Search Results - "Falak, A."

Heterocyclic Compounds as Dipeptidyl Peptidase-IV Inhibitors with Special Emphasis on Oxadiazoles as Potent Anti-Diabetic Agents by Mohammad, Badrud Duza, Baig, Mirza Shahed, Bhandari, Neeraj, Siddiqui, Falak A, Khan, Sharuk L, Ahmad, Zubair, Khan, Farhat S, Tagde, Priti, Jeandet, Philippe

“…Dipeptidyl peptidase-IV (DPP-IV) inhibitors, often known as gliptins, have been used to treat type 2 diabetes mellitus (T2DM). They may be combined with other…”
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Fighting Antibiotic Resistance: New Pyrimidine-Clubbed Benzimidazole Derivatives as Potential DHFR Inhibitors by Haque, M Akiful, Marathakam, Akash, Rana, Ritesh, Almehmadi, Samar J, Tambe, Vishal B, Charde, Manoj S, Islam, Fahadul, Siddiqui, Falak A, Culletta, Giulia, Almerico, Anna Maria, Tutone, Marco, Khan, Sharuk L

“…The present work describes the design and development of seventeen pyrimidine-clubbed benzimidazole derivatives as potential dihydrofolate reductase (DHFR)…”
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Ethosomes: A novel drug carrier by Chauhan, Neha, Vasava, Parul, Khan, Sharuk L., Siddiqui, Falak A., Islam, Fahadul, Chopra, Hitesh, Emran, Talha Bin

“…Ethosomal systems are newer lipid vesicular carriers that have been around for 20 years, but over that period they have grown significantly as a means of…”
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An Overview of Diabetic Foot Ulcers and Associated Problems with Special Emphasis on Treatments with Antimicrobials by Baig, Mirza Shahed, Banu, Ahmadi, Zehravi, Mehrukh, Rana, Ritesh, Burle, Sushil S., Khan, Sharuk L., Islam, Fahadul, Siddiqui, Falak A., Massoud, Ehab El Sayed, Rahman, Md. Habibur, Cavalu, Simona

“…One of the most significant challenges of diabetes health care is diabetic foot ulcers (DFU). DFUs are more challenging to cure, and this is particularly true…”
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Coumarin-Based Sulfonamide Derivatives as Potential DPP-IV Inhibitors: Pre-ADME Analysis, Toxicity Profile, Computational Analysis, and In Vitro Enzyme Assay by Vawhal, Pallavi Kishor, Jadhav, Shailaja B, Kaushik, Sumit, Panigrahi, Kahnu Charan, Nayak, Chandan, Urmee, Humaira, Khan, Sharuk L, Siddiqui, Falak A, Islam, Fahadul, Eftekhari, Aziz, Alzahrani, Abdullah R, Azlina, Mohd Fahami Nur, Sarker, Md Moklesur Rahman, Ibrahim, Ibrahim Abdel Aziz

“…Recent research on dipeptidyl peptidase-IV (DPP-IV) inhibitors has made it feasible to treat type 2 diabetes mellitus (T2DM) with minimal side effects…”
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An overview of polymer surface coated synthetic quantum dots as therapeutics and sensors applications by Babu, Ancha Kishore, Raja, M. K. Mohan Maruga, Zehravi, Mehrukh, Mohammad, Badrud Duza, Anees, Mohammed Imran, Prasad, Cheepurupalli, Yahya, Barrawaz Aateka, Sultana, Rokeya, Sharma, Rohit, Singh, Jay, Khan, Khalid Ali, Siddiqui, Falak A., Khan, Sharuk L., Emran, Talha Bin

“…Quantum dots (QDs) are a class of remarkable materials that have garnered significant attention since their initial discovery. It is noteworthy to mention that…”
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Comparing two commercial domestic dog (Canis familiaris) STR genotyping kits for forensic identity calculations in a mixed‐breed dog population sample by Kanthaswamy, S., Oldt, R. F., Montes, M., Falak, A.

