Search Results - "Estrada‐Soto, Samuel"

Ursolic acid derivatives as potential antidiabetic agents: In vitro, in vivo, and in silico studies by Guzmán‐Ávila, Ricardo, Flores‐Morales, Virginia, Paoli, Paolo, Camici, Guido, Ramírez‐Espinosa, Juan José, Cerón‐Romero, Litzia, Navarrete‐Vázquez, Gabriel, Hidalgo‐Figueroa, Sergio, Yolanda Rios, Maria, Villalobos‐Molina, Rafael, Estrada‐Soto, Samuel

“…Hit, Lead & Candidate Discovery Protein tyrosine phosphatase 1B (PTP‐1B) has attracted interest as a novel target for the treatment of type 2 diabetes, this…”
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Vasorelaxant and antioxidant activity of some medicinal plants from Campeche, Mexico by Aguirre Crespo, Francisco, Pérez, Elias, Valdovinos Estrella, Janice, Maldonado Velazquez, Maria, Ortega Morales, Benjamin, Crecencio, Pedro, Nuñez, Emanuel, Estrada Soto, Samuel

“…Context: Brosimum alicastrum, Cnidoscolus chayamansa, Tradescantia spathacea, Turnera diffusa, Manilkara zapota, and Jatropha gaumeri are medicinal plants…”
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Acute and subacute antidiabetic studies of ENP‐9, a new 1,5‐diarylpyrazole derivative by Hernández‐Vázquez, Eduardo, Young‐Peralta, Sandra, Cerón‐Romero, Litzia, García‐Jiménez, Sara, Estrada‐Soto, Samuel

“…Objectives To explore the antihyperglycaemic and antidiabetic effects and to determine the acute toxicity of…”
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Tilianin content and morphological characterization of colchicine-induced autotetraploids in Agastache mexicana by Martínez-Aguilar, Angélica, Villanueva Sánchez, Evert, Valencia-Díaz, Susana, Estrada-Soto, Samuel E., Napsucialy-Mendivil, Selene, Barba-Gonzalez, Rodrigo, Alia-Tejacal, Iran, Arellano-García, José de Jesús, Villegas Torres, Oscar Gabriel, Cruz Torres, Karla Catalina, Perea-Arango, Irene

“…BackgroundAgastache mexicana Linton & Epling subsp. mexicana (Lamiaceae) is an aromatic medicinal plant, characterized by a high concentration of tilianin, a…”
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Functional mechanism of tracheal relaxation, antiasthmatic, and toxicological studies of 6‐hydroxyflavone by Flores‐Flores, Angélica, Estrada‐Soto, Samuel, Millán‐Pacheco, César, Bazán‐Perkins, Blanca, Villