressin receptor by Chini, B., Mouillac, B., Ala, Y., Balestre, M.N., Trumpp-Kallmeyer, S., Hoflack, J., Elands, J., Hibert, M., Manning, M., Jard, S.

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Angiotensin II and dopamine modulate both cAMP and inositol phosphate productions in anterior pituitary cells. Involvement in prolactin secretion by Enjalbert, A, Sladeczek, F, Guillon, G, Bertrand, P, Shu, C, Epelbaum, J, Garcia-Sainz, A, Jard, S, Lombard, C, Kordon, C

“…Despite their opposite effects on prolactin secretion, both dopamine and angiotensin II inhibit adenylate cyclase activity in homogenates of anterior pituitary…”
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[3H]-[Thr4,Gly7]OT: a highly selective ligand for central and peripheral OT receptors by Elands, J, Barberis, C, Jard, S

“…Oxytocin receptors in rat hippocampal synaptic plasma membranes were compared with mammary gland and uterine oxytocin receptors. For this purpose, a highly…”
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Vasopressin antagonists allow demonstration of a novel type of vasopressin receptor in the rat adenohypophysis by Jard, S, Gaillard, R C, Guillon, G, Marie, J, Schoenenberg, P, Muller, A F, Manning, M, Sawyer, W H

“…The ligand specificity of rat adenohypophyseal vasopressin receptors was directly compared to that of peripheral receptors of the V1 and V2 types. For this…”
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Close association of the alpha subunits of Gq and G11 G proteins with actin filaments in WRK1 cells: relation to G protein-mediated phospholipase C activation by Ibarrondo, J, Joubert, D, Dufour, M N, Cohen-Solal, A, Homburger, V, Jard, S, Guillon, G

“…A selective polyclonal antibody directed toward the C-terminal decapeptide common to the alpha subunits of Gq and G11 G proteins (G alpha q/G alpha 11) was…”
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Vasopressin: mechanisms of receptor activation by Jard, S

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Vasopressin and angiotensin II receptors in rat aortic smooth muscle cells in culture by Penit, J, Faure, M, Jard, S

“…Rat aortic smooth muscle cells were isolated and maintained in primary culture. After 2-3 days, cells recovered their contractile phenotype and could be…”
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A radioiodinated linear vasopressin antagonist: A ligand with high affinity and specificity for V1a receptors by Schmidt, A., Audigier, S., Barberis, C., Jard, S., Manning, M., Kolodziejczyk, A.S., Sawyer, W.H.

“…A linear vasopressin antagonist, Phaa‐D‐Tyr(Me)‐Phe‐Gin‐Asn‐Arg‐Pro‐Arg‐Tyr‐NH2 (Linear AVP Antag) (Phaa = Phenylacetyl), was monoiodinated at the phenyl…”
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Vasopressin receptors from cultured mesangial cells resemble V1a type by Jard, S, Lombard, C, Marie, J, Devilliers, G

“…Mesangial cells respond to vasopressin by contraction and increased prostaglandin production. The purpose of the present study is to characterize vasopressin…”
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Functional Architecture of Vasopressin/Oxytocin Receptors by Hibert, M., Hoflack, J., Trumpp-Kallmeyer, S., Mouillac, B., Chini, B., Mahea, E., Cotte, N., Jard, S., Manning, M., Barberis, C.

“…Abstract Three-dimensional models of G protein-coupled receptors (GPCR) have been defined using most experimental data available and protein modeling…”
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Oxytocin receptors in rat kidney during development by Schmidt, A, Jard, S, Dreifuss, J J, Tribollet, E

“…The development and characteristics of oxytocin (OT) receptors in the rat kidney were studied by light-microscopic autoradiography and on membrane preparations…”
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Angiotensin II and alpha-adrenergic agonists inhibit rat liver adenylate cyclase by Jard, S, Cantau, B, Jakobs, K H

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Deglycosylation and fragmentation of purified rat liver angiotensin II receptor : application to the mapping of hormone-binding domains by DESARNAUD, F, MARIE, J, LOMBARD, C, LARGUIER, R, SEYER, R, LORCA, T, JARD, S, BONNAFOUS, J.-C

“…We report new structural data about the rat liver angiotensin II receptor, which belongs to the AT1 subclass. This receptor has been purified at analytical or…”
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Identification of a Single Residue Responsible for Agonist Selectivity in the Oxytocin-Vasopressin Receptors by CHINI, B., MOUILLAC, B., ALA, Y., BALESTRE, M. N., TRUMPP-KALLMEYER, S., HOFLACK, J., ELANDS, J., HIBERT, M., MANNING, M., JARD, S., BARBERIS, C.

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