Search Results - "Grosu, G."

Maxwell’s relations and thermal coefficients for repulsive clathrates by Eroshenko, V. A., Grosu, Ya. G.

“…Prospects of nanotechnologies used for designing more effective thermomechanical devices and systems based on repulsive clathrates are outlined. Basic…”
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Selective Hydrolysis of Ethyl 5,6-Dihydro-4H-pyrrolo[1,2-b]pyrazole-2-carboxylate and Ethyl 5,6-Dihydro-4H-pyrrolo[1,2-b]pyrazole-3-carboxylate as a Key Step in the Large-Scale Synthesis of Bicyclic Heteroaryl Carboxyaldehydes by Nikitenko, A. A, Winkley, M. W, Zeldis, J, Kremer, K, Chan, A. W.-Y, Strong, H, Jennings, M, Jirkovsky, I, Blum, D, Khafizova, G, Grosu, G. T, Venkatesan, A. M

“…The isomeric mixture of ethyl 5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole-2- and −3-carboxylates (14 and 15), derived from a proline meso-ionic synthon, demonstrated…”
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Highly sensitive solid forms discrimination on the whole tablet of the active ingredients in quercetin dietary supplements by NMR crystallography approaches by Miclaus, Maria O., Filip, Xenia, Filip, Claudiu, Martin, Flavia A., Grosu, Ioana G.

“…[Display omitted] •Non-destructive solid-forms determination by combined PXRD and ss-NMR is demonstrated on quercetin dietary supplements.•Good sensitivity to…”
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Prodrugs of CL316243: a selective β3-adrenergic receptor agonist for treating obesity and diabetes by Sum, F.W., Gilbert, A., Venkatesan, A.M., Lim, K., Wong, V., O'Dell, M., Francisco, G., Chen, Z., Grosu, G., Baker, J., Ellingboe, J., Malamas, M., Gunawan, I., Primeau, J., Largis, E., Steiner, K.

“…CL316243 is a highly selective and potent β 3-adrenergic receptor agonist, and has been shown in rodent models to be an effective agent for treating obesity…”
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5-fluoro-2-methyl-N-[5-(5 H-pyrrolo[2,1- c][1,4]benzodiazepine-10(11 H)-yl carbonyl)-2-pyridinyl]benzamide (CL-385004) and analogs as orally active arginine vasopressin receptor antagonists by Aranapakam, Venkatesan, Albright, J.Donald, Grosu, George T., Delos Santos, Efren G., Chan, Peter S., Coupet, Joseph, Ru, Xun, Saunders, Trina, Mazandarani, H.

“…Synthesis and structure-activity relationships (SAR) of orally active arginine vasopressin (AVP) receptor antagonists are discussed. Potent and orally active…”
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4,10-Dihydro-5h-thieno[3,2-c][1]benzazepine derivatives and 9,10-dihydro-4h-thieno[2,3-c][1]benzazepine derivatives as orally active arginine vasopressin receptor antagonists by ARANAPAKAM, V, ALBRIGHT, J. D, GROSU, G. T, CHAN, P. S, COUPET, J, SAUNDERS, T, XUN RU, MAZANDARANI, H

“…Synthesis and structure-activity relationships (SAR) of arginine vasopressin receptor (AVP) antagonists are described. Potent and orally active compounds are…”
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Thermomechanical and thermophysical properties of repulsive clathrates by Eroshenko, V. A., Grosu, Ya. G.

“…The range of the characteristic properties of repulsive clathrates (RCs), which are new working media used for efficient energy conversion in thermomechanical…”
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Visual processing of configuration-dependent spatial characteristics of shapes and patterns. A model useful in the study of the role of the departure from circularity or dispersion of shapes in human visual perception by Bonciocat, C A, Grosu, G, Ghiţă, S

“…In this work a theoretical model was used in combination with testings on normal subjects to get more insight in the role of the departure from circularity or…”
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Thermal fragmentation reactions of dihydroaromatic molecules by Miller, Bernard, Shi, Xiaolian, Grosu, George, Zhou, Renmo

“…Thermal decompositions of 1,4-dihydrobenzene derivatives (usually at temperatures in the 300-350[degrees]C range) result in elimination of hydrogen, provided…”
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The impact of automated hippocampal volumetry on diagnostic confidence in patients with suspected Alzheimer's disease: An EADC study by Bosco, Paolo, Redolfi, Alberto, Bocchetta, Martina, Ferrari, Clarissa, Mega, Anna, Galluzzi, Samantha, Austin, Mark, Chincarini, Andrea, Collins, D. Louis, Duchesne, Simon, Maréchal, Bénédicte, Roche, Alexis, Sensi, Francesco, Wolz, Robin, Alegret, Montserrat, Assal, Frederic, Balasa, Mircea, Bastin, Christine, Bougea, Anastasia, Emek-Savaş, Derya Durusu, Engelborghs, Sebastiaan, Grimmer, Timo, Grosu, Galina, Kramberger, Milica G, Lawlor, Brian, Mandic Stojmenovic, Gorana, Marinescu, Mihaela, Mecocci, Patrizia, Molinuevo, José Luis, Morais, Ricardo, Niemantsverdriet, Ellis, Nobili, Flavio, Ntovas, Konstantinos, O'Dwyer, Sarah, Paraskevas, George P, Pelini, Luca, Picco, Agnese, Salmon, Eric, Santana, Isabel, Sotolongo-Grau, Oscar, Spiru, Luiza, Stefanova, Elka, Popovic, Katarina Surlan, Tsolaki, Magda, Yener, Görsev G, Zekry, Dina, Frisoni, Giovanni B

