Search Results - "Heusler, P"

Signal transduction and functional selectivity of F15599, a preferential post‐synaptic 5‐HT1A receptor agonist by Newman‐Tancredi, A, Martel, J‐C, Assié, M‐B, Buritova, J, Lauressergues, E, Cosi, C, Heusler, P, Bruins Slot, L, Colpaert, FC, Vacher, B, Cussac, D

“…Background and purpose:  Activation of post‐synaptic 5‐HT1A receptors may provide enhanced therapy against depression. We describe the signal transduction…”
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Levomilnacipran (F2695), a norepinephrine-preferring SNRI: Profile in vitro and in models of depression and anxiety by Auclair, A.L., Martel, J.C., Assié, M.B., Bardin, L., Heusler, P., Cussac, D., Marien, M., Newman-Tancredi, A., O'Connor, J.A., Depoortère, R.

“…Levomilnacipran (LVM; F2695) is the more active enantiomer of the serotonin/norepinephrine (5-HT/NE) reuptake inhibitor (SNRI) milnacipran and is currently…”
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In vitro profile of the new antipsychotic, F17464, at recombinant human neurotransmitter receptors by Heusler, P, Martel, J.C, Gatti-McArthur, S

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Signal transduction and functional selectivity of F15599, a preferential post‐synaptic 5‐HT 1A receptor agonist by Newman‐Tancredi, A, Martel, J‐C, Assié, M‐B, Buritova, J, Lauressergues, E, Cosi, C, Heusler, P, Bruins Slot, L, Colpaert, FC, Vacher, B, Cussac, D

“…Background and purpose:  Activation of post‐synaptic 5‐HT 1A receptors may provide enhanced therapy against depression. We describe the signal transduction…”
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P.2.d.013 F15599, a post-synaptic cortical preferential 5-HT1A agonist: I) functionally-selective signal transduction profile by Newman-Tancredi, A, Martel, J.C, Buritova, J, Lauressergues, E, Assie, M.B, Slot, L. Bruins, Cosi, C, Heusler, P, Cussac, D

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A repetitive intracortical microstimulation pattern induces long-lasting synaptic depression in brain slices of the rat primary somatosensory cortex by HEUSLER, Peter, CEBULLA, Bernhard, BOEHMER, Gerd, DINSE, Hubert R

“…Repetitive intracortical microstimulation (ICMS) applied to the rat primary somatosensory cortex (SI) in vivo was reported to induce reorganization of…”
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P.3.a.006 - In vitro profile of the new antipsychotic, F17464, at recombinant human neurotransmitter receptors by Heusler, P., Martel, J.C., Gatti-McArthur, S.

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F17464 a new antipsychotic with preferential D3 antagonist, 5-HT1A partial agonist properties. Neurochemical studies by Cosi, C., N’Guyen, V., Consul-Denjean, N., Auclair, A., Heusler, P., Martel, J.C., Leriche, L., Sokoloff, P., Gatti-McArthur, S.

“…F17464 is a new dopamine receptor antagonist that recently demonstrated antipsychotic activity in a proof of concept study in schizophrenic patients under…”
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Platelet-activating factor contributes to the induction of long-term potentiation in the rat somatosensory cortex in vitro by Heusler, Peter, Boehmer, Gerd

“…Abstract The contribution of platelet-activating factor (PAF) to the induction of neocortical LTP was examined in rat brain slices containing the primary…”
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The superoxide anion is involved in the induction of long-term potentiation in the rat somatosensory cortex in vitro by Heusler, Peter, Boehmer, Gerd

“…The involvement of the superoxide anion (O 2 −) in the induction of neocortical long-term potentiation (LTP) was examined in rat brain slices containing the…”
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Differential ion current activation by human 5-HT1A receptors in Xenopus oocytes: Evidence for agonist-directed trafficking of receptor signalling by Heusler, Peter, Pauwels, Petrus J., Wurch, Thierry, Newman-Tancredi, Adrian, Tytgat, Jan, Colpaert, Francis C., Cussac, Didier

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P.3.d.004 F15063, a novel antipsychotic with D2/D3 antagonist, 5-HT1A agonist and D4 partial agonist properties: I. Receptor affinity and efficacy in vitro and activity in neurochemical and neuroendocrine tests in rodents by Newman-Tancredi, A., Assié, M.B., Martel, J.C., Cosi, C., Heusler, P., Bruins Slot, L., Carilla-Durand, E., Cussac, D.

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