Search Results - "Gherbovet, Olga"

Regioselective chemoenzymatic syntheses of ferulate conjugates as chromogenic substrates for feruloyl esterases by Gherbovet, Olga, Ferreira, Fernando, Clément, Apolline, Ragon, Mélanie, Durand, Julien, Bozonnet, Sophie, O'Donohue, Michael J, Fauré, Régis

“…Generally, carbohydrate-active enzymes are studied using chromogenic substrates that provide quick and easy color-based detection of enzyme-mediated…”
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Regioselective chemo-enzymatic syntheses of ferulate conjugates as chromogenic substrates for feruloyl esterases by Gherbovet, Olga, Ferreira, Fernando, Clément, Apolline, Ragon, Mélanie, Durand, Julien, Bozonnet, Sophie, O'Donohue, Michael, Fauré, Régis

“…Generally, carbohydrate-active enzymes are studied using chromogenic substrates that provide quick and easy color-based detection of enzyme-mediated…”
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Original Vinca Derivatives: From P‑Glycoprotein Substrates to P‑Glycoprotein Inhibitors by Gherbovet, Olga, García Alvarez, María Concepción, Bignon, Jérôme, Roussi, Fanny

“…The first example of vinca derivatives 16–18 able to modulate P-glycoprotein (Pgp) efflux activity is reported. They were elaborated in two steps from…”
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Directed evolution of the type C feruloyl esterase from Fusarium oxysporum FoFaeC and molecular docking analysis of its improved variants by Cerullo, Gabriella, Varriale, Simona, Bozonnet, Sophie, Antonopoulou, Io, Christakopoulos, Paul, Rova, Ulrika, Gherbovet, Olga, Fauré, Régis, Piechot, Alexander, Jütten, Peter, Brás, Joana L.A., Fontes, Carlos M.G.A., Faraco, Vincenza

“…[Display omitted] •A library of around 30,000 random mutants of FoFaeC was generated.•Screening for enzymatic activity led to the selection of 96 improved…”
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Synthesis and biological evaluation of C-13' substituted 7'-homo-anhydrovinblastine derivatives by Gherbovet, Olga, La Spisa, Fabio, Thoret, Sylviane, Alvarez, Maria Concepcion Garcia, Levaique, Hélène, Bignon, Jérôme, Roussi, Fanny

“…Recent publications highlighted that vinca derivatives either functionalized on C-12' or enlarged on cycle C' could be more cytotoxic than vinblastine or…”
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One-Pot Synthesis of Vinca Alkaloids–Phomopsin Hybrids by Gherbovet, Olga, Coderch, Claire, García Alvarez, María Concepción, Bignon, Jérôme, Thoret, Sylviane, Guéritte, Françoise, Gago, Federico, Roussi, Fanny

“…Hybrids of vinca alkaloids and phomopsin A have been elaborated with the aim of interfering with the “vinca site” and the “peptide site” of the vinca domain in…”
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Design of chromogenic probes for efficient screening and evaluation of feruloyl esterase-like activities by Gherbovet, Olga, Fauré, Régis, Ferreira, Fernando, Durand, Julien, Ragon, Mélanie, Hostyn, Guillaume, Record, Eric, Bozonnet, Sophie, O’Donohue, Michael J.

“…[Display omitted] •Hydroxycinnamate-based chromogenic substrates were synthesized in good yields.•Detection of esterase activity was achieved in both solid and…”
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Synthesis and Biological Evaluation of a New Series of Highly Functionalized 7′-homo-Anhydrovinblastine Derivatives by Gherbovet, Olga, Coderch, Claire, García Alvarez, María Concepción, Bignon, Jérôme, Thoret, Sylviane, Martin, Marie-Thèrese, Guéritte, Françoise, Gago, Federico, Roussi, Fanny

“…Sixteen new 7′-homo-anhydrovinblastine derivatives were prepared in one or two steps from vinorelbine by means of an original and regiospecific rearrangement…”
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Regioselective chemo-enzymatic syntheses of ferulate conjugates as chromogenic substrates for feruloyl esterases by Gherbovet, Olga, Ferreira, Fernando, Clément, Apolline, Ragon, Mélanie, Durand, Julien, Bozonnet, Sophie, O'Donohue, Michael, Fauré, Régis

“…Generally, carbohydrate-active enzymes are studied using chromogenic substrates that provide quick and easy color-based detection of enzyme-mediated…”
Get full text