Search Results - "Geesi, Mohammed H."

Baicalin-Loaded Lipid-Polymer Hybrid Nanoparticles Inhibiting the Proliferation of Human Colon Cancer: Pharmacokinetics and In Vivo Evaluation by Riadi, Yassine, Afzal, Obaid, Geesi, Mohammed H, Almalki, Waleed H, Singh, Tanuja

“…This research work is focused on pharmacokinetic and biochemical experiments to assess baicalin-loaded lipid-polymer hybrid nanoparticles (LPHNPs) with…”
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Comparative Studies of the Dynamics Effects of BAY60-2770 and BAY58-2667 Binding with Human and Bacterial H-NOX Domains by Rehan Khalid, Rana, Tahir Ul Qamar, Muhammad, Maryam, Arooma, Ashique, Ayesha, Anwar, Farooq, H Geesi, Mohammed, Siddiqi, Abdul Rauf

“…Soluble guanylate cyclase (sGC) is a key enzyme implicated in various physiological processes such as vasodilation, thrombosis and platelet aggregation. The…”
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Limon-citrus extract as a capping/reducing agent for the synthesis of titanium dioxide nanoparticles: characterization and antibacterial activity by Ouerghi, Oussama, Geesi, Mohammed H., Riadi, Yassine, Ibnouf, Elmutasim O.

“…In this paper, we focused on the green synthesis of titanium dioxide (TiO 2 ) nanoparticles via an ecofriendly process using Citrus limon extract. Several…”
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Novel 2-Sulfanylquinazolin-4(3 H )-one Derivatives as Multi-Kinase Inhibitors and Apoptosis Inducers: A Synthesis, Biological Evaluation, and Molecular Docking Study by Altharawi, Ali, Alanazi, Mohammed M, Alossaimi, Manal A, Alanazi, Ashwag S, Alqahtani, Safar M, Geesi, Mohammed H, Riadi, Yassine

“…The discovery of multi-targeted kinase inhibitors emerged as a potential strategy in the therapy of multi-genic diseases, such as cancer, that cannot be…”
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Synthesis, Molecular Docking and β-Glucuronidase Inhibitory Potential of Indole Base Oxadiazole Derivatives by Anouar, El Hassane, Moustapha, Moustapha Eid, Taha, Muhammad, Geesi, Mohammed H, Farag, Zeinab R, Rahim, Fazal, Almandil, Noor Barak, Farooq, Rai Khalid, Nawaz, Muhammad, Mosaddik, Ashik

“…β-glucuronidase is a lysosomal glycosidase enzyme which catalyzes the extracellular matrix of cancer and normal cells and the glycosaminoglycans of the cell…”
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Design, synthesis, molecular docking, and in vitro studies of 2-mercaptoquinazolin-4(3H)-ones as potential anti-breast cancer agents by Alossaimi, Manal A., Riadi, Yassine, Alnuwaybit, Ghaida N., Md, Shadab, Alkreathy, Huda Mohammed, Elekhnawy, Engy, Geesi, Mohammed H., Alqahtani, Safar M., Afzal, Obaid

“…[Display omitted] •Quinazolinone derivatives were designed keeping Ispinesib and Idelalisib as reference structures.•Compounds 3a, 3b, 3e, 3g and 3h revealed…”
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Synergistic inhibitive effect of a hybrid zinc oxide-benzalkonium chloride composite on the corrosion of carbon steel in a sulfuric acidic solution by AlBeladi, Muntathir, Geesi, Mohammed H., Riadi, Yassine, Alahiane, Mustapha, Aljohani, Talal A., Berisha, Avni, Reka, Arianit, Kaiba, Abdellah, Ouerghi, Oussama

“…Zinc oxide and quaternary ammonium-type surfactants have been separately recognized for their anti-corrosive efficiencies. Their composite, not investigated so…”
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Water-mediated synthesis of disubstituted 5-aminopyrimidines from vinyl azides under microwave irradiation by Dehbi, Oussama, Ishak, Esam A., Bakht, Mohammed A., Geesi, Mohammed H., Alshammari, Mohammed B., Chagnault, Vincent, Kaiba, Abdellah, Lazar, Saïd, Riadi, Yassine

“…An efficient and ecofriendly method for the synthesis of disubstituted 5-aminopyrimidines from vinyl azides and urea or thiourea was developed. This reaction…”
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A simple and eco-friendly microwave mediated route the synthesis of novel antimicrobial substituted quinoline-2-thiones by Geesi, Mohammed H., AL-Hadedi, Azzam Ahmed Mohammed, Bakht, Mohammed A., Kaiba, Abdellah, Boukili, Meryem, Alshammari, Mohammed B., Dehbi, Oussama, Riadi, Yassine

“…An eco-friendly and efficient method was developed for the preparation of a new series of sulfur-containing quinolinthiones. Compounds 6a-o were synthesized…”
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Synthesis of novel ( R )-carvone-tagged thiazolidinone as anticancer leads: characterization, in vitro antiproliferative evaluation and in silico studies by Riadi, Yassine, Afzal, Obaid, Kumar, Shashank, Varadharajan, Venkatramanan, Geesi, Mohammed H

