Search Results - "Faigl Ferenc"
-
1
The route from problem to solution in multistep continuous flow synthesis of pharmaceutical compounds
Published in Bioorganic & medicinal chemistry (01-12-2017)“…[Display omitted] Recent advances in the field of continuous flow chemistry allow the multistep preparation of complex molecules such as APIs (Active…”
Get full text
Journal Article -
2
A new pyrrolidine-derived atropisomeric amino alcohol as a highly efficient chiral ligand for the asymmetric addition of diethylzinc to aldehydes
Published in Tetrahedron letters (10-12-2014)“…[Display omitted] A highly efficient pyrrolidine-derived atropisomeric amino alcohol,…”
Get full text
Journal Article -
3
Z- and E-selective Horner-Wadsworth-Emmons reactions
Published in Synthetic communications (03-07-2017)“…In the present work, we determined and evaluated the stereochemical outcome of the Horner-Wadsworth-Emmons (HWE) reaction of 2-oxoalkylphosphonates with…”
Get full text
Journal Article -
4
A novel and convenient method for the preparation of 5-(diphenylmethylene)-1 H -pyrrol-2(5 H )-ones; synthesis and mechanistic study
Published in Tetrahedron (01-09-2016)Get full text
Journal Article -
5
Racemization-free synthesis of atropisomeric 1-phenylpyrrole based diamines using diphenylphosphoryl azide
Published in Tetrahedron: asymmetry (31-07-2015)“…[Display omitted] An efficient, highly stereoconservative synthesis has been developed for the preparation of aniline derived 1-arylpyrrole-2-carboxamide…”
Get full text
Journal Article -
6
Separation of non-racemic mixtures of enantiomers: an essential part of optical resolution
Published in Organic & biomolecular chemistry (01-01-2010)“…Non-racemic enantiomeric mixtures form homochiral and heterochiral aggregates in melt or suspension, during adsorption or recrystallization, and these…”
Get more information
Journal Article -
7
Highly efficient stereoconservative syntheses of new, bifunctional atropisomeric organocatalysts
Published in ARKIVOC (29-03-2016)Get full text
Journal Article Web Resource -
8
Synthesis of new, optically active 1-(substituted aryl)pyrrole derivatives via atropisomerism directed diastereoselective metalation
Published in ARKIVOC (25-04-2015)Get full text
Journal Article Web Resource -
9
Enzyme-catalyzed kinetic resolution of N-Boc-trans-3-hydroxy-4-phenylpyrrolidine
Published in Open Chemistry (01-01-2014)Get full text
Journal Article -
10
Efficient synthesis of optically active 1-(2-carboxymethyl-6-ethylphenyl)- 1H-pyrrole-2-carboxylic acid: a novel atropisomeric 1-arylpyrrole derivative
Published in Tetrahedron: asymmetry (01-01-2009)“…An efficient synthesis and resolution of (±)-1-(2-carboxymethyl-6-ethylphenyl)- 1H-pyrrole-2-carboxylic acid has been developed for the preparation of novel…”
Get full text
Journal Article -
11
Synthesis and enantioselective rearrangement of (Z)-4-triphenylmethoxy-2,3-epoxybutan-1-ol enantiomers
Published in Chirality (New York, N.Y.) (01-03-2007)“…Efficient enzyme catalyzed kinetic resolutions of a synthetically useful chiral building block, (Z)‐4‐triphenylmethoxy‐2,3‐epoxybutan‐1‐ol, are reported. The…”
Get full text
Journal Article -
12
A rational synthesis of trans-2-(3-phenylprop-1-yl)cyclohexylamino-2-oxazoline enantiomers
Published in Tetrahedron: asymmetry (17-04-2008)“…A novel method has been developed for the synthesis of the optical antipodes of trans-2-(3-phenylprop-1-yl)cyclohexylamino-2-oxazoline 1 from racemic…”
Get full text
Journal Article -
13
Regio- and Diastereoselective Synthesis of 2‑Arylazetidines: Quantum Chemical Explanation of Baldwin’s Rules for the Ring-Formation Reactions of Oxiranes
Published in Journal of organic chemistry (04-09-2020)“…A general, scalable two-step regio- and diastereoselective method has been described for the synthesis of versatile alkaloid-type azetidines from simple…”
Get full text
Journal Article -
14
Preface to the Sixtieth Volume of Periodica Polytechnica Chemical Engineering
Published in Periodica polytechnica. Chemical engineering. (2016)“…Preface to the Sixtieth Volume of Periodica Polytechnica Chemical Engineering…”
Get full text
Journal Article -
15
Useful base promoted elaborations of oxiranyl ethers
Published in Tetrahedron (17-09-2001)“…Functionalized oxiranyl ethers can be regio- and stereoselectively converted into hydroxy oxetanes or cis-diols by treatment with organometallic bases. These…”
Get full text
Journal Article -
16
Synthesis of 8,9-dialkoxybenzodiazepines and 7,8-dialkoxyisoquinolines
Published in Journal of heterocyclic chemistry (01-11-2006)“…o‐Aroylarylacetone type 1,5‐diketone derivatives (5, 6) were synthesised from arylacetones (1) protected as 1,3‐dioxolanes (4) through directed ortho…”
Get full text
Journal Article -
17
Continuous end-to-end production of solid drug dosage forms: Coupling flow synthesis and formulation by electrospinning
Published in Chemical engineering journal (Lausanne, Switzerland : 1996) (15-10-2018)“…[Display omitted] •Coupling flow synthesis with drug formulation via electrospinning.•First presentation of the two-step flow synthesis of acetylsalicylic…”
Get full text
Journal Article -
18
Copper-facilitated Suzuki-Miyaura coupling for the preparation of 1,3-dioxolane-protected 5-arylthiophene-2-carboxaldehydes
Published in Tetrahedron (19-04-2018)“…5-Formyl-2-thiopheneboronic acid is a widely used building block for the synthesis of diverse structures, however, due to a significant instability its…”
Get full text
Journal Article -
19
Access to Fluorazones by Intramolecular Dehydrative Cyclization of Aromatic Tertiary Amides: A Synthetic and Mechanistic Study
Published in Journal of organic chemistry (16-02-2018)“…An efficient synthesis has been developed for the preparation of 9H-pyrrolo[1,2-a]indol-9-ones (fluorazones) from readily available anthranilic acid…”
Get full text
Journal Article -
20
A practical process for the preparation of bis(2,2,2-trifluoroethyl) 2-oxoalkylphosphonates by acylation with carboxylic esters
Published in Tetrahedron letters (19-08-2015)“…[Display omitted] The preparation of bis(2,2,2-trifluoroethyl) 2-oxoalkylphosphonates by the acylation of bis(2,2,2-trifluoroethyl) methylphosphonate was…”
Get full text
Journal Article