Search Results - "Gyovai, András"
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Antiproliferative and Antimicrobial Activities of Selected Bryophytes
Published in Molecules (Basel, Switzerland) (23-06-2018)“…One-hundred and sixty-eight aqueous and organic extracts of 42 selected bryophyte species were screened in vitro for antiproliferative activity on a panel of…”
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Journal Article -
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Preparation of Dearomatized p‐Coumaric Acid Derivatives as DNA Damage Response Inhibitors with Potent In Vitro Antitumor Effect
Published in ChemMedChem (01-10-2024)“…Our research group previously identified graviquinone (1) as a promising antitumor metabolite that is formed in situ when the antioxidant methyl caffeate…”
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Stereoselective synthesis of new type of estradiol hybrid molecules and their antiproliferative activities
Published in Steroids (01-08-2019)“…[Display omitted] •Novel 16-substituted estrone hybrids were synthesized.•Certain compounds proved to be antiproliferative against human cancer cell lines.•The…”
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Microwave-assisted stereoselective approach to novel steroidal ring D-fused 2-pyrazolines and an evaluation of their cell-growth inhibitory effects in vitro
Published in Steroids (01-08-2016)“…•Microwave-assisted reactions of 16-dehydropregnenolone and hydrazines were carried out.•Pyrazoline heteroring was introduced into ring D of the sterane…”
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Stereocontrolled synthesis of the four 16-hydroxymethyl-19-nortestosterone isomers and their antiproliferative activities
Published in Steroids (01-01-2016)“…[Display omitted] •Synthesis of 16-hydroxymethyl-19-nortestosterone isomers by Birch reduction.•Synthesis of 17α-hydroxy-19-nortestosterone esters by Mitsunobu…”
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Antiproliferative Properties of Newly Synthesized 19-Nortestosterone Analogs Without Substantial Androgenic Activity
Published in Frontiers in pharmacology (27-07-2018)“…19-Nortestosterone C-17 epimers with prominent antiproliferative properties have been previously described. In our present study, five novel…”
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A novel cluster of C5-curcuminoids: design, synthesis, in vitro antiproliferative activity and DNA binding of bis(arylidene)-4-cyclanone derivatives based on 4-hydroxycyclohexanone scaffold
Published in Research on chemical intermediates (2019)“…A new series ( 6 ) of C 5 -curcuminoid derivatives (2 E ,6 E- 2,6-dibenzylidene-4-hydroxycyclohexanones) is described here with their evaluation for in vitro…”
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Characterization of Antineoplastic Properties of Novel Androstane-Based Synthetic Steroids
Published 01-01-2019“…On the basis of our current scientific results, the following statements can be declared:• 14 hybrid compounds from the 15 prepared androstane-quinoline…”
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Dissertation -
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