“…Summary Almost half of all US households own a dog (Canis familiaris). Though these household pets can attack humans and other animals, they are also…”
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Fluorescent-Nanoparticle-Impregnated Nanocomposite Polymeric Gels for Biosensing and Drug Delivery Applications by Gandla, Kumaraswamy, Kumar, K. Praveen, Rajasulochana, P, Charde, Manoj Shrawan, Rana, Ritesh, Singh, Laliteshwar Pratap, Haque, M. Akiful, Bakshi, Vasudha, Siddiqui, Falak A, Khan, Sharuk L, Ganguly, S

“…Nanocomposite polymeric gels infused with fluorescent nanoparticles have surfaced as a propitious category of substances for biomedical purposes owing to their…”
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Carotenoids: Role in Neurodegenerative Diseases Remediation by Gandla, Kumaraswamy, Babu, Ancha Kishore, Unnisa, Aziz, Sharma, Indu, Singh, Laliteshwar Pratap, Haque, Mahammad Akiful, Dashputre, Neelam Laxman, Baig, Shahajan, Siddiqui, Falak A, Khandaker, Mayeen Uddin, Almujally, Abdullah, Tamam, Nissren, Sulieman, Abdelmoneim, Khan, Sharuk L, Emran, Talha Bin

“…Numerous factors can contribute to the development of neurodegenerative disorders (NDs), such as Alzheimer's disease, Parkinson's disease, amyotrophic lateral…”
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Natural polymers as potential P-glycoprotein inhibitors: Pre-ADMET profile and computational analysis as a proof of concept to fight multidrug resistance in cancer by Gandla, Kumaraswamy, Islam, Fahadul, Zehravi, Mehrukh, Karunakaran, Anandakumar, Sharma, Indu, Haque, M. Akiful, Kumar, Sanjay, Pratyush, Kumar, Dhawale, Sachin A., Nainu, Firzan, Khan, Sharuk L., Islam, Md Rezaul, Al-Mugren, Kholoud Saad, Siddiqui, Falak A., Emran, Talha Bin, Khandaker, Mayeen Uddin

“…P-glycoprotein (P-gp) is known as the "multidrug resistance protein" because it contributes to tumor resistance to several different classes of anticancer…”
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A rapid and large volume synthesis of mono-, di-, tri-, and tetra-substituted imidazole derivatives via ultrasonic radiation-driven technique by Shaikh, Mohd Sayeed, Kale, Mayura A., Zehravi, Mehrukh, Unnisa, Aziz, Haque, M. Akiful, Kumar, Kusuma Praveen, Khan, Sharuk L., Ali, Syed Sarfaraz, Siddiqui, Falak A., Emran, Talha Bin, AbdElrahim, Elrashed, Khandaker, Mayeen Uddin

“…Sonochemistry under controlled conditions has proven effective in medicinal chemistry and drug development. It can substantially shorten reaction timelines…”
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Potential Epha2 Receptor Blockers Involved in Cerebral Malaria from Taraxacum officinale, Tinospora cordifolia, Rosmarinus officinalis and Ocimum basilicum: A Computational Approach by Shaikh, Mohd Sayeed, Islam, Fahadul, Gargote, Parag P., Gaikwad, Rutuja R., Dhupe, Kalpana C., Khan, Sharuk L., Siddiqui, Falak A., Tapadiya, Ganesh G., Ali, Syed Sarfaraz, Dey, Abhijit, Emran, Talha Bin

“…Cerebral malaria (CM) is a severe manifestation of parasite infection caused by Plasmodium species. In 2018, there were approximately 228 million malaria cases…”
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Surface decorated quantum dots: Synthesis, properties and role in herbal therapy by Baig, Mirza Shahed, Suryawanshi, Ravikiran Maheshrao, Zehravi, Mehrukh, Mahajan, Hitendra S, Rana, Ritesh, Banu, Ahemadi, Subramanian, Muthukumar, Kaundal, Amit Kumar, Puri, Sachin, Siddiqui, Falak A, Sharma, Rohit, Khan, Sharuk L, Chen, Kow-Tong, Emran, Talha Bin

