Search Results - "HIBERT, M."

Squaraine as a bright, stable and environment-sensitive far-red label for receptor-specific cellular imaging by Karpenko, I A, Klymchenko, A S, Gioria, S, Kreder, R, Shulov, I, Villa, P, Mély, Y, Hibert, M, Bonnet, D

“…Herein, we show that a far-red arylidene-squaraine dye is stable against nucleophiles, in contrast to arene-squaraines. Owing to the fluorescence enhancement…”
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Alginate Encapsulant Incorporating CXCL12 Supports Long‐Term Allo‐ and Xenoislet Transplantation Without Systemic Immune Suppression by Chen, T., Yuan, J., Duncanson, S., Hibert, M. L., Kodish, B. C., Mylavaganam, G., Maker, M., Li, H., Sremac, M., Santosuosso, M., Forbes, B., Kashiwagi, S., Cao, J., Lei, J., Thomas, M., Hartono, C., Sachs, D., Markmann, J., Sambanis, A., Poznansky, M. C.

“…Islet transplantation represents a potentially curative approach for individuals with Type I Diabetes. The requirement for systemic immune suppression to…”
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Altered Blood Flow in the Ophthalmic and Internal Carotid Arteries in Patients with Age-Related Macular Degeneration Measured Using Noncontrast MR Angiography at 7T by Hibert, M L, Chen, Y I, Ohringer, N, Feuer, W J, Waheed, N K, Heier, J S, Calhoun, M W, Rosenfeld, P J, Polimeni, J R

“…Age-related macular degeneration is associated with reduced perfusion of the eye; however, the role of altered blood flow in the upstream ophthalmic or…”
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Key Amino Acids Located within the Transmembrane Domains 5 and 7 Account for the Pharmacological Specificity of the Human V1b Vasopressin Receptor by Derick, S, Pena, A, Durroux, T, Wagnon, J, Serradeil-Le Gal, C, Hibert, M, Rognan, D, Guillon, G

“…In mammals, the vasopressin V1b receptor (V1b-R) is known to regulate ACTH secretion and, more recently, stress and anxiety. The characterization of the…”
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On the Use of Nonfluorescent Dye Labeled Ligands in FRET-Based Receptor Binding Studies by Tahtaoui, Chouaib, Guillier, Fabrice, Klotz, Philippe, Galzi, Jean-Luc, Hibert, Marcel, Ilien, Brigitte

“…The efficiency of fluorescence resonance energy transfer (FRET) is dependent upon donor−acceptor proximity and spectral overlap, whether the acceptor partner…”
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Tyr115 is the key residue for determining agonist selectivity in the V1a vasopressin receptor by Chini, B., Mouillac, B., Ala, Y., Balestre, M.N., Trumpp‐Kallmeyer, S., Hoflack, J., Elands, J., Hibert, M., Manning, M., Jard, S.

“…Using a three‐dimensional model of G protein‐coupled receptors (GPCR), we have previously succeeded in docking the neurohypophysial hormone…”
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This is not a G protein-coupled receptor by Hibert, M F, Trumpp-Kallmeyer, S, Hoflack, J, Bruinvels, A

“…On his canvas entitled 'La trahison des Images' ('The Perfidy of Images'), René Magritte painted a tobacco pipe in a very realistic manner and added the words:…”
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Tyr115 is the key residue for determining agonist selectivity in the V1a vasopressin receptor by Chini, B., Mouillac, B., Ala, Y., Balestre, M.N., Trumpp-Kallmeyer, S., Hoflack, J., Elands, J., Hibert, M., Manning, M., Jard, S.

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Characterization of MDL 73005EF as a 5‐HT1A selective ligand and its effects in animal models of anxiety: comparison with buspirone, 8‐OH‐DPAT and diazepam by Moser, P.C., Tricklebank, M.D., Middlemiss, D.N., Mir, A.K., Hibert, M.F., Fozard, J.R.

“…1 With radioligand binding techniques, MDL 73005 EF (8‐[2‐(2,3‐dihydro‐1,4‐benzodioxin‐2‐yl‐methylamino)ethyl]‐8‐azaspiro[4,5]decane‐7,9‐dione methyl…”
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Three-dimensional models of neurotransmitter G-binding protein-coupled receptors by Hibert, M F, Trumpp-Kallmeyer, S, Bruinvels, A, Hoflack, J

“…Graphics computer-generated three-dimensional models of all G-binding protein-coupled receptors were built and analyzed. These models were defined using…”
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Fluorogenic Squaraine Dimers with Polarity-Sensitive Folding As Bright Far-Red Probes for Background-Free Bioimaging by Karpenko, Iuliia A, Collot, Mayeul, Richert, Ludovic, Valencia, Christel, Villa, Pascal, Mély, Yves, Hibert, Marcel, Bonnet, Dominique, Klymchenko, Andrey S

“…Polarity-sensitive fluorogenic dyes raised considerable attention because they can turn on their fluorescence after binding to biological targets, allowing…”
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Graphics computer-aided receptor mapping as a predictive tool for drug design: development of potent, selective, and stereospecific ligands for the 5-HT1A receptor by Hibert, Marcel F, Gittos, Maurice W, Middlemiss, Derek N, Mir, Anis K, Fozard, John R

“…A conformational study of four 5-HT1A (serotonin) receptor ligands ((R-(-)-methiothepin, spiperone, (S)-(-)-propranolol, and buspirone) led to the definition…”
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P14.05.A A PROSPECTIVE, MULTICENTER TRIAL OF FOCUSED ULTRASOUND FOR BLOOD-BRAIN BARRIER DISRUPTION FOR LIQUID BIOPSY IN GLIOBLASTOMA (LIBERATE) by Ahluwalia, M S, Ozair, A, Burns, T C, McDermott, M W, Sahgal, A, De Groot, J F, Mogilner, A, Hibert, M, Zhu, J, Achrol, A S, Shah, B, Patel, T, Rincon-Toroella, J, Mishra, M V, Everson, R J, Sporrer, J, Hilliard, J, Bezchlibnyk, Y B, Weinberg, J, Cifarelli, C, Rezai, A, Lipsman, N, Woodworth, G F

“…Abstract BACKGROUND Liquid biopsy in glioblastoma (GBM) is hindered by a lack of requisite circulating tumor (ct) and cell-free (cf) DNA levels in blood due to…”
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Protein-based virtual screening of chemical databases. II. Are homology models of g-protein coupled receptors suitable targets? by Bissantz, Caterina, Bernard, Philippe, Hibert, Marcel, Rognan, Didier

“…The aim of the current study is to investigate whether homology models of G‐Protein‐Coupled Receptors (GPCRs) that are based on bovine rhodopsin are reliable…”
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Convenient Method To Access New 4,4-Dialkoxy- and 4,4-Diaryloxy-diaza-s-indacene Dyes:  Synthesis and Spectroscopic Evaluation by Tahtaoui, Chouaib, Thomas, Cécile, Rohmer, François, Klotz, Philippe, Duportail, Guy, Mély, Yves, Bonnet, Dominique, Hibert, Marcel

“…A straightforward method for the synthesis of original 4,4-dialkoxy- or 4,4-diaryloxy-diaza-s-indacenes (BODIPY) derivatives obtained by treatment of BODIPY 1…”
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Reply by Hibert, M L, Chen, Y I, Ohringer, N, Wilbur, L R, Waheed, N K, Heier, J S, Calhoun, M W, Rosenfeld, P J, Polimeni, J R

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Reply by Hibert, M L, Chen, Y I, Ohringer, N, Wilbur, L R, Waheed, N K, Heier, J S, Calhoun, M W, Rosenfeld, P J, Polimeni, J R

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Functional Architecture of Vasopressin/Oxytocin Receptors by Hibert, M., Hoflack, J., Trumpp-Kallmeyer, S., Mouillac, B., Chini, B., Mahea, E., Cotte, N., Jard, S., Manning, M., Barberis, C.

“…Abstract Three-dimensional models of G protein-coupled receptors (GPCR) have been defined using most experimental data available and protein modeling…”
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Time-Resolved FRET Binding Assay to Investigate Hetero-Oligomer Binding Properties: Proof of Concept with Dopamine D1/D3 Heterodimer by Hounsou, Candide, Margathe, Jean-François, Oueslati, Nadia, Belhocine, Abderazak, Dupuis, Elodie, Thomas, Cécile, Mann, André, Ilien, Brigitte, Rognan, Didier, Trinquet, Eric, Hibert, Marcel, Pin, Jean-Philippe, Bonnet, Dominique, Durroux, Thierry

“…G protein-coupled receptors (GPCRs) have been described to form hetero-oligomers. The importance of these complexes in physiology and pathology is considered…”
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P349Catheter ablation of AF recurrences after PVI: only Re-PVI or further substrate modification? A retrospective long term follow up analysis by Bordignon, S, Hibert, M, Nagase, T, Chen, S, Bologna, F, Perrotta, L, Weise, F K, Konstantinou, A, Schmidt, B, Chun, KRJ

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