Search Results - "Ezumi, Kiyoshi"
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Quantitative Structure-Activity Relationships of Antibacterial Agents, 7-Heterocyclic Amine Substituted 1-Cyclopropyl-6, 8-difluoro-4-oxoquinoline-3-carboxylic Acids
Published in Chemical & pharmaceutical bulletin (01-01-1993)“…Quantitative structure-activity relationships (QSAR) of various 7-(3-substituted-azetidin-1-yl)-1-cyclopropyl-6, 8-difluoro-1,…”
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2
Intramolecular orbital interactions in triptycene studied by photoelectron spectroscopy
Published in Journal of the American Chemical Society (01-04-1983)Get full text
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3
Anti-Human IgE Monoclonal Antibodies Recognizing Epitopes Related to the Binding Sites of High and Low Affinity IgE Receptors
Published in MICROBIOLOGY and IMMUNOLOGY (01-01-1994)“…Anti-human IgE monoclonal antibodies (mAbs) were produced and eight clones recognizing epitopes on native IgE were selected. Epitopes were mapped by a…”
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4
Simultaneous Determination of Acid Dissociation Constants and True Partition Coefficients by Analysis of the Apparent Partition Coefficients. II. Dibasic Acid and Diacidic Base
Published in Chemical & pharmaceutical bulletin (1980)“…The simultaneous determination of acid dissociation constants (pKa) and true partition coefficients (P) of a dibasic acid and a diacidic base was achieved by…”
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5
Electronic structures of carbazole and indole and the solvent effects on the electronic spectra
Published in Theoretica Chimica Acta (1964)Get full text
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6
Steric Parameters Useful for the Study of Quantitative Structure-Activity Relationships : Calculation by Means of a Through-Space Interaction Model
Published in Chemical & pharmaceutical bulletin (1982)“…Various steric parameters used for the analysis of quantitative structure-activity relationships (QSAR) were examined in relation to CNDO/2 molecular orbital…”
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7
Stretching vibration of nitro and N-oxide groups of the anion radicals of 4-nitropyridine N-oxide and related nitro compounds
Published in Journal of physical chemistry (1952) (01-05-1970)Get full text
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8
In Vitro Effects of Various Heterocyclic Thiol Compounds and β-Lactam Antibiotics on Vitamin K-Dependent γ-Glutamylcarboxylation Activity in Liver Microsomes
Published in Japanese journal of pharmacology (1988)“…The in vitro effect of N-methyltetrazolethiol (NMTT), one of the common substituents at the 3'-position of the cephem in various β-lactam antibiotics, on liver…”
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9
Electronic spectra of the anion radicals of heterocyclic amine N-oxides and related substances
Published in Journal of physical chemistry (1952) (01-04-1976)Get full text
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10
Molecular Orbital Study of the Nitrosation of Active Methyl and Methylene Groups of Pyridine and Pyrimidine Derivatives
Published in Chemical & pharmaceutical bulletin (01-01-1980)“…The reactivity of active methyl and methylene groups of nitrogen-containing hetero-aromatics with alkyl nitrite in the presence of an amide ion is discussed in…”
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11
In Vitro Effects of Various Heterocyclic Thiol Compounds and β-Lactam Antibiotics on Vitamin K-Dependent γ-Glutamylcarboxylation Activity in Liver Microsomes
Published in Japanese journal of pharmacology (01-01-1988)“…The in vitro effect of N-methyitetrazoiethiol (NMTT), one of the common substituents at the 3’-position of the cephem in various β-lactam antibiotics, on liver…”
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12
Computer-aided molecular modeling of a thromboxane receptor antagonist S-145 and its related compounds
Published in Journal of medicinal chemistry (01-04-1990)“…Conformational analyses on thromboxane A2 (TxA2), its receptor agonist, U-46619, and its receptor antagonist, sulotroban, were carried out by molecular…”
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13
Synthesis and antibacterial activities of novel oxazine and thiazine ring‐fused tricyclic quinolonecarboxylic acids: 10‐(Alicyclic amino)‐9‐fluoro‐7‐oxo‐7 H ‐pyrido[1,2,3‐ de ][1,4]benzoxazine‐6‐carboxylic acids and the corresponding 1‐thia congeners
Published in Journal of heterocyclic chemistry (01-06-1991)“…Several analogs 4 and 5 of Ofloxacin ( 1 ) which contain the oxazine and thiazine rings fused with a quinolone carboxylic acid moiety, respectively, were…”
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14
Synthesis and antibacterial activities of novel oxazine and thiazine ring-fused tricyclic quinolonecarboxylic acids: 10-(Alicyclic amino)-9-fluoro-7-oxo-7H-pyrido[1,2,3-de][1,4]benzoxazine-6-carboxylic acids and the corresponding 1-thia congeners
Published in Journal of heterocyclic chemistry (01-06-1991)“…Several analogs 4 and 5 of Ofloxacin (1) which contain the oxazine and thiazine rings fused with a quinolone carboxylic acid moiety, respectively, were…”
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15
Synthesis and substituent effects on antibacterial activity, alkaline hydrolysis rates, and infrared absorption frequencies of some cephem analogs related to latamoxef (moxalactam)
Published in Journal of medicinal chemistry (01-11-1983)“…Relationships between intrinsic antibacterial activity and beta-lactam reactivity of 7 beta-[(4-hydroxyphenyl)acetyl]amino- and 7…”
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16
Steric Parameters Useful for the Study of Quantitative Structure-Activity Relationships
Published in Chemical & pharmaceutical bulletin (01-02-1982)“…Various steric parameters used for the analysis of quantitative structure-activity relationships (QSAR) were examined in relation to CNDO/2 molecular orbital…”
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17
Simultaneous Determination of Acid Dissociation Constants and True Partition Coefficients by Analyses of the Apparent Partition Coefficients. I
Published in Chemical & pharmaceutical bulletin (1980)“…Since the partition coefficient P and the dissociation constant pKa are important in studies of structure-activity relationships, the pH dependence of the…”
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