“…Quantum dots are the serendipitous outcome of materials research. It is the tiny carbonaceous nanoparticles with diameters ranging from 1 to 10 nm. This review…”
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The Design, Synthesis, and Evaluation of Diaminopimelic Acid Derivatives as Potential dapF Inhibitors Preventing Lysine Biosynthesis for Antibacterial Activity by Shaikh, Mohd Sayeed, Kale, Mayura A., Muralidharan, V., Venkatachalam, T., Ali, Syed Sarfaraz, Islam, Fahadul, Khan, Sharuk L., Siddiqui, Falak A., Urmee, Humaira, Tapadiya, Ganesh G., Dhawale, Sachin A., Ming, Long Chiau, Ibrahim, Ibrahim Abdel Aziz, Alzahrani, Abdullah R., Sarker, Md. Moklesur Rahman, Azlina, Mohd Fahami Nur

“…We created thiazole and oxazole analogues of diaminopimelic acid (DAP) by replacing its carboxyl groups and substituting sulphur for the central carbon atom…”
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The clinical impact of HCV clearance with direct antiviral agents, in a cohort of HIV/HCV coinfected individuals by Laufer, N., Stover, S., Falak, A., Sisto, A., Martinez, A., Rolon, M.J., Pérez, H.

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Β-SITOSTEROL: ISOLATION FROM MUNTINGIA CALABURA LINN BARK EXTRACT, STRUCTURAL ELUCIDATION AND MOLECULAR DOCKING STUDIES AS POTENTIAL INHIBITOR OF SARS-CoV-2 Mpro (COVID-19) by CHAUDHARI, RAKESH N, L.KHAN, SHARUK, CHAUDHARY, RAVINDRA S, JAIN, SHIRISH P, SIDDUQUI, FALAK A

“…Objecive: A novel human coronavirus (HCoV), labelled as SARS-CoV-2 (COVID-19), causing pneumonia is spreading around the world. At present, there are no…”
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Cascade of HCV care among HIV/HCV coinfected patients by Stover, S., Laufer, N., Falak, A., Poblete, G., Noé, A. López, Martinez, A., Rolon, M.J., Pérez, H.

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Potential Epha2 Receptor Blockers Involved in Cerebral Malaria from ITaraxacum officinale/I, ITinospora cordifolia/I, IRosmarinus officinalis/I and IOcimum basilicum/I: A Computational Approach by Shaikh, Mohd Sayeed, Islam, Fahadul, Gargote, Parag P, Gaikwad, Rutuja R, Dhupe, Kalpana C, Khan, Sharuk L, Siddiqui, Falak A, Tapadiya, Ganesh G, Ali, Syed Sarfaraz, Dey, Abhijit, Emran, Talha Bin

“…Cerebral malaria (CM) is a severe manifestation of parasite infection caused by Plasmodium species. In 2018, there were approximately 228 million malaria cases…”
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Polysubstituted 2H-pyran-2-ones: A new class of hepatoprotective agents by Ram, Vishnu J, Haque, Navedul, Nath, Mahendra, Singh, Sunil K, Hussaini, Falak A, Tripathi, S.C, Shoeb, A

“…The synthesis and hepatoprotective activity of 6-aryl-3-substituted-4-methylthio-2H-pyran-2-ones ( 3, 5, 7) and the corresponding 2-thiones ( 6),…”
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The Design, Synthesis, and Evaluation of Diaminopimelic Acid Derivatives as Potential dap F Inhibitors Preventing Lysine Biosynthesis for Antibacterial Activity by Shaikh, Mohd Sayeed, Kale, Mayura A, Muralidharan, V, Venkatachalam, T, Ali, Syed Sarfaraz, Islam, Fahadul, Khan, Sharuk L, Siddiqui, Falak A, Urmee, Humaira, Tapadiya, Ganesh G, Dhawale, Sachin A, Ming, Long Chiau, Ibrahim, Ibrahim Abdel Aziz, Alzahrani, Abdullah R, Sarker, Md Moklesur Rahman, Azlina, Mohd Fahami Nur

“…We created thiazole and oxazole analogues of diaminopimelic acid (DAP) by replacing its carboxyl groups and substituting sulphur for the central carbon atom…”
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