“…This work describes the successful synthesis of a series of three novel thiazolidinone-carvone-O-alkyl hybrids through a two-step approach involving…”
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Computational screening of medicinal plant phytochemicals to discover potent pan-serotype inhibitors against dengue virus by Tahir ul Qamar, Muhammad, Maryam, Arooma, Muneer, Iqra, Xing, Feng, Ashfaq, Usman Ali, Khan, Faheem Ahmed, Anwar, Farooq, Geesi, Mohammed H., Khalid, Rana Rehan, Rauf, Sadaf Abdul, Siddiqi, Abdul Rauf

“…Emergence of Dengue as one of the deadliest viral diseases prompts the need for development of effective therapeutic agents. Dengue virus (DV) exists in four…”
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Sol-gel TiO2 nanostructures single doped with copper and nickel as nanocatalysts for enhanced performance for the Liebeskind–Srogl reaction by Riadi, Yassine, Geesi, Mohammed H., Ouerghi, Oussama, Azzallou, Rachid, Dehbi, Oussama, Lazar, Saïd

“…Design of nanostructured catalytic materials plays a strategic role in the synthesis of organic compounds with outstanding physicochemical properties. In this…”
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Phytosynthesis of anatase TiO2 nanostructures using grapefruit extract for antimicrobial and catalytic applications by Ouerghi, Oussama, Geesi, Mohammed H., Riadi, Yassine, Ibnouf, Elmutasim O., Kaiba, Abdellah

“…Plant extracts have been broadly considered to be an environmentally-benign alternative for the in vitro synthesis of stable and shape-controlled metal and…”
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Synthesis, Characterization of TiO2-Based Nanostructure as Efficient Catalyst for the Synthesis of New Heterocycles Benzothiazole-Linked Pyrrolidin-2-One: Catalytic Performances Are Particle's Size Dependent by Elsanousi, Ammar, Riadi, Yassine, Ouerghi, Oussama, Geesi, Mohammed H.

“…Nano and micro-rutile TiO 2 structures were prepared via sol-gel and hydrothermal approaches, respectively. The as-prepared structures were subjected to…”
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Photocatalytic Synthesis of Quinazolinone Derivatives as Mediated by Titanium Dioxide (TiO2) Nanoparticles Greenly Synthesised via Citrus limon Juice by Riadi, Yassine, Geesi, Mohammed H., Dehbi, Oussama, Ouerghi, Oussama

“…In this study, we focused on the ultrasonic synthesis of titanium dioxide (TiO 2 ) nanoparticles via a green chemistry process using Citrus limon (lemon)…”
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Sol-gel synthesized rutile TiO2 nanoparticles loaded with cardamom essential oil: Enhanced antibacterial activity by Ouerghi, Oussama, Geesi, Mohammed H., Ibnouf, Elmutasim O., Ansari, Mohammad Javed, Alam, Pravej, Elsanousi, Ammar, Kaiba, Abdellah, Riadi, Yassine

“…Nanoparticles have been recognized as a promising alternative to overcome problems associated with antibiotic-resistant bacterial strains. In the current…”
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Microwave Irradiation-Mediated Synthesis of New Substituted Pyridopyrimidines via the Suzuki-Miyaura Coupling Reaction and Biological Evaluation by Riadi, Yassine, Geesi, Mohammed H., Dehbi, Oussama, Ibnouf, Elmutasim O.

“…In this work, an eco-friendly, effective and easy route to synthesize substituted pyridopyrimidines is reported starting from…”
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Synthesis, characterization, biological evaluation and molecular docking of a new quinazolinone-based derivative as a potent dual inhibitor for VEGFR-2 and EGFR tyrosine kinases by Riadi, Yassine, Alamri, Mubarak A., Geesi, Mohammed H., Anouar, El Hassane, Ouerghi, Oussama, Alabbas, Alhumaidi B., Alossaimi, Manal A., Altharawi, Ali, Dehbi, Oussama, Alqahtani, Safar M.

“…An efficient process for the preparation of a new ethyl 2-((3-(4-fluorophenyl)-6-methyl-4-oxo-3,4-dihydroquinazolin-2-yl)thio) acetate (5) was described. The…”
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Thiazolidinone-linked-1,2,3-triazoles with (R)-Carvone as new potential anticancer agents by Oubella, Ali, Alossaimi, Manal A, Riadi, Yassine, Bhat, Mashooq Ahmad, Bakheit, Ahmed Hassan, Taha, Mohamed Labd, Auhmani, Aziz, Morjani, Hamid, Geesi, Mohammed H, Ait Itto, Moulay Youssef

“…This study explores the cytotoxic and apoptotic effects of novel thiazolidinone-1,2,3-triazole hybrids on HT-1080, A-549, and MDA-MB-231 cancer cell lines. The…”
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Characterization and catalytic performance of Ni-Doped TiO2 as a potential heterogeneous nanocatalyst for the preparation of substituted pyridopyrimidines by Kaiba, Abdellah, Ouerghi, Oussama, Geesi, Mohammed H., Elsanousi, Ammar, Belkacem, Afif, Dehbi, Oussama, Alharthi, Abdulrahman I., Alotaibi, Mshari A., Riadi, Yassine

“…An effective and a novel synthesis route for accessing 2-substituted-pyridopyrimidines is described, starting from (2-amino-pyridin-3-yl)-methanol through the…”
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