Search Results - "Guerrero, Adrian M"

High incidence of lung cancer and malignant mesothelioma linked to erionite fibre exposure in a rural community in Central Mexico by Ortega-Guerrero, M Adrián, Carrasco-Núñez, Gerardo, Barragán-Campos, Héctor, Ortega, Martín R

“…Objective To report the high incidence of lung cancer (LC) and malignant mesothelioma (MM) linked to environmental exposure to erionite fibres in a rural…”
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Bismuth nitrate-induced novel nitration of estradiol: An entry to new anticancer agents by Bandyopadhyay, Debasish, Rivera, Gildardo, Sanchez, Jorge L., Rivera, Jesse, Granados, Jose C., Guerrero, Adrian M., Chang, Fang-Mei, Dearth, Robert K., Short, John D., Banik, Bimal K.

“…Direct nitration of estradiol was carried out using metal nitrates on solid surfaces under mild condition, and a combination of bismuth nitrate pentahydrate…”
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Investigation of Novel Primary and Secondary Pharmacophores and 3-Substitution in the Linking Chain of a Series of Highly Selective and Bitopic Dopamine D 3 Receptor Antagonists and Partial Agonists by Shaik, Anver Basha, Kumar, Vivek, Bonifazi, Alessandro, Guerrero, Adrian M, Cemaj, Sophie L, Gadiano, Alexandra, Lam, Jenny, Xi, Zheng-Xiong, Rais, Rana, Slusher, Barbara S, Newman, Amy Hauck

“…Dopamine D receptors (D R) play a critical role in neuropsychiatric conditions including substance use disorders (SUD). Recently, we reported a series of…”
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Investigation of Novel Primary and Secondary Pharmacophores and 3‑Substitution in the Linking Chain of a Series of Highly Selective and Bitopic Dopamine D3 Receptor Antagonists and Partial Agonists by Shaik, Anver Basha, Kumar, Vivek, Bonifazi, Alessandro, Guerrero, Adrian M, Cemaj, Sophie L, Gadiano, Alexandra, Lam, Jenny, Xi, Zheng-Xiong, Rais, Rana, Slusher, Barbara S, Newman, Amy Hauck

“…Dopamine D3 receptors (D3R) play a critical role in neuropsychiatric conditions including substance use disorders (SUD). Recently, we reported a series of…”
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Novel Bivalent Ligands Based on the Sumanirole Pharmacophore Reveal Dopamine D2 Receptor (D2R) Biased Agonism by Bonifazi, Alessandro, Yano, Hideaki, Ellenberger, Michael P, Muller, Ludovic, Kumar, Vivek, Zou, Mu-Fa, Cai, Ning Sheng, Guerrero, Adrian M, Woods, Amina S, Shi, Lei, Newman, Amy Hauck

“…The development of bivalent ligands has attracted interest as a way to potentially improve the selectivity and/or affinity for a specific receptor subtype. The…”
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Novel Bivalent Ligands Based on the Sumanirole Pharmacophore Reveal Dopamine D 2 Receptor (D 2 R) Biased Agonism by Bonifazi, Alessandro, Yano, Hideaki, Ellenberger, Michael P, Muller, Ludovic, Kumar, Vivek, Zou, Mu-Fa, Cai, Ning Sheng, Guerrero, Adrian M, Woods, Amina S, Shi, Lei, Newman, Amy Hauck

“…The development of bivalent ligands has attracted interest as a way to potentially improve the selectivity and/or affinity for a specific receptor subtype. The…”
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The Significance of Chirality in Drug Design and Synthesis of Bitopic Ligands as D3 Receptor (D3R) Selective Agonists by Battiti, Francisco O, Cemaj, Sophie L, Guerrero, Adrian M, Shaik, Anver Basha, Lam, Jenny, Rais, Rana, Slusher, Barbara S, Deschamps, Jeffery R, Imler, Greg H, Newman, Amy Hauck, Bonifazi, Alessandro

“…Because of the large degree of homology among dopamine D2-like receptors, discovering ligands capable of discriminating between the D2, D3, and D4 receptor…”
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The Significance of Chirality in Drug Design and Synthesis of Bitopic Ligands as D 3 Receptor (D 3 R) Selective Agonists by Battiti, Francisco O, Cemaj, Sophie L, Guerrero, Adrian M, Shaik, Anver Basha, Lam, Jenny, Rais, Rana, Slusher, Barbara S, Deschamps, Jeffery R, Imler, Greg H, Newman, Amy Hauck, Bonifazi, Alessandro

“…Because of the large degree of homology among dopamine D -like receptors, discovering ligands capable of discriminating between the D , D , and D receptor…”
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Novel and Potent Dopamine D 2 Receptor Go-Protein Biased Agonists by Bonifazi, Alessandro, Yano, Hideaki, Guerrero, Adrian M, Kumar, Vivek, Hoffman, Alexander F, Lupica, Carl R, Shi, Lei, Newman, Amy Hauck