“…Abstract Introduction Hippocampal volume is a core biomarker of Alzheimer's disease (AD). However, its contribution over the standard diagnostic workup is…”
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Metoprolol infusion reduces fentanyl requirements during ballanced general anesthesia for moderate amplitude surgery: 4AP5-9 by Guran, C., Dragulin, E., Grosu, G. Vasile, Moise, A., Mincu, N.

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Structure–activity study of novel tricyclic benzazepine arginine vasopressin antagonists by Sum, Fuk-Wah, Dusza, John, Santos, Efren Delos, Grosu, George, Reich, Marvin, Du, Xumei, Albright, J.Donald, Chan, Peter, Coupet, Joseph, Ru, Xun, Mazandarani, Hossein, Saunders, Trina

“…Novel tricyclic benzazepine derivatives were synthesized as arginine vasopressin (AVP) antagonists. Several tricyclic compounds showed potent antagonistic…”
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Thermodynamic and operational properties of heterogeneous lyophobic systems by Eroshenko, Valentin, Grosu, Yaroslav

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In vitro antimicrobial activity of new 1,10-phenantroline derivatives by Druta, I, Danac, R, Ungureanu, M, Grosu, G, Drochioiu, G

“…The antimicrobial and antifungical activities of some 1,10-phenanthroline derivatives are described. The test was performed using the diffusimetric method with…”
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New derivatives of 1-methyl-phthalazine with antimicrobial and fungistatic action by Dima, S, Caprosu, M, Ungureanu, M, Grosu, G, Petrovanu, M

“…In this paper we present the antimicrobial and antifungical action of some new salts of 1-methyl-phtalaziniums and their corresponding ylids. We also present…”
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Tetrazolium salts and metal complexes of some formazans by Stefănescu, E, Dorneanu, M, Dănilă, C, Aprotosoaie, C, Grosu, G

“…This paper presents the synthesis of some tetrazolium salts and metal complexes combinations, which are derived from aromatic and heterocyclic formazans…”
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Prodrugs of CL316243: a selective beta3-adrenergic receptor agonist for treating obesity and diabetes by Sum, F W, Gilbert, A, Venkatesan, A M, Lim, K, Wong, V, O'Dell, M, Francisco, G, Chen, Z, Grosu, G, Baker, J, Ellingboe, J, Malamas, M, Gunawan, I, Primeau, J, Largis, E, Steiner, K

“…CL316243 is a highly selective and potent beta3-adrenergic receptor agonist, and has been shown in rodent models to be an effective agent for treating obesity…”
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Antimicrobial activity of some derivatives of pyrimidine by Mangalagiu, I, Ungureanu, M, Mangalagiu, G, Grosu, G, Petrovanu, M

“…In this paper the authors present the antimicrobial and antifungical tests of some new 3-methylpyrimidine compounds. The test was performed using the…”
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Synthesis and Structure−Activity Relationship of N-Substituted 4-Arylsulfonylpiperidine-4-hydroxamic Acids as Novel, Orally Active Matrix Metalloproteinase Inhibitors for the Treatment of Osteoarthritis by Aranapakam, Venkatesan, Davis, Jamie M, Grosu, George T, Baker, Ellingboe, John, Zask, Arie, Levin, Jeremy I, Sandanayaka, Vincent P, Du, Mila, Skotnicki, Jerauld S, DiJoseph, John F, Sung, Amy, Sharr, Michele A, Killar, Loran M, Walter, Thomas, Jin, Guixian, Cowling, Rebecca, Tillett, Jeff, Zhao, Weiguang, McDevitt, Joseph, Xu, Zhang Bao

“…The matrix metalloproteinases (MMPs) are a family of zinc-containing endopeptidases that play a key role in both physiological and pathological tissue…”
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Synthesis and Structure−Activity Relationship of α-Sulfonylhydroxamic Acids as Novel, Orally Active Matrix Metalloproteinase Inhibitors for the Treatment of Osteoarthritis by Aranapakam, Venkatesan, Grosu, George T, Davis, Jamie M, Hu, Baihua, Ellingboe, John, Baker, Jannie L, Skotnicki, Jerauld S, Zask, Arie, DiJoseph, John F, Sung, Amy, Sharr, Michele A, Killar, Loran M, Walter, Thomas, Jin, Guixian, Cowling, Rebecca

“…The matrix metalloproteinases (MMPs) are a family of zinc-containing endopeptidases that play a key role in both physiological and pathological tissue…”
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