Search Results - "Ghazi, Somayeh"

An efficient ultrasonic-assisted synthesis of ethyl-5-(aryl)-2-(2-alkokxy-2-oxoethylidene)-7-methyl-3-oxo-3, 5-dihydro-2H-thiazolo [3, 2-a] pyrimidine-6-carboxylate derivatives by Darehkordi, Ali, Ghazi, Somayeh

“…Dihydropyrimidinone derivatives were used as key intermediates for the synthesis of ethyl-5-(aryl)-2-(2-alkokxy-2-oxoethylidene)-7-methyl-3-oxo-3,…”
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Synthesis of a New Class of Tris- and Bis(1,3,4-thiadiazol-2-amine) Methyl and Ethyl Tris- and Bis-2-(2-(2-benzoyl hydrazinyl)-4-oxothiazolidine) Acetate Derivatives by Darehkordi, Ali, Ghazi, Somayeh

“…Hydrazine, carbothioamide derivatives 2, 3, and 4 were synthesized by the condensation of 1, 3, 5-tri carbonyl tri chloride, Terephthaloyl dichloride, and 1,…”
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Urease: A highly biocompatible catalyst for switchable Biginelli reaction and synthesis of 1,4-dihydropyridines from the in situ formed ammonia by Tamaddon, Fatemeh, Ghazi, Somayeh

“…Urease is a superior biocompatible catalyst for switching from the Biginelli reaction to urea-based synthesis of 1,4-dihydropyridines in water, where 100%…”
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An enzymatic route to the synthesis of tricyclic fused hexahydrofuranofuran P2-Ligand for a series of highly potent HIV-1 protease inhibitors by Ghosh, Arun K., Sharma, Ashish, Ghazi, Somayeh

“…[Display omitted] We describe a stereoselective synthesis of an optically active (1R, 3aS, 5R, 6S, 7aR)-octahydro-1,6-epoxy-isobenzo-furan-5-ol derivative…”
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Urease-catalyzed synthesis of aminocyanopyridines from urea under fully green conditions by Tamaddon, Fatemeh, Ghazi, Somayeh, Noorbala, Mohammad Reza

“…[Display omitted] •This work supports the catalytic performance of urease in organic synthesis.•This specific urease-catalyzed reaction inhibits by trace…”
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Type II c-Met inhibitors: molecular insight into crucial interactions for effective inhibition by Damghani, Tahereh, Elyasi, Maryam, Pirhadi, Somayeh, Haghighijoo, Zahra, Ghazi, Somayeh

“…The c-Met tyrosine kinase plays an important role in human cancers. Preclinical studies demonstrated that c-Met is over-expressed, mutated and amplified in a…”
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In silico screening of c-Met tyrosine kinase inhibitors targeting nucleotide and drug-substrate binding sites of ABCB1 as potential MDR reversal agents by Moosavi, Fatemeh, Damghani, Tahereh, Ghazi, Somayeh, Pirhadi, Somayeh

“…Cancer is a significant public health problem and ranks as a leading cause of death globally. Multidrug resistance (MDR) affects the therapeutic potential of…”
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Aurones and derivatives as promising New Delhi metallo-β-lactamase (NDM-1) inhibitors by Caburet, Jérémy, Verdirosa, Federica, Moretti, Matis, Roulier, Brayan, Simoncelli, Giorgia, Haudecoeur, Romain, Ghazi, Somayeh, Jamet, Hélène, Docquier, Jean-Denis, Boucherle, Benjamin, Peuchmaur, Marine

“…Bacterial resistance is undoubtedly one of the main public health concerns especially with the emergence of metallo-β-lactamases (MBLs) able to hydrolytically…”
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Exploration of P1 and P4 modifications of nirmatrelvir: Design, synthesis, biological evaluation, and X-ray structural studies of SARS-CoV-2 Mpro inhibitors by Ghosh, Arun K., Yadav, Monika, Iddum, Satyanarayana, Ghazi, Somayeh, Lendy, Emma K., Jayashankar, Uttara, Beechboard, Sydney N., Takamatsu, Yuki, Hattori, Shin-ichiro, Aamano, Masayuki, Higashi-Kuwata, Nobuyo, Mitsuya, Hiroaki, Mesecar, Andrew D.

“…We report the synthesis, biological evaluation, and X-ray structural studies of a series of SARS-CoV-2 Mpro inhibitors based upon the X-ray crystal structure…”
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Synthesis of N-aryl-2,2,2-trifluoroacetimidoyl piperazinylquinolone derivatives and their antibacterial evaluations by Darehkordi, Ali, Javanmiri, Mahmood, Ghazi, Somayeh, Assar, Shokrollah

“…N-substituted trifluoroacetimidoyl chlorides were used for synthesis of new piperazinylquinolone derivatives. These reactions provided…”
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Facile one-pot synthesis of sugar–thiazolidinone derivatives by Darehkordi, Ali, Saidi, Kazem, Ghazi, Somayeh

“…A simple, efficient, and cost-effective method for the synthesis of a series of sugar–thiazolidinone derivatives by a one-pot reaction of the corresponding…”
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