Search Results - "Gold, Madeleine"

New naphthopyran analogues of LY290181 as potential tumor vascular-disrupting agents by Schmitt, Florian, Gold, Madeleine, Rothemund, Matthias, Andronache, Ion, Biersack, Bernhard, Schobert, Rainer, Mueller, Thomas

“…A series of 19 analogues of the antiproliferative naphthopyran LY290181 were prepared for structure–activity relationship studies. We found the best activities…”
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Fluoro and pentafluorothio analogs of the antitumoral curcuminoid EF24 with superior antiangiogenic and vascular-disruptive effects by Schmitt, Florian, Gold, Madeleine, Begemann, Gerrit, Andronache, Ion, Biersack, Bernhard, Schobert, Rainer

“…[Display omitted] •Curcuminoids 3–6 are more cytotoxic than lead compound EF24 in cancer cells.•Hexafluorinated piperidones 3c and 3d inhibit NF-κB…”
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Copper(ii) complexes with tridentate Schiff base-like ligands: solid state and solution structures and anticancer activity by Dankhoff, Katja, Gold, Madeleine, Kober, Luisa, Schmitt, Florian, Pfeifer, Lena, Dürrmann, Andreas, Kostrhunova, Hana, Rothemund, Matthias, Brabec, Viktor, Schobert, Rainer, Weber, Birgit

“…We report 15 new Cu(ii) complexes with tridentate NNO β-acylenamino ligands derived from 2-picolylamine and bearing up to three alkyl, alkoxy, alkoxycarbonyl,…”
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Synthesis and bioevaluation of new vascular-targeting and anti-angiogenic thieno[2,3-d]pyrimidin-4(3H)-ones by Gold, Madeleine, Köhler, Leonhard, Lanzloth, Clarissa, Andronache, Ion, Anant, Shrikant, Dandawate, Prasad, Biersack, Bernhard, Schobert, Rainer

“…A series of forty-six 5,6-annulated 2-arylthieno [2,3-d]pyrimidin-4(3H)-ones were prepared as potentially pleiotropic anticancer drugs with variance in the…”
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A new 4-(pyridinyl)-4H-benzo[g]chromene-5,10-dione ruthenium(II) complex inducing senescence in 518A2 melanoma cells by Gold, Madeleine, Mujahid, Yusufi, Ahmed, Khursheed, Kostrhunova, Hana, Kasparkova, Jana, Brabec, Viktor, Biersack, Bernhard, Schobert, Rainer

“…2-Amino-5,10-dihydro-5,10-dioxo-4(pyridine-3-yl)-4 H -benzo[ g ]chromene-3-carbonitrile 5 , a cytotoxic lawsone derivative, was reacted with [Ru( p -cymene)Cl…”
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Guided Antitumoural Drugs: (Imidazol‐2‐ylidene)(L)gold(I) Complexes Seeking Cellular Targets Controlled by the Nature of Ligand L by Bär, Sofia I., Gold, Madeleine, Schleser, Sebastian W., Rehm, Tobias, Bär, Alexander, Köhler, Leonhard, Carnell, Lucas R., Biersack, Bernhard, Schobert, Rainer

“…Three [1,3‐diethyl‐4‐(p‐methoxyphenyl)‐5‐(3,4,5‐trimethoxyphenyl)imidazol‐2‐ylidene](L)gold(I) complexes, 4 a (L=Cl), 5 a (L=PPh3), and 6 a (L=same…”
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Luminescent Gold(I) Complexes of 1‑Pyridyl-3-anthracenylchalcone Inducing Apoptosis in Colon Carcinoma Cells and Antivascular Effects by González, Juan Jesús, Ortega, Enrique, Rothemund, Matthias, Gold, Madeleine, Vicente, Consuelo, de Haro, Concepción, Bautista, Delia, Schobert, Rainer, Ruiz, José

“…The luminescent chalcone gold­(I) conjugates [Au­(PPh3)­(AN3E)]­PF6(1) and [Au­(SIMes)­(AN3E)]­PF6 (2) (AN3E = (E)-3-(9-anthracenyl)-1-(4-pyridyl)­propenone;…”
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Monitoring of circulating epithelial tumor cells using the Maintrac ® method and its potential benefit for the treatment of patients with colorectal cancer by Gold, Madeleine, Pachmann, Katharina, Kiani, Alexander, Schobert, Rainer

“…Circulating tumor cells are an important link between primary tumors and metastases. A longitudinal monitoring of their numbers and properties can provide…”
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A new 4-(pyridinyl)-4H-benzo[g]chromene-5,10-dione ruthenium(II) complex inducing senescence in 518A2 melanoma cells by Gold, Madeleine, Mujahid, Yusufi, Ahmed, Khursheed, Kostrhunova, Hana, Kasparkova, Jana, Brabec, Viktor, Biersack, Bernhard, Schobert, Rainer

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