Search Results - "FAUST, K. A"

Potent, orally active imidazo[4,5-b]pyridine-based angiotensin II receptor antagonists by Mantlo, Nathan B, Chakravarty, Prasun K, Ondeyka, Debra L, Siegl, Peter K. S, Chang, Raymond S, Lotti, Victor J, Faust, Kristie A, Schorn, Terry W, Chen, Tsing Bau

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Nonpeptide angiotensin II antagonists derived from 1H-pyrazole-5-carboxylates and 4-aryl-1H-imidazole-5-carboxylates by Ashton, Wallace T, Hutchins, Steven M, Greenlee, William J, Doss, George A, Chang, Raymond S. L, Lotti, Victor J, Faust, Kristie A, Chen, Tsing Bau, Zingaro, Gloria J

“…Two series of potential angiotensin II antagonists derived from carboxyl-functionalized "diazole" heterocycles have been prepared and evaluated. Initially, a…”
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Nonpeptide angiotensin II antagonists derived from 4H-1,2,4-triazoles and 3H-imidazo[1,2-b][1,2,4]triazoles by Ashton, Wallace T, Cantone, Christine L, Chang, Linda L, Hutchins, Steven M, Strelitz, Robert A, MacCoss, Malcolm, Chang, Raymond S. L, Lotti, Victor J, Faust, Kristie A

“…By a variety of synthetic routes, we have synthesized a series of 3,4,5-trisubstituted 4H-1,2,4-triazoles and a related series of…”
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The acute effects of whole-body vibration on gait parameters in adults with cerebral palsy by Dickin, D C, Faust, K A, Wang, H, Frame, J

“…As adults with cerebral palsy (CP) are surviving longer, interventions are needed to reduce spasticity and increase strength to improve mobility and life…”
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A potent, orally active, balanced affinity angiotensin II AT1 antagonist and AT2 binding inhibitor by de Laszlo, Stephen E, Quagliato, Carol S, Greenlee, William J, Patchett, Arthur A, Chang, Raymond S. L, Lotti, Victor J, Chen, Tsing Bau, Scheck, Stacey A, Faust, Kristi A

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A highly potent, orally active imidazo-[4,5-b]pyridine biphenylacylsulfonamide (MK-996;L-159,282) : a new AT1-selective angiotensin II receptor antagonist by CHAKRAVARTY, P. K, NAYLOR, E. M, SCHORN, T. W, SCHAFFER, L. W, BROTEN, T. P, SIEGL, P. K. S, PATCHETT, A. A, GREENLEE, W. J, CHEN, A, CHANG, R. S. L, TSING-BAU CHEN, FAUST, K. A, LOTTI, V. J, KIVLIGHN, S. D, GABLE, R. A, ZINGARO, G. J

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Novel and potent gastrin and brain cholecystokinin antagonists from Streptomyces olivaceus. Taxonomy, fermentation, isolation, chemical conversions, and physico-chemical and biochemical properties by Lam, Y K, Bogen, D, Chang, R S, Faust, K A, Hensens, O D, Zink, D L, Schwartz, C D, Zitano, L, Garrity, G M, Gagliardi, M M

“…The discovery and physico-chemical characterization of three novel and minor virginiamycin M1 analogs as potent gastrin antagonists from a culture of a strain…”
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Triazolinone Biphenylsulfonamide Derivatives as Orally Active Angiotensin II Antagonists with Potent AT1 Receptor Affinity and Enhanced AT2 Affinity by Ashton, Wallace T, Chang, Linda L, Flanagan, Kelly L, Hutchins, Steven M, Naylor, Elizabeth M, Chakravarty, Prasun K, Patchett, Arthur A, Greenlee, William J, Chen, Tsing-Bau

“…Several series of 2,4-dihydro-2,4,5-trisubstituted-3H-1,2,4-triazol-3-ones with acidic sulfonamide replacements of tetrazole at the 2'-position of the…”
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Triazolinones as nonpeptide angiotensin II antagonists. 1. Synthesis and evaluation of potent 2,4,5-trisubstituted triazolinones by Chang, Linda L, Ashton, Wallace T, Flanagan, Kelly L, Strelitz, Robert A, MacCoss, Malcolm, Greenlee, William J, Chang, Raymond S. L, Lotti, Victor J, Faust, Kristie A

“…A series of 2,4-dihydro-2,4,5-trisubstituted-3H-1,2,4-triazol-3-ones was prepared via several synthetic routes and evaluated as AII receptor antagonists in…”
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Two angiotensin II binding sites in rat brain revealed using [125I]Sar1, Ile8-angiotensin II and selective nonpeptide antagonists by Chang, R S, Lotti, V J, Chen, T B, Faust, K A

“…[125I]Sar1, Ile8 angiotensin II labeled two distinct binding sites in rat brain. The displacement potencies of WL-19, a selective ligand for the angiotensin II…”
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AT1 selective angiotensin II antagonists with phenoxyphenylacetic acid as a biphenyl replacement part I by Fitch, K.J., Walsh, T.F., Patchett, A.A., Chang, R.S.L., Siegl, P.K.S., Faust, K.A., Chen, T.-B., Lotti, V.J., Kivlighn, S.D., Zingaro, G.J., Greenlee, W.J.

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Triazolinones as nonpeptide angiotensin II antagonists. I: Synthesis and evaluation of potent 2,4,5-trisubstituted triazolinones by CHANG, L. L, ASHTON, W. T, BUNTING, P, ZINGARO, G. J, KIVLIGHN, S. D, SIEGL, P. K. S, FLANAGAN, K. L, STRELITZ, R. A, MACCOSS, M, GREENLEE, W. J, CHANG, R. S. L, LOTTI, V. J, FAUST, K. A, TSING-BAU CHEN

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