Search Results - "Gudimani, Parashuram"

Solvent-Free Synthesis, Characterization, and In Vitro Biological Activity Study of Xanthenediones and Acridinediones by Madar, Jyoti M., Samundeeswari, S., Holiyachi, Megharaja, Naik, Nirmala S., Pawar, Varsha, Gudimani, Parashuram, Shastri, Lokesh A., Kumbar, Vijay M., Sunagar, Vinay A.

“…The present work highlights the broad range of oxygen and nitrogen heterocycles and their applications in medicinal field. A facial approach has been developed…”
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Rational design, synthesis and SAR study of novel warfarin analogous of 4-hydroxy coumarin-beta-aryl propanoic acid derivatives as potent anti-inflammatory agents by Pawar, Varsha, Shastri, Lokesh A., Gudimani, Parashuram, Joshi, Shrinivas, Kumbar, Vijay M., Sunagar, Vinay

“…•A simple, economic, eco-friendly acid catalysed pyran ring opening led to warfarin analogue 3-(4‑hydroxy-2-oxo-2H-chromen-3-yl)−3-arylpropanoic acid…”
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Synthesis, characterization and molecular docking of novel lonazolac analogues 3-(3-hydroxy-5-methyl-1H-pyrazol-4-yl)-3-arylpropanoic acid derivatives: Highly potential COX-1/COX-2, matrix metalloproteinase and protein denaturation inhibitors by Pawar, Varsha, Shastri, Lokesh A., Gudimani, Parashuram, Joshi, Shrinivas, Sunagar, Vinay

“…•A simple, economic, eco-friendly acid catalysed pyran ring opening led to single isomer of novel lonazolac analogous,…”
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Click approach for synthesis of 3,4-dihydro-2(1H) quinolinone, coumarin moored 1,2,3-triazoles as inhibitor of mycobacteria tuberculosis H37RV, their antioxidant, cytotoxicity and in-silico studies by Hebbar, Nagashree U., Patil, Anilkumar R., Gudimani, Parashuram, Shastri, Samundeeswari L., Shastri, Lokesh A., Joshi, Shrinivas D., Vootla, Shyam Kumar, Khanapure, Sheela, Shettar, Arun K., Sungar, Vinay A.

“…•Simple synthetic procedures were employed to synthesize new triazole bridged bi-heterocycles.•Synthesized scaffolds were assessed for their in vitro…”
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A new approach for the synthesis of tri-substituted pyrazole propionic acids derivatives: Anti-inflammatory, antimicrobial and molecular docking studies by Gudimani, Parashuram, Hebbar, Nagashree U, Shastri, Samundeeswari L, Shastri, Lokesh A., Shettar, Arun K, Hoskeri, Joy H, Joshi, Shrinivas, Sunagar, Vinay A

“…•Efficient synthetic route for the synthesis oftri-substituted propanoic acid derivatives which are analogous to known drug lonazolac.•Synthesized scaffolds…”
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Synthesis, characterization of 1,2,4-triazolidine-3-thione tethered beta-aryl butanoic acid and butanoate derivatives as potent antimicrobial and antioxidant agents and their molecular docking studies by Hebbar, Nagashree U, Hebbar, Prateeksha Subray, Rathode, Pooja Prakash, Negalura, Beerappa, Hiremath, Aishwarya, Gudimani, Parashuram, Shastri, Lokesh A, Praveen Kumar, S.K., Kadapure, Arihant Jayawant, Joshi, Shrinivas

“…•Environmentally friendly synthetic procedures were employed to synthesize new triazolidine 3-thione substituted beta aryl compounds.•Synthesized scaffolds…”
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Indirect, catalyst free β-arylation of acyclic 1,5-dicarbonyl compounds via green method by Gudimani, Parashuram, Shastri, Samundeeswari.L., Pawar, Varsha, Shastri, Lokesh A., Sungar, Vinay A.

“…•Reaction performed in aqueous ethanol (first step) and formic acid (second step).•Experimental condition is high substrate scope and ecofriendly.•No metal…”
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1,6-Diamino-dihydropyridine and triazolo[1,5-a]pyridine analogues as a highly promising coumarin scaffold for the development of bacterial infection inhibitors by Naik, Nirmala S., S, Samundeeswari, Chougala, Bahubali M., H, Megharaja, Pawar, Varsha, Gudimani, Parashuram, Shastri, Lokesh A., Dodamani, Suneel, Jalalpure, Sunil, Sunagar, Vinay

“…•Keeping in mind the biological activity of coumarin and pyridino-triazole scaffolds were designed and synthesized successfully using ecofriendly method.•The…”
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