Search Results - "Illyes, Eszter"

Discovery of N-[4-(Quinolin-4-yloxy)phenyl]benzenesulfonamides as Novel AXL Kinase Inhibitors by Szabadkai, István, Torka, Robert, Garamvölgyi, Rita, Baska, Ferenc, Gyulavári, Pál, Boros, Sándor, Illyés, Eszter, Choidas, Axel, Ullrich, Axel, Őrfi, László

“…The overexpression of AXL kinase has been described in many types of cancer. Due to its role in proliferation, survival, migration, and resistance, AXL…”
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Synthesis and Structure–Activity relationship of 1-(5-isoquinolinesulfonyl)piperazine analogues as inhibitors of Mycobacterium tuberculosis IMPDH by Singh, Vinayak, Pacitto, Angela, Donini, Stefano, Ferraris, Davide M., Boros, Sándor, Illyés, Eszter, Szokol, Bálint, Rizzi, Menico, Blundell, Tom L., Ascher, David B., Pato, Janos, Mizrahi, Valerie

“…Tuberculosis (TB) is a major infectious disease associated increasingly with drug resistance. Thus, new anti-tubercular agents with novel mechanisms of action…”
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Design and synthesis of new imidazo[1,2-a]pyridine and imidazo[1,2-a]pyrazine derivatives with antiproliferative activity against melanoma cells by Garamvölgyi, Rita, Dobos, Judit, Sipos, Anna, Boros, Sándor, Illyés, Eszter, Baska, Ferenc, Kékesi, László, Szabadkai, István, Szántai-Kis, Csaba, Kéri, György, Őrfi, László

“…Melanoma is an aggressive form of skin cancer and it is generally associated with poor prognosis in patients with late-stage disease. Due to the increasing…”
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Hungarian landscape types: classification of landscapes based on the relative cover of (semi-) natural habitats by Bölöni, János, Botta-Dukát, Zoltán, Illyés, Eszter, Molnár, Zsolt

“…Aim: This paper introduces a new method for vegetation-based landscape classification. As a case study, we present the landscape classification of Hungary with…”
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Effect of SXWS/WSXWS peptides on chemotaxis and adhesion of the macrophage-like cell line J774 by Szabó, Rita, Láng, Orsolya, Láng, Júlia, Illyés, Eszter, Kőhidai, László, Hudecz, Ferenc

“…WSXWS motif is a conserved amino acid sequence that is present in type I cytokine receptors. This motif that can be found both in the ligand binding chains and…”
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N-terminal acylation of the SV40 nuclear localization signal peptide enhances its oligonucleotide binding and membrane translocation efficiencies by Laczkó, Ilona, Váró, György, Bottka, Sándor, Bálint, Zoltán, Illyés, Eszter, Vass, Elemér, Bertrand, Jean-Remy, Malvy, Claude, Hollósi, Miklós

“…Octanoyl and palmitoyl groups were coupled to the N-terminus of an analog of the SV40 nuclear localization signal peptide, SV 126–133(Ser 128), to study the…”
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Photochemical and Structural Studies on Cyclic Peptide Models by Nagy, Tamás Milán, Knapp, Krisztina, Illyés, Eszter, Timári, István, Schlosser, Gitta, Csík, Gabriella, Borics, Attila, Majer, Zsuzsa, Kövér, Katalin E

“…Ultra-violet (UV) irradiation has a significant impact on the structure and function of proteins that is supposed to be in relationship with the…”
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Novel compounds with potent CDK9 inhibitory activity for the treatment of myeloma by Czudor, Zsófia, Balogh, Mária, Bánhegyi, Péter, Boros, Sándor, Breza, Nóra, Dobos, Judit, Fábián, Márk, Horváth, Zoltán, Illyés, Eszter, Markó, Péter, Sipos, Anna, Szántai-Kis, Csaba, Szokol, Bálint, Őrfi, László

“…[Display omitted] Cyclin-dependent kinases (CDKs) and Polo-like kinases (PLKs) play key role in the regulation of the cell cycle. The aim of our study was…”
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Synthesis and characterization of amino acid substituted sunitinib analogues for the treatment of AML by Nemes, Zoltán, Takács-Novák, Krisztina, Völgyi, Gergely, Valko, Klara, Béni, Szabolcs, Horváth, Zoltán, Szokol, Bálint, Breza, Nóra, Dobos, Judit, Szántai-Kis, Csaba, Illyés, Eszter, Boros, Sándor, Kok, Robbert Jan, Őrfi, László

“…[Display omitted] •62 amino acid substituted sunitinib analogues were synthesized, inhibiting FLT3-ITD kinase and AML cell line.•Physical-chemical properties…”
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Discovery and optimization of novel benzothiophene-3-carboxamides as highly potent inhibitors of Aurora kinases A and B by Gyulavári, Pál, Szokol, Bálint, Szabadkai, István, Brauswetter, Diána, Bánhegyi, Péter, Varga, Attila, Markó, Péter, Boros, Sándor, Illyés, Eszter, Szántai-Kis, Csaba, Krekó, Marcell, Czudor, Zsófia, Őrfi, László

“…[Display omitted] •Two lead compounds were tested against kinase selectivity panel including 35 kinases.•The most effective compounds tested against two cancer…”
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Semi-dry grasslands along a climatic gradient across Central Europe: Vegetation classification with validation by Illyés, Eszter, Chytrý, Milan, Botta-Dukát, Zoltán, Jandt, Ute, Škodová, Iveta, Janišová, Monika, Willner, Wolfgang, Hájek, Ondřej

“…Question: What is the variation in species composition of Central European semi-dry grasslands? Can we apply a training-and-test validation approach for…”
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Anti-influenza virus activity and structure–activity relationship of aglycoristocetin derivatives with cyclobutenedione carrying hydrophobic chains by Naesens, Lieve, Vanderlinden, Evelien, Rőth, Erzsébet, Jekő, József, Andrei, Graciela, Snoeck, Robert, Pannecouque, Christophe, Illyés, Eszter, Batta, Gyula, Herczegh, Pál, Sztaricskai, Ferenc

“…Previous studies have demonstrated that glycopeptide compounds carrying hydrophobic substituents can have favorable pharmacological (i.e. antibacterial and…”
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Heteroclitic recognition of combinatorial TX1TX2T peptide mixtures by mucin-2 protein specific monoclonal antibody by Windberg, Emôke, Uray, Katalin, Illyés, Eszter, Skribanek, Zsolt, Price, Michael R., Sebestyén, Ferenc, Hudecz, Ferenc

“…The mucin‐2 (MUC2) glycoprotein secreted by the epithelial cells of human colon may be abnormally under‐glycosylated in the case of cancer. Monoclonal antibody…”
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The role of nanoparticle concentration-dependent induction of cellular stress in the internalization of non-toxic cationic magnetoliposomes by Soenen, Stefaan J.H, Illyes, Eszter, Vercauteren, Dries, Braeckmans, Kevin, Majer, Zsuzsa, De Smedt, Stefaan C, De Cuyper, Marcel

“…Abstract Magnetoliposomes (MLs), built up of ultrasmall iron oxide cores each individually surrounded by a lipid bilayer, have emerged as highly biocompatible…”
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Synthesis of oligopeptides with the sequence SXWS and their chemotactic effects on a ciliated protozoan Tetrahymena pyriformis by Illyés, Eszter, Hudecz, Ferenc, Köhidai, László, Láng, Orsolya, Szabó, Pál, Sebestyén, Ferenc

“…In this paper, the solid phase synthesis and chemical characterization of members of an SXWS sub‐library (SAWS, SDWS and SKWS) as well as the comparison of…”
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Two Functional Active Conformations of the Integrin α2β1, Depending on Activation Condition and Cell Type by Van de Walle, Gerlinde R., Vanhoorelbeke, Karen, Majer, Zsuzsa, Illyés, Eszter, Baert, Johan, Pareyn, Inge, Deckmyn, Hans

“…For several integrins, the existence of multiple conformational states has been studied intensively. For the integrin α2β1, a major collagen receptor on…”
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A Grid-Based, Satellite-Image Supported, Multi-Attributed Vegetation Mapping Method (MÉTA) by Molnár, Zsolt, Bartha, Sándor, Seregélyes, Tibor, Illyés, Eszter, Botta-Dukát, Zoltán, Tímár, Gábor, Horváth, Ferenc, Révész, András, Kun, András, Bölöni, János, Biró, Marianna, Bodonczi, László, József, Áron Deák, Fogarasi, Péter, Horváth, András, Isépy, István, Karas, László, Kecskés, Ferenc, Molnár, Csaba, Ajkai, Adrienne Ortmann-né, Rév, Szilvia

“…In this paper we present the main characteristics of a new, grid-based, landscape-ecology-oriented, satellite-image supported, field vegetation mapping method,…”
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Synthesis and Studies on Cell-Penetrating Peptides by Bertrand, Jean-Remi, Malvy, Claude, Auguste, Tiphanie, Tóth, Gábor K, Kiss-Ivánkovits, Orsolya, Illyés, Eszter, Hollósi, Miklós, Bottka, Sándor, Laczkó, Ilona

“…The ability of different synthetic cell penetrating peptides, as Antennapedia (wild and Phe6 mutated penetratins), flock house virus, and integrin peptides to…”
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Fluorescence contributions of the individual Trp residues in goat α-lactalbumin by Vanhooren, Ann, Illyes, Eszter, Majer, Zsuzsa, Hanssens, Ignace

“…Goat α-lactalbumin (GLA) contains four tryptophan (Trp) residues. In order to obtain information on the fluorescence contribution of the individual Trp…”
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Coloured peptides: synthesis, properties and use in preparation of peptide sub-library kits by Sebestyén, Ferenc, Szendrei, Györgyi, Mák, Marianna, Dóda, Margit, Illyés, Eszter, Szókán, Gyula, Kindla, Krisztina, Rapp, Wolfgang, Szegő, Péter, Câmpian, Eugen, Furka, Árpád

“…Several methods were developed for the solid‐phase synthesis (SPPS) of coloured peptides and peptide libraries. At first a bifunctional red compound,…”
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