Search Results - "Ghiringhelli, Francesca"

Novel chemical probes for the investigation of nonribosomal peptide assembly by Ho, Y T Candace, Leng, Daniel J, Ghiringhelli, Francesca, Wilkening, Ina, Bushell, Dexter P, Kostner, Otto, Riva, Elena, Havemann, Judith, Passarella, Daniele, Tosin, Manuela

“…Chemical probes were devised and evaluated for the capture of biosynthetic intermediates involved in the bio-assembly of the nonribosomal peptide echinomycin…”
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Direct β‐ and γ‐C(sp3)−H Alkynylation of Free Carboxylic Acids by Ghiringhelli, Francesca, Uttry, Alexander, Ghosh, Kiron Kumar, Gemmeren, Manuel

“…In this study we report the identification of a novel class of ligands for palladium‐catalyzed C(sp3)−H activation that enables the direct alkynylation of free…”
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Sterically Controlled C−H Olefination of Heteroarenes by Chen, Hao, Farizyan, Mirxan, Ghiringhelli, Francesca, Gemmeren, Manuel

“…The regioselective functionalization of heteroarenes is a highly attractive synthetic target due to the prevalence of multiply substituted heteroarenes in…”
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Ligand‐Enabled γ‐C(sp3)−H Olefination of Free Carboxylic Acids by Ghosh, Kiron Kumar, Uttry, Alexander, Mondal, Arup, Ghiringhelli, Francesca, Wedi, Philipp, Gemmeren, Manuel

“…We report the ligand‐enabled C−H activation/olefination of free carboxylic acids in the γ‐position. Through an intramolecular Michael addition, δ‐lactones are…”
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The Direct Conversion of α‑Hydroxyketones to Alkynes by Ghiringhelli, Francesca, Nattmann, Lukas, Bognar, Sabine, van Gemmeren, Manuel

“…Alkynes are highly important functional groups in organic chemistry, both as part of target structures and as versatile synthetic intermediates. In this study,…”
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Copper‐Catalysed Synthesis of Propargyl Alcohol and Derivatives from Acetylene and other Terminal Alkynes by Sitte, Nikolai A., Ghiringhelli, Francesca, Shevchenko, Grigory A., Rominger, Frank, Hashmi, A. Stephen K., Schaub, Thomas

“…A copper(I)/phosphine system that homogeneously catalyses the alkynylation of formaldehyde with acetylene or terminal alkynes is reported. Using acetylene at…”
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Direkte β‐ und γ‐C(sp3)‐H Alkinylierung freier Carbonsäuren by Ghiringhelli, Francesca, Uttry, Alexander, Ghosh, Kiron Kumar, Gemmeren, Manuel

“…In dieser Studie berichten wir über die Identifizierung einer neuen Klasse von Liganden für die Palladium‐katalysierte C(sp3)‐H‐Aktivierung, welche die direkte…”
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Sterically Controlled C−H Olefination of Heteroarenes by Chen, Hao, Farizyan, Mirxan, Ghiringhelli, Francesca, Gemmeren, Manuel

“…The regioselective functionalization of heteroarenes is a highly attractive synthetic target due to the prevalence of multiply substituted heteroarenes in…”
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Liganden‐vermittelte γ‐C(sp3)‐H‐Olefinierung freier Carbonsäuren by Ghosh, Kiron Kumar, Uttry, Alexander, Mondal, Arup, Ghiringhelli, Francesca, Wedi, Philipp, Gemmeren, Manuel

“…Wir beschreiben die Liganden‐vermittelte C‐H‐Aktivierung/Olefinierung freier Carbonsäuren in der γ‐Position. Durch eine intramolekulare Michael‐Addition werden…”
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Direkte β‐ und γ‐C(sp3)‐H Alkinylierung freier Carbonsäuren by Ghiringhelli, Francesca, Uttry, Alexander, Ghosh, Kiron Kumar, Manuel van Gemmeren

“…In dieser Studie berichten wir über die Identifizierung einer neuen Klasse von Liganden für die Palladium‐katalysierte C(sp3)‐H‐Aktivierung, welche die direkte…”
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Imidazo[2,1‑b]benzothiazol Derivatives as Potential Allosteric Inhibitors of the Glucocorticoid Receptor by Christodoulou, Michael S, Dapiaggi, Federico, Ghiringhelli, Francesca, Pieraccini, Stefano, Sironi, Maurizio, Lucafò, Marianna, Curci, Debora, Decorti, Giuliana, Stocco, Gabriele, Chirumamilla, Chandra Sekhar, Vanden Berghe, Wim, Balaguer, Patrick, Michel, Benoît Y, Burger, Alain, Beccalli, Egle M, Passarella, Daniele, Martinet, Nadine

“…Glucocorticoid receptor (GCR) transactivation reporter gene assays were used as an initial high-throughput screening on a diversified library of 1200 compounds…”
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