Search Results - "Gade, Narendar Reddy"
-
1
Self-Assembly of pH-Labile Polymer Nanoparticles for Paclitaxel Prodrug Delivery: Formulation, Characterization, and Evaluation
Published in International journal of molecular sciences (05-12-2020)“…The efficacy of paclitaxel (PTX) is limited due to its poor solubility, poor bioavailability, and acquired drug resistance mechanisms. Designing paclitaxel…”
Get full text
Journal Article -
2
[18F]ONO-8430506: A novel radioligand for PET imaging of autotaxin (ATX)
Published in Bioorganic & medicinal chemistry letters (15-06-2023)“…Radioligand [18F]ONO-8430506 ([18F]8) was prepared and tested as a novel autotaxin (ATX) PET imaging agent derived from highly potent ATX inhibitor…”
Get full text
Journal Article -
3
Stereoselective formal synthesis of macrolidecore of migrastatin using late stage C–H oxidation
Published in Tetrahedron letters (07-08-2013)“…An efficient synthesis of macrolide core of migrastatin is described here by following a novel approach of Pd(II)-catalyzed late stage intramolecular C–H…”
Get full text
Journal Article -
4
A Common Synthetic Protocol for the Cyclic and Acyclic Core of Migrastatin, Isomigrastatin, and Dorrigocin via a Chiral β-Hydroxy-γ-butyrolactone Intermediate
Published in European journal of organic chemistry (01-10-2014)“…A facile synthetic route has been developed for the synthesis of the cyclic and acyclic cores of migrastatin, isomigrastatin, and dorrigocin. The common…”
Get full text
Journal Article -
5
A Common Synthetic Protocol for the Cyclic and Acyclic Core of Migrastatin, Isomigrastatin, and Dorrigocin via a Chiral [beta]-Hydroxy-[gamma]-butyrolactone Intermediate
Published in European journal of organic chemistry (01-10-2014)“…A facile synthetic route has been developed for the synthesis of the cyclic and acyclic cores of migrastatin, isomigrastatin, and dorrigocin. The common…”
Get full text
Journal Article -
6
N‑Alkyl Carbamoylimidazoles as Versatile Synthons for the Synthesis of Urea-Based PSMA Inhibitors
Published in ACS medicinal chemistry letters (13-07-2023)“…We describe N-alkyl carbamoylimidazoles as readily available and highly versatile synthons for synthesizing urea-based prostate-specific membrane antigen…”
Get full text
Journal Article -
7
Natural Product Inspired Topology Directed Synthesis of Hybrid Macrocyclic Compounds: A Simple Approach to Natural Product Analogues
Published in ChemistrySelect (Weinheim) (15-06-2018)“…Herein we report a new approach of designing natural product‐like macrolide analogues by combining the critical structural features of two different class of…”
Get full text
Journal Article -
8
1-[(4S)-4-Benzyl-2-thioxo-1,3-thia-zol-idin-3-yl]propan-1-one
Published in Acta crystallographica. Section E, Structure reports online (15-08-2009)“…The analysis of the title chiral auxiliary compound, C(13)H(15)NOS(2), has enabled the determination of the absolute configuration at the benzyl-bearing ring C…”
Get full text
Journal Article -
9
1-[(4S)-4-Benzyl-2-thioxo-1,3-thiazolidin-3-yl]propan-1-oneILS Publication No. ILS-MCO-0904
Published in Acta crystallographica. Section E, Structure reports online (01-09-2009)“…The analysis of the title chiral auxiliary compound, C13H15NOS2, has enabled the determination of the absolute configuration at the benzyl-bearing ring C atom…”
Get full text
Journal Article -
10
1-[(4S)-4-Benzyl-2-thioxo-1,3-thiazolidin-3-yl]propan-1-one1
Published in Acta crystallographica. Section E, Structure reports online (15-08-2009)“…The analysis of the title chiral auxiliary compound, C 13 H 15 NOS 2 , has enabled the determination of the absolute configuration at the benzyl-bearing ring C…”
Get full text
Journal Article