Search Results - "Grella, G E"

Synthesis and aldose reductase inhibitory activities of novel thienocinnolinone derivatives by Pau, A, Asproni, B, Boatto, G, Grella, G.E, De Caprariis, P, Costantino, L, Pinna, G.A

“…A novel series of tetrahydrothieno[2,3- h]cinnolinone derivatives were synthesized and evaluated in vitro for their ability to inhibit aldose reductase (ALR2),…”
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Synthesis and cytotoxicity of substituted 2-benzylnaphth[2,3- d]imidazoles by Grella, G.E, Cabras, M.C, Murineddu, G, Pau, A, Pinna, G.A

“…Designed as a new series of so called “bivalent ligand” containing the proposed 2-benzylnaphthimidazole-type structure, a number of 2-benzylnaphth[2,3-…”
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Thienocinnolinone alkanoic acid derivatives as aldose reductase inhibitors by Pau, A, Asproni, B, Murineddu, G, Boatto, G, Grella, G E, Rakowitz, D, Costantino, L, Pinna, G A

“…A new series of 8-halogen-4,4a,5,6-tetrahydrothieno[2,3-h]cinnolinone-N2-alkanoic acids was prepared and tested for aldose reductase (ALR2) inhibitory…”
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Synthesis and cytotoxicity of bis(benzo[g]indole-3-carboxamides) and related compounds by Pinna, Gérard A., Pirisi, Maria A., Grella, Giuseppe E., Gherardini, Laura, Mussinu, Jean M., Paglietti, Giuseppe, Ferrari, Anna M., Rastelli, Giulio

“…A series of bis(benzo[g]indoles) bridged by CX‐(CH2)nN(Me)(CH2)n‐CX (X = O, S, H2; n = 2,3) was synthesized as bifunctional antitumor agents and evaluated for…”
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Synthesis of novel diazatricyclodecanes (DTDs). Effects of structural variation at the C3′ allyl end and at the phenyl ring of the cinnamyl chain on μ-receptor affinity and opioid antinociception by Pinna, Gérard Aimè, Cignarella, Giorgio, Ruiu, Stefania, Loriga, Giovanni, Murineddu, Gabriele, Villa, Stefania, Grella, Giuseppe Enrico, Cossu, Gregorio, Fratta, Walter

“…Two series of analogues of 9-propionyl-10-cinnamyl-9,10-diazatricyclo[4.2.1.1 2,5]decane ( 1a) and 2-propionyl-7-cinnamyl-2,7-diazatricyclo[4.4.0.0 3,8]decane…”
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Preparation and pharmacologic activity of 2-(4'R')benzyl-5R-benzimidazole and 2-(4'-pyridinyl)-5R-benzimidazoles. Analgesic activity and effect on conditioned avoidance response by Paglietti, G, Pirisi, M A, Loriga, M, Grella, G E, Sparatore, F, Satta, M, Manca, P

“…Sixteen 2-(4'R')phenyl-5R-benzimidazoles and two 2-(4'-pyridinyl)-5R-benzimidazoles were prepared and tested, together with 2-phenylbenzimidazole, for their…”
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Preparation and pharmacologic activity of 2-(4'R')benzyl-5R-benzimidazole. Analgesic activity and effect on conditioned avoidance response by Paglietti, G, Pirisi, M A, Loriga, M, Grella, G E, Sparatore, F, Satta, M, Manca, P, Peana, A

“…Several derivatives of 2-benzylbenzimidazole (dibazole) bearing substituents on positions 5 and 4' were prepared and tested, together with dibazole, for their…”
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