Search Results - "Hao, Zesheng"

Design, synthesis and fungicidal activity of pyrazole–thiazole carboxamide derivatives by Hao, Zesheng, Yu, Bin, Gao, Wei, Chen, Haoyin, Yang, Dongyan, Lv, You, Zhang, Yue, Chen, Lei, Fan, Zhijin

“…Twenty-one novel pyrazole–thiazole carboxamide derivatives were rationally designed and synthesized. Bioassay results indicated that 6d (EC 50  = 5.11 μg/mL)…”
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Design, synthesis and fungicidal activity of 3,4-dichloroisothiazolocoumarin-containing strobilurins by Lv, You, Li, Kun, Gao, Wei, Hao, Zesheng, Wang, Weibo, Liu, Xiaoyu, Tang, Liangfu, Fan, Zhijin

“…Twenty-one novel 3,4-dichloroisothiazolocoumarin-containing strobilurins were rationally designed and synthesized. Preliminary bioassay showed that compounds…”
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Thiazolylhydrazone dervatives as inhibitors for insect N-acetyl-β-d-hexosaminidase and chitinase by Yang, Huibin, Qi, Huitang, Hao, Zesheng, Shao, Xusheng, Liu, Tian, Yang, Qing, Qian, Xuhong

“…Here, a series of thiazolylhydrazones I and II were designed, synthesised and evaluated as competitive inhibitors of OfHex1and OfChi-h. Derivatives I-3d and…”
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Design, synthesis and antifungal activity of (E)-3-acyl-5-(methoxyimino)-1,5-dihydrobenzo[e][1,2]oxazepin-4(3H)-one analogues by Yang, Dongyan, Wang, Haixia, Fan, Zhijin, Li, Zhengming, Zhou, Shuang, Hao, Zesheng, Lv, You, Kalinina, Tatiana A., Glukhareva, Tatiana V.

“…Nitrogen- or oxygen-containing organic compounds which have significant antifungal activity, twenty one novel nitrogen or oxygen-containing ( E…”
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Design, Synthesis, and Evaluation of the Antifungal Activity of Novel Pyrazole–Thiazole Carboxamides as Succinate Dehydrogenase Inhibitors by Yu, Bin, Zhou, Shuang, Cao, Lixin, Hao, Zesheng, Yang, Dongyan, Guo, Xiaofeng, Zhang, Nailou, Bakulev, Vasiliy A, Fan, Zhijin

“…Succinate dehydrogenase (SDH) is regarded as a promising target for fungicide discovery. To continue our ongoing studies on the discovery of novel SDH…”
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Design, synthesis and biological evaluation of pyrazole-aromatic containing carboxamides as potent SDH inhibitors by Yu, Bin, Zhao, Bin, Hao, Zesheng, Chen, Lei, Cao, Lixin, Guo, Xiaofeng, Zhang, Nailou, Yang, Dongyan, Tang, Liangfu, Fan, Zhijin

“…To continue our ongoing studies on discovery of new potent antifungal leads, 43 novel pyrazole-aromatic containing carboxamides were rationally designed and…”
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Discovery of a polysubstituted phenyl containing novel N-phenylpyrazole scaffold as potent ryanodine receptor activator by Liu, Jingbo, Li, Fengyun, Hao, Zesheng, Wang, Yuanhong, Hua, Xuewen, Li, Yuxin, Li, Zhengming

“…[Display omitted] •Novel N-phenylpyrazole derivatives containing a polysubstituted phenyl ring scaffold 7a-p were designed and synthesized.•LC50 values of 7f…”
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Design, Synthesis, and Evaluation of Novel Isothiazole-Purines as a Pyruvate Kinase-Based Fungicidal Lead Compound by Wang, Weibo, Li, Zhixinyi, Gao, Wei, Liu, Xiaoyu, Lv, You, Hao, Zesheng, Tang, Liangfu, Li, Kun, Zhao, Bin, Fan, Zhijin

“…Target identification is one of the most important bases for novel pesticide development; pyruvate kinase (PK) was discovered as a potent fungicide target in…”
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Bioactivity-Guided Synthesis Accelerates the Discovery of Evodiamine Derivatives as Potent Insecticide Candidates by Liu, Jingbo, Shi, Yabing, Tian, Zhicheng, Li, Fengyun, Hao, Zesheng, Wen, Wen, Zhang, Li, Wang, Yuanhong, Li, Yuxin, Fan, Zhijin

“…Pests threaten worldwide food security by decreasing crop yields and damaging their quality. Natural product-based molecular design and structural optimization…”
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Novel Evodiamine-Based Sulfonamide Derivatives as Potent Insecticide Candidates Targeting Insect Ryanodine Receptors by Liu, Jingbo, Guo, Bingyan, Zhong, Siying, Shi, Yabing, Li, Zhengping, Yu, Zhenwu, Hao, Zesheng, Zhang, Li, Li, Fengyun, Wang, Yuanhong, Li, Yuxin

“…Pests represent an important impediment to efficient agricultural production and pose a threat to global food security. On the basis of our prior research…”
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Design and synthesis of thiazolylhydrazone derivatives as inhibitors of chitinolytic N-acetyl-β-d-hexosaminidase by Yang, Huibin, Liu, Tian, Qi, Huitang, Huang, Zhisong, Hao, Zesheng, Ying, Junwu, Yang, Qing, Qian, Xuhong

“…[Display omitted] N-acetyl-β-d-hexosaminidase (Hex) is potential target for pesticide design. Here, a series of thiazolylhydrazone derivatives were designed,…”
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Design, Synthesis, and Evaluation of Fungicidal Activity of Novel Pyrazole‐Containing Strobilurin Derivatives by Hao, Zesheng, Wang, Weibo, Yu, Bin, Qi, Xin, Lv, You, Liu, Xiaoyu, Chen, Haoyin, Kalinina, Tatiana A., Glukhareva, Tatiana V., Fan, Zhijin

“…Main observation and conclusion In searching for novel fungicidal leads, a series of pyrazole‐containing strobilurins were rationally designed, synthesized and…”
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气质、父母教养方式与幼儿心理韧性的关系 by NIU, Yubai, ZHANG, Lingyan, HAO, Zesheng, JI, Yuzhu

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Relationship between temperament, parenting style and resilience of children aged 3-5 years by Niu, Yubai, Zhang, Lingyan, Hao, Zesheng, Ji, Yuzhu

“…To investigate the developmental characteristics of resilience in children aged 3-5, and to explore the relationship between temperament, parenting style and…”
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气质、父母教养方式与幼儿心理韧性的关系 by 牛玉柏, 张凌燕, 郝泽生, 季雨竹

“…B844; 目的:考察3～5岁幼儿心理韧性的发展特点并探讨气质、父母教养方式与幼儿心理韧性之间的关系,检验父母教养方式的中介作用.方法:选取杭州市570名幼儿为被试对象,由幼儿教师完成Devereux幼儿心理韧性量表评定,由幼儿父母完成气质问卷和教养方式问卷的评定.采用AMOS…”
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