Search Results - "Fischer, Rolf"

An Efficient Process for the Manufacture of Carmegliptin by Abrecht, Stefan, Adam, Jean-Michel, Bromberger, Ulrike, Diodone, Ralph, Fettes, Alec, Fischer, Rolf, Goeckel, Volker, Hildbrand, Stefan, Moine, Gérard, Weber, Martin

“…A short and high-yielding synthesis of carmegliptin (1) suitable for large-scale production is reported. The tricyclic core was assembled efficiently by a…”
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The Synthetic-Technical Development of Oseltamivir Phosphate Tamiflu™: A Race against Time by Stefan Abrecht, René Trussardi, Gösta Rimmler, Thomas Oberhauser, Hans-Jürgen Mair, Martin Karpf, Rolf Fischer, Heinrich Estermann, Muriel Cordon Federspiel, Ulrich Zutter

“…The clinical development of the first orally available neuraminidase inhibitor prodrug oseltamivir phosphate (Tamiflu™) proceeded very fast. In order to…”
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Industrial Synthesis of the Key Precursor in the Synthesis of the Anti-Influenza Drug Oseltamivir Phosphate (Ro 64-0796/002, GS-4104-02):  Ethyl (3R,4S,5S)-4,5-epoxy-3-(1-ethyl-propoxy)-cyclohex-1-ene-1-carboxylate by Federspiel, Muriel, Fischer, Rolf, Hennig, Michael, Mair, Hans-Jürgen, Oberhauser, Thomas, Rimmler, Gösta, Albiez, Thomas, Bruhin, Jürg, Estermann, Heinrich, Gandert, Carsten, Göckel, Volker, Götzö, Stephan, Hoffmann, Ursula, Huber, Gabriel, Janatsch, Günter, Lauper, Stephan, Röckel-Stäbler, Odette, Trussardi, Rene, Zwahlen, Andreas G

“…Starting from (−)-quinic acid, the title compound was synthesized in seven chemical steps and an overall yield of 35−38%. The route of the improved Gilead…”
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Development of a Practical and Greener Process for the Dual Leucine Zipper Kinase Inhibitor GDC-0134 Comprising Two S N Ar Reactions, Oxidation and Suzuki Coupling by Hoffmann-Emery, Fabienne, Niedermann, Katrin, Rege, Pankaj D., Konrath, Manuel, Lautz, Christian, Kraft, Anne Katrin, Steiner, Carine, Bliss, Fritz, Hell, André, Fischer, Rolf, Carrera, Diane E., Beaudry, Danial, Angelaud, Remy, Malhotra, Sushant, Gosselin, Francis

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Development of a Practical and Greener Process for the Dual Leucine Zipper Kinase Inhibitor GDC-0134 Comprising Two SNAr Reactions, Oxidation and Suzuki Coupling by Hoffmann-Emery, Fabienne, Niedermann, Katrin, Rege, Pankaj D, Konrath, Manuel, Lautz, Christian, Kraft, Anne Katrin, Steiner, Carine, Bliss, Fritz, Hell, André, Fischer, Rolf, Carrera, Diane E, Beaudry, Danial, Angelaud, Remy, Malhotra, Sushant, Gosselin, Francis

“…A sustainable second-generation process for GDC-0134 was developed with a particular focus on safety and greenness, while complying with strong specifications…”
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Overview of a Proposed Ecological Risk Assessment Process for Honey bees (Apis mellifera) and Non-Apis Bees by Moriarty, Tom, Fischer, David

“…This chapter proposes a method for estimating risk to honey bees (Apis mellifera) and non‐Apis bees from pesticides that are applied through sprays (acting on…”
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Beschäftigung ausländischer Arbeitnehmer in der Bundesrepublik (I): Eine rechtssystematische Darstellung by Fischer, Rolf

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Beschäftigung ausländischer Arbeitnehmer in der Bundesrepublik: Eine rechtssythematische Darstellung by Fischer, Rolf

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Die Internationale Arbeitsorganisation und die nichtstaatlichen Organisationen by Fischer, Rolf

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Der Europarat und die nichtstaatlichen Organisationen by Fischer, Rolf

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Entwicklungsstufen des Antisemitismus in Ungarn 1867-1939: Die Zerstörung der Magyarisch-Jüdischen Symbiose by Kieval, Hillel J., Fischer, Rolf

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Effects of clamp force in limiting dome height (LDH) test by SCHEY, J. A, FISCHER, R. F

“…The effects of specimen width and blankholder (clamp) force on LDH were investigated in tests with bare DDQ SK steel strip. Specimen width ranged from 109-143…”
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Buchbesprechungen by Fischer, Rolf, Schittenhelm, A., Reishaus, Kauffmann, Fr, Curschmann, H., Grafe, E., Ickert, Lange

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Serologie, Blutgruppen, Endokrinologie, Bakteriologie, Immunitätslehre by Krah, Pietrusky, Mayser, Ottensooser, F., Fritz-Hölder, Helene, Lang, Seggel, Karl-Ad, Belonoschkin, Meinicke, Reschke, Hartmann, Köhler, Mauss, Schultz, Werner, Jores, Haagen, Schüller, A., Auersbach, Wiethold, Fischer, Rolf, Tobler, Thauer, Müller, R., Roggenbau, Brosowski, Kafka, V., Fischer, Ö., Waelsch, Jungmichel

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