Search Results - "Homon, Anton A."

Structure-based Design of Novel Hepatitis B Virus Capsid Assembly Modulators by Detta, Elena, Corcuera, Angelica, Urban, Andreas, Goldner, Thomas, Bonsmann, Susanne, Engel, Florian, May, Marina M., Buschmann, Helmut, Fianchini, Mauro, Alza, Esther, Pericàs, Miquel A., Pushkarev, Pavel A., Varenyk, Anatolii O., Yakovyuk, Taras Y., Homon, Anton A., Sokoliuk, Pavlo A., Smaliy, Radomyr, Donald, Alastair

“…[Display omitted] •Capsid Assembly Modulators are promising agents for curing chronic HBV infection.•Target-based in silico screening study leads to the…”
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Synthesis of 3‐Azabicyclo[3.2.0]heptane‐Derived Building Blocks via [3+2] Cycloaddition by Homon, Anton A., Hryshchuk, Oleksandr V., Trofymchuk, Serhii, Michurin, Oleg, Kuchkovska, Yuliya, Radchenko, Dmytro S., Grygorenko, Oleksandr O.

“…An efficient approach to synthesis of various substituted 3‐azabicyclo[3.2.0]heptane‐derived building blocks based on [3+2] cycloaddition of…”
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Synthesis of 1,3-bifunctional cyclobutane derivatives with α-CHF2/CF3 group – advanced building blocks for medicinal chemistry by Homon, Anton A., Shynder, Lada V., Demchuk, Oleksandr P., Hryshchuk, Oleksandr V., Kondratov, Ivan S., Gerus, Igor I., Grygorenko, Oleksandr O.

“…•Synthesis of α-CF3/CHF2-substituted 1,3-bifunctional cyclobutanes is described.•Conformationally restricted analogs of γ-amino- and γ-hydroxybutyric acids are…”
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4‐(Di‐/Trifluoromethyl)‐2‐heterabicyclo[2.1.1]hexanes: Advanced Fluorinated Phenyl Isosteres and Proline analogues by Homon, Anton A., Hryshchuk, Oleksandr V., Mykhailenko, Olha V., Vashchenko, Bohdan V., Melnykov, Kostiantyn P., Michurin, Oleg M., Daniliuc, Constantin G., Gerus, Igor I., Kovtunenko, Volodymyr O., Kondratov, Ivan S., Grygorenko, Oleksandr O.

“…A gram‐scale synthesis, physico‐chemical characterization, and lead‐likeness assessment of 4‐di/trifluoromethyl‐2‐heterabicyclo[2.1.1]hexanes as fluorinated…”
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4‐(Di‐/Trifluoromethyl)‐2‐heterabicyclohexanes: Advanced Fluorinated Phenyl Isosteres and Proline analogues by Homon, Anton A, Hryshchuk, Oleksandr V, Mykhailenko, Olha V, Vashchenko, Bohdan V, Melnykov, Kostiantyn P, Michurin, Oleg M, Daniliuc, Constantin G, Gerus, Igor I, Kovtunenko, Volodymyr O, Kondratov, Ivan S, Grygorenko, Oleksandr O

“…A gram‐scale synthesis, physico‐chemical characterization, and lead‐likeness assessment of 4‐di/trifluoromethyl‐2‐heterabicyclo[2.1.1]hexanes as fluorinated…”
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