Search Results - "Hese, Shrikant V."

Chloroxylon swietenia (Roxb.) DC induces cell death and apoptosis by down‐regulating the NF‐κB pathway in MCF‐7 breast cancer cells: In vitro and in vivo investigations by Kamble, Sonali S., Choudhari, Jasoda, Nimma, Ramakrishna, Kumar, Totakura Venkata Santosh, Patil, Kapil K., Hese, Shrikant V., Dawane, Bhaskar S., Gacche, Rajesh N.

“…Background Natural products with targeted bioactivity have gained major attention in the field of cancer research owing to emerging anti‐cancer drug resistance…”
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Synthesis and in silico investigation of thiazoles bearing pyrazoles derivatives as anti-inflammatory agents by Kamble, Rahul D., Meshram, Rohan J., Hese, Shrikant V., More, Rahul A., Kamble, Sonali S., Gacche, Rajesh N., Dawane, Bhaskar S.

“…[Display omitted] •Efficient one-pot synthesis of thiazole bearing pyrazole derivatives.•Compound showing selective COX-II inhibition.•Molecular docking is in…”
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Design, synthesis and in silico study of pyridine based 1,3,4-oxadiazole embedded hydrazinecarbothioamide derivatives as potent anti-tubercular agent by Ambhore, Ajay N., Kamble, Sonali S., Kadam, Shuddhodan N., Kamble, Rahul D., Hebade, Madhav J., Hese, Shrikant V., Gaikwad, Milind V., Meshram, Rohan J., Gacche, Rajesh N., Dawane, Bhaskar S.

“…[Display omitted] •Anti-tubercular study of the newly synthesized compounds showed promising results.•Hemolytic Study of newly synthesized compounds.•Molecular…”
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DTP/SiO2 Assisted Synthesis of New Benzimidazole-Thiazole Conjugates Targeting Antitubercular and Antioxidant Activities by Hebade, Madhav J., Dhumal, Sambhaji T., Kamble, Sonali S., Deshmukh, Tejshri R., Khedkar, Vijay M., Hese, Shrikant V., Gacche, Rajesh N., Dawane, Bhaskar S.

“…A series of new substituted benzimidazole-thiazoles (9a-l) have been designed and synthesized using 2-aminothiazole as a starting material by using molecular…”
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Synthesis and evaluation of N-(4-(substituted)-3-(trifluoromethyl) phenyl) isobutyramides and their N-ethyl analogous as anticancer, anti-angiogenic & antioxidant agents: In vitro and in silico analysis by Sawant, Ajay S., Kamble, Sonali S., Pisal, Parshuram M., Sawant, Sanjay S., Hese, Shrikant V., Bagul, Kamini T, Pinjari, Rahul V., Kamble, Vinod T., Meshram, Rohan J., Gacche, Rajesh N.

“…[Display omitted] •Novel flutamide derivatives were synthesized.•Biological assessment of all compounds was done in the form of cytotoxic, anti-angiogenic and…”
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Antidiabetic and allied biochemical roles of new chromeno-pyrano pyrimidine compounds: synthesis, in vitro and in silico analysis by Hese, Shrikant V., Meshram, Rohan J., Kamble, Rahul D., Mogle, Pratima P., Patil, Kapil K., Kamble, Sonali S., Gacche, Rajesh N., Dawane, Bhaskar S.

“…Diabetes is embracing the human population in logarithmic fashion both in developed as well as developing countries. Aldose reductase is one of the important…”
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Green synthesis and in silico investigation of dihydro-2H-benzo[1,3]oxazine derivatives as inhibitors of Mycobacterium tuberculosis by Kamble, Rahul D., Hese, Shrikant V., Meshram, Rohan J., Kote, Jivan R., Gacche, Rajesh N., Dawane, Bhaskar S.

“…In the midst of increasing multidrug resistance and the growing incidence of infections of Mycobacterium tuberculosis , there is compelling evidence for the…”
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A rapid, mild, and efficient method for C-5 iodination/thiocyanation of 2-aminothiazoles by Hebade, Madhav J., Kamble, Rahul D., Hese, Shrikant V., Mogle, Pratima P., Ambhore, Ajay N., Kadam, Shuddhodan N., Dawane, Bhaskar S.

“…An efficient, green, rapid multitasking protocol for the selective C-5 substitution of 2-aminothiazole using iodic acid and aqueous PEG-400 was developed. The…”
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DTP/SiO 2 Assisted Synthesis of New Benzimidazole-Thiazole Conjugates Targeting Antitubercular and Antioxidant Activities by Hebade, Madhav J., Dhumal, Sambhaji T., Kamble, Sonali S., Deshmukh, Tejshri R., Khedkar, Vijay M., Hese, Shrikant V., Gacche, Rajesh N., Dawane, Bhaskar S.

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An efficient synthesis of isoxazoline libraries of thiophene analogs and its antimycobacterial investigation by Mandawad, Gajanan G., Kamble, Rahul D., Hese, Shrikant V., More, Rahul A., Gacche, Rajesh N., Kodam, Kisan M., Dawane, Bhaskar S.

“…Synthesis of novel thiophene substituted isoxazoline libraries is currently of high interest. Here, we have reported detailed syntheses of…”
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Bleaching earth clay (pH 12.5)/PEG-400: an efficient recyclable catalytic system for synthesis of 5,6,7,8-tetrahydroquinoline-3-carbonitrile derivatives by Mogle, Pratima P., Kamble, Rahul D., Hese, Shrikant V., Dawane, Bhaskar S.

“…A green, efficient, and simple method for synthesis of 5,6,7,8-tetrahydroquinoline-3-carbonitrile derivatives via one-pot three-component condensation of…”
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Green method for synthesis of 3-[2-(substituted-phenyl)-2-oxo ethylidene]-1,3-dihydro-indol-2-one and their in vitro antimicrobial activity by Acharya, Ashok P., Kamble, Rahul D., Patil, Snehalkumar D., Hese, Shrikant V., Yemul, Omprakash S., Dawane, Bhaskar S.

“…The cross-aldol condensation between isatin ( I ) and substituted acetophenone ( IIa – e ) in one-pot reaction afforded…”
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Bleaching earth clay pH 12.5/PEG-400 catalytic system for synthesis of some novel α, β-unsaturated ketones (chalcones) by Gaikwad, Milind V., Kamble, Rahul D., Hese, Shrikant V., Acharya, Ashok P., Mogle, Pratima P., Kadam, Shuddhodan N., Dawane, Bhaskar S.

“…We report bleaching earth clay pH 12.5/PEG-400 as an efficient catalytic system for preparation of α,β-unsaturated ketones (chalcones). The method presents one…”
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Green approach towards synthesis of substituted pyrazole-1,4-dihydro,9-oxa,1,2,6,8-tetrazacyclopentano[b]naphthalene-5-one derivatives as antimycobacterial agents by Chobe, Santosh S., Kamble, Rahul D., Patil, Snehalkumar D., Acharya, Ashok P., Hese, Shrikant V., Yemul, Omprakash S., Dawane, Bhaskar S.

“…In the present communication, a simple and efficient synthesis of some new Pyrano-[2,3- c ]-pyrazoles derivatives are described by the one-pot condensation of…”
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