Search Results - "Gouda, Moustafa. A."
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Design, synthesis and identification of novel substituted isothiochromene analogs as potential antiviral and cytotoxic agents
Published in Medicinal chemistry research (01-10-2018)“…In this study, we present the synthesis of novel isothiochromenes, thiazolidonone, thiazinone, arylidines, triazoles, and pyrimidinone compounds based on the…”
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2
Synthesis of Benzofuran Derivatives via Different Methods
Published in Synthetic communications (18-08-2014)“…This review presents a systematic and comprehensive survey of the methods of preparation of benzofurans. These compounds are important intermediates for the…”
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3
Recent progress on coumarin scaffold‐based anti‐microbial agents (Part III)
Published in Journal of heterocyclic chemistry (01-11-2020)“…The biological, therapeutic, and medicinal properties of coumarins (chromen‐2‐ones), and its analogs have triggered enormous studies aimed toward growing…”
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4
Recent Progress on Nicotinonitrile Scaffold‐based Anticancer, Antitumor, and Antimicrobial Agents: A Literature Review
Published in Journal of heterocyclic chemistry (01-10-2018)“…The considerable biological activities of nicotinonitriles and its analogues are attracting attention of chemist aimed at developing synthetic routes to these…”
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5
Synthesis, Characterization, Antioxidant and Antitumor Evaluation of Some New Thiazolidine and Thiazolidinone Derivatives
Published in Archiv der Pharmazie (Weinheim) (01-03-2011)“…2‐(2‐Cyano‐acetylamino)‐4,5,6,7‐tetrahydrobenzo[b]thiophene‐3‐carboxylic acid ethyl ester (2) was utilized as a key intermediate for the synthesis of…”
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6
Design and In vitro Investigation of Grafted Chitosan as Chitosan Nanoparticles Containing Deflazacort Drug Coated by Calcium Starch Glycolate
Published in Fibers and polymers (01-12-2020)“…Novel chitosan nanoparticles (SCN) were synthesized via reaction of chitosan with different concentration of 2-chloro- N -(3-methylisoxazol-5-yl) acetamide (5…”
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7
Synthesis and Antioxidant Activity of Some New Binary Pyrazoles Containing Core Phenothiazine Moiety
Published in Journal of heterocyclic chemistry (01-03-2017)“…α,β‐Unsaturated ketones containing phenothiazine moiety 4, 5, and 7 were synthesized by condensation of 2‐acetylphenothiazine (1) with different aryl aldehydes…”
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8
Synthesis and Antioxidant Evaluation of Some New 3-Substituted Coumarins
Published in Archiv der Pharmazie (Weinheim) (01-11-2011)“…3‐Acetylcoumarin (1) was utilized as a key intermediate for the synthesis of 2‐aminothiazole derivative 3 via bromination of 1 to afford acetylbromide 2…”
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9
Recent progress in the chemical reactivity of 3-Amino-1H-pyrazol-5(4H)-one derivatives (part II)
Published in Synthetic communications (18-08-2021)“…Pyrazolone and its derivatives are an crucial class of heterocyclic compounds that may be traced in in a number of well-established drugs, such as celecoxib,…”
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10
Recent progress on the synthetic routes of 5-amino-2,4-dihydro-3H-pyrazol-3-one derivatives and their reactivity Part (I)
Published in Synthetic communications (03-05-2021)“…Pyrazolone and its derivatives are an important class of heterocyclic compounds that are found in many drugs. They represent an interesting model for…”
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11
An overview of the synthetic routes to Faipiravir and their analogous
Published in Journal of heterocyclic chemistry (01-08-2021)“…The biological and medicinal properties of Favipiravir and its analogs have prompted enormous research aimed at developing synthetic routes to these…”
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12
Overview of the synthetic routes to tadalafil and its analogues
Published in Synthetic communications (17-12-2017)“…The biological and medicinal properties of tadalafil and its analogues have prompted enormous research aimed at developing synthetic routes to these…”
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13
Synthesis of 1,2,4‐triazolopyridazines, isoxazolofuropyridazines, and tetrazolopyridazines as antimicrobial agents
Published in Journal of heterocyclic chemistry (01-09-2020)“…Through current and previous researches, it was found that the derivatives of pyridazine, isoxazole, tetrazole, quinazoline, hydrazinyl, and 1,2,4‐triazole…”
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14
Synthesis and Antioxidant Evaluation of Some Novel Thiophene, Pyrazole, Chromene, Pyrazolotriazine Derivatives Bearing Sulfonamide Moiety
Published in Journal of heterocyclic chemistry (01-01-2017)“…As a part of ongoing studies in developing new potent antioxidant agents, N‐[4‐(aminosulfonyl)phenyl]‐2‐cyanoacetamide (3) was utilized as key intermediate for…”
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15
Recent Advances in Imidazo[5,1‐f][1,2,4]triazin‐4(3H)‐ones Chemistry: An Overview of the Synthetic Routes to Vardenafil and Its Analogues
Published in Journal of heterocyclic chemistry (01-03-2018)“…The biological and medicinal properties of imidazo[5,1‐f][1,2,4]triazin‐4(3H)‐ones and its analogues have prompted enormous research aimed at developing…”
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16
Piperazine Heterocycles as Potential Anticancer Agents: A Review
Published in Pharmaceutical chemistry journal (01-04-2022)“…Cancer is a rapid, out of control, and proliferation pathology of ordinary cells, which has become one of the most infamous and aggressive health afflictions…”
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17
Chemistry of 4,4′-(arylmethylene)-bis(3-methyl-1-phenyl-1H-pyrazol-5-ol)s
Published in Journal of heterocyclic chemistry (01-03-2016)“…This review presents a systematic and comprehensive survey of the method of preparation and the chemical reactivity of…”
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18
Overview of the synthetic routes of 2-alkyl-4-hydroxy-2H-1,2-benzothiazine-3-carboxamides-1,1-dioxides (oxicams) and their analogues
Published in Synthetic communications (01-01-2017)“…The biological and medicinal properties of oxicams and its analogues have prompted enormous research aimed at developing synthetic routes to these…”
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19
Synthesis and Antioxidant Evaluation of Some New Pyridopyrazolotriazine Derivatives
Published in Journal of heterocyclic chemistry (01-07-2015)“…Diazodization of pyrazolo[3,4‐b]pyridine 1 afforded diazonium salt 2 that coupled with active methylene compounds such as 3a,3b, 6, 7, 8, 15a,15b, 16a,16b, 17,…”
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20
2-Cyano-N-(4-sulfamoylphenyl) Acetamide as a Synthon in Heterocyclic Synthesis
Published in Synthetic communications (02-12-2014)“…This review describes the synthesis and reactions of 2-cyano-N-(4-sulfamoylphenyl) acetamide as a building block for the synthesis of polyfunctionalized…”
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