Search Results - "Foster, Bruce S"

Diastereoselective Reductive Amination of Aryl Trifluoromethyl Ketones and α-Amino Esters by Hughes, Greg, Devine, Paul N., Naber, John R., O'Shea, Paul D., Foster, Bruce S., McKay, Daniel J., Volante, R. P.

“…Reductionist art: Careful choice of the reducing agent in the reductive amination of trifluoromethyl ketones with α‐amino esters allows stereoselective access,…”
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Palladium-Catalyzed Regioselective Arylation of Imidazo[1,2-b][1,2,4]triazine:  Synthesis of an α2/ 3-Selective GABA Agonist by Gauthier, Donald R, Limanto, John, Devine, Paul N, Desmond, Richard A, Szumigala, Ronald H, Foster, Bruce S, Volante, R. P

“…A convergent, practical, and efficient synthesis of 2‘,6-difluoro-5‘-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile (1),…”
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The Expedient Synthesis of 4,2‘-Difluoro-5‘-(7-trifluoromethyl- imidazo[1,2-a]pyrimidin-3-yl)biphenyl-2-carbonitrile, a GABA α2/3 Agonist by Cameron, Mark, Foster, Bruce S, Lynch, Joseph E, Shi, Yao-Jun, Dolling, Ulf-H

“…An expedient regioselective synthesis of a GABA α2/3 agonist 1 is described. The key step is an efficient regioselective palladium-catalyzed coupling of…”
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Efficient Synthesis of Losartan, A Nonpeptide Angiotensin II Receptor Antagonist by Larsen, Robert D, King, Anthony O, Chen, Cheng Y, Corley, Edward G, Foster, Bruce S, Roberts, F. Edward, Yang, Chunhua, Lieberman, David R, Reamer, Robert A, Tschaen, David M, Verhoeven, Thomas R, Reider, Paul J, Lo, Young S, Rossano, Lucius T, Brookes, A. Sidney, Meloni, David, Moore, James R, Arnett, John F

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An Asymmetric Synthesis of 3-Aryl-1,4-oxazin-2-ones: Synthesis of a Key Intermediate of an NK1 Receptor Antagonist by N. Devine, Paul, S. Foster, Bruce, J. J. Grabowski, Edward, J. Reider, Paul

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The behavior of indene oxide in the ritter reaction: A simple route to cis-aminoindanol by Senanayake, Chris H., Roberts, F.Edward, DiMichele, Lisa M., Ryan, Kenneth M., Liu, Ji, Fredenburgh, Laura E., Foster, Bruce S., Douglas, Alan W., Larsen, Robert D., Verhoeven, Thomas R., Reider, Paul J.

“…A regio- and stereoselective synthesis of cis-1-aminoindan-2-ol via a Ritter reaction is described. A regio- and stereoselective synthesis of chiral…”
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Palladium-catalyzed regioselective arylation of imidazo[1,2-b][1,2,4]triazine: synthesis of an alpha 2/3-selective GABA agonist by Gauthier, Jr, Donald R, Limanto, John, Devine, Paul N, Desmond, Richard A, Szumigala, Jr, Ronald H, Foster, Bruce S, Volante, R P

“…A convergent, practical, and efficient synthesis of 2',6-difluoro-5'-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile (1),…”
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A stereoselective, palladium-catalyzed route to 4-oxygenated 5-alkylidenecyclopentenones and 3-oxygenated 2-alkylideneindanones by Liebeskind, Lanny S, Mitchell, David, Foster, Bruce S

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Stannylquinones. Synthesis and utilization as quinone carbanion synthetic equivalents by Liebeskind, Lanny S, Foster, Bruce S

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Diastereoselective Reductive Amination of Aryl Trifluoromethyl Ketones and α-Amino Esters by Hughes, Greg, Devine, Paul N., Naber, John R., O'Shea, Paul D., Foster, Bruce S., McKay, Daniel J., Volante, R. P.

“…Reduktionistische Kunst: Durch sorgfältige Wahl des Reduktionsmittels gelingt die reduktive Aminierung von Trifluormethylketonen mit α‐Aminosäureestern…”
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Diastereoselective Reductive Amination of Aryl Trifluoromethyl Ketones and α‐Amino Esters by Hughes, Greg, Devine, Paul N., Naber, John R., O'Shea, Paul D., Foster, Bruce S., McKay, Daniel J., Volante, R. P.

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Metal mediated routes to 5-membered rings by Liebeskind, L. S., Chidambaram, Ramakrishnan, Mitchell, D., Foster, B. S.

“…Abstract…”
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