Search Results - "Ewenson, A"
-
1
Effect of substance P on rat gastrointestinal transit
Published in Digestive diseases and sciences (1988)“…The in vivo effect of substance P and related peptide analogs on gastrointestinal transit in unanesthetized rats was studied. Fasted male rats were given…”
Get full text
Conference Proceeding Journal Article -
2
Small Molecules That Dramatically Alter Multidrug Resistance Phenotype by Modulating the Substrate Specificity of P-Glycoprotein
Published in Proceedings of the National Academy of Sciences - PNAS (20-11-2001)“…By screening a chemical library for the compounds protecting cells from adriamycin (Adr), a series of small molecules was isolated that interfered with the…”
Get full text
Journal Article -
3
N-[Chloro(dimethylamino)methylene]- N-methylmethanaminium chloride (TMUCl Cl), the reagent of choice for the solid-phase synthesis of anilides
Published in Tetrahedron letters (08-08-2005)“…An effective solid-phase preparation of anilides from supported carboxylic acids is described by their activation as the corresponding acid chlorides with…”
Get full text
Journal Article -
4
“One-Pot” Preparation of N-Carbamate Protected Amino Acids via the Azide
Published in Organic process research & development (01-11-2004)“…A convenient and efficient method for the preparation of fluorenylmethyloxycarbonyl (Fmoc) and allyloxycarbonyl (Alloc) amino acids is proposed. This method is…”
Get full text
Journal Article -
5
Dehydro keto methylene and keto methylene analogues of substance P: synthesis and biological activity
Published in Journal of medicinal chemistry (01-02-1988)“…The synthesis of dehydro keto methylene and keto methylene analogues of substance P using classical peptide synthesis is described. The following analogues…”
Get full text
Journal Article -
6
Ketomethylene pseudopeptide analogs of substance P: synthesis and biological activity
Published in Journal of medicinal chemistry (01-02-1986)“…Two pseudopeptide analogues [Bz-(RS)Phe8 psi (COCH2)Gly9]SP8-11 (I) and [pGlu6,(RS)Phe8 psi (COCH2)Gly9]SP6-11 (II) of the substance P related C-terminal…”
Get full text
Journal Article -
7
Synthetic probes for the alpha-factor receptor
Published in Biopolymers (01-01-1990)“…The binding of the tridecapeptide yeast mating pheromone, alpha-factor, to its receptor represents an excellent model for the investigation of peptide…”
Get more information
Journal Article -
8
Solution phase synthesis of Saccharomyces cerevisiae a-mating factor and its analogs
Published in International journal of peptide and protein research (01-10-1990)“…The solution phase synthesis of the Saccharomyces cerevisiae a-mating factor and nonfarnesylated and nonmethylated a-factor analogs are reported. The a-factor,…”
Get more information
Journal Article -
9
Inhibition of substance P degradation in rat brain preparations by peptide hydroxamic acids
Published in European journal of biochemistry (01-07-1985)“…A peptidase activity of rat diencephalon membranes, which acts on the C‐terminal hexapeptide sequence of substance P, was characterized using the radiolabeled…”
Get full text
Journal Article -
10
Synthesis of biologically active analogs of the dodecapeptide a-factor mating pheromone of Saccharomyces cerevisiae
Published in International journal of peptide and protein research (01-03-1990)“…A number of dodecapeptides with the sequence YIIKGVFWDPAC were synthesized using solid phase peptide synthesis. The purity of the crude cleavage product was…”
Get more information
Journal Article