“…The discovery of functionally biased and physiologically beneficial ligands directed toward G-protein coupled receptors (GPCRs) has provided the impetus to…”
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Novel and Potent Dopamine D2 Receptor Go-Protein Biased Agonists by Bonifazi, Alessandro, Yano, Hideaki, Guerrero, Adrian M, Kumar, Vivek, Hoffman, Alexander F, Lupica, Carl R, Shi, Lei, Newman, Amy Hauck

“…The discovery of functionally biased and physiologically beneficial ligands directed toward G-protein coupled receptors (GPCRs) has provided the impetus to…”
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Presencia, distribución, hidrogeoquímica y origen de arsénico, fluoruro y otros elementos traza disueltos en agua subterránea, a escala de cuenca hidrológica tributaria de Lerma-Chapala, México by Ortega-Guerrero, M. Adrián

“…The occurrence, distribution and origin of total inorganic arsenic (iAs), fl uoride (F ¿) and other trace elements (Se, Sb, V, Cr, Mo, Re, Pb, Cu, Cd, Co y Zn)…”
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Evidence for a Stereoselective Mechanism for Bitopic Activity by Extended-Length Antagonists of the D3 Dopamine Receptor by Moritz, Amy E, Bonifazi, Alessandro, Guerrero, Adrian M, Kumar, Vivek, Free, R. Benjamin, Lane, J. Robert, Verma, Ravi Kumar, Shi, Lei, Newman, Amy Hauck, Sibley, David R

“…The D3 dopamine receptor (D3R) has been suggested as a drug target for the treatment of a number of neuropsychiatric disorders, including substance use…”
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Efficient Routes to a Diverse Array of Amino Alcohol-Derived Chiral Fragments by Haftchenary, Sina, Nelson, Shawn D, Furst, Laura, Dandapani, Sivaraman, Ferrara, Steven J, Bošković, Žarko V, Figueroa Lazú, Samuel, Guerrero, Adrian M, Serrano, Juan C, Crews, DeMarcus K, Brackeen, Cristina, Mowat, Jeffrey, Brumby, Thomas, Bauser, Marcus, Schreiber, Stuart L, Phillips, Andrew J

“…Efficient syntheses of chiral fragments derived from chiral amino alcohols are described. Several unique scaffolds were readily accessed in 1–5 synthetic steps…”
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Design, synthesis and biological evaluation of novel pyrenyl derivatives as anticancer agents by Bandyopadhyay, Debasish, Sanchez, Jorge L., Guerrero, Adrian M., Chang, Fang-Mei, Granados, Jose C., Short, John D., Banik, Bimal K.

“…Polycyclic aromatic hydrocarbons are widespread in nature with a toxicity range from non-toxic to extremely toxic. A series of pyrenyl derivatives has been…”
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Evidence for a Stereoselective Mechanism for Bitopic Activity by Extended-Length Antagonists of the D 3 Dopamine Receptor by Moritz, Amy E, Bonifazi, Alessandro, Guerrero, Adrian M, Kumar, Vivek, Free, R Benjamin, Lane, J Robert, Verma, Ravi Kumar, Shi, Lei, Newman, Amy Hauck, Sibley, David R

“…The D3 dopamine receptor (D3R) has been suggested as a drug target for the treatment of a number of neuropsychiatric disorders, including substance use…”
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Environmental occurrence, origin, physical and geochemical properties, and carcinogenic potential of erionite near San Miguel de Allende, Mexico by Ortega-Guerrero, M. Adrián, Carrasco-Núñez, Gerardo

“…Detailed geologic surveys and different microscopic and analytical techniques were conducted near Tierra Blanca de Abajo where lung cancer and malignant…”
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Análisis numérico acoplado de los desplazamientos verticales y generación de fracturas por extracción de agua subterránea en las proximidades de la Ciudad de México by Lugo Hubp, José, Aguilar Pérez, Antonio, Ortiz-Zamora, Dalia del C, Ortega-Guerrero, M. Adrián

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High incidence of lung cancer and malignant mesothelioma linked to erionite fibre exposure in a rural community in Central Mexico: Table 1 by Ortega-Guerrero, M Adrián, Carrasco-Núñez, Gerardo, Barragán-Campos, Héctor, Ortega, Martín R

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Elementos de tierras raras en agua subterránea y su relación con los sistemas flujo en rocas marinas y volcánicas del Centro de México by Salinas-Reyes, Tatiana, Ortega-Guerrero, M. Adrián

“…Se utilizan Elementos de Tierras Raras (ETR) - serie de los lantánidos - disueltos en agua subterránea para determinar su interacción con medios granulares y…”
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Análisis de la dinámica del agua en la zona no saturada en un suelo sujeto a prácticas de conservación: implicaciones en la gestión de acuíferos y adaptación al cambio climático by Aguilar García, Ramón, Ortega Guerrero, Marcos Adrián

“…Se estima que entre el 80 y el 85 % del agua que se extrae de los acuíferos en México se destina a producción agropecuaria y, en general, existe una gestión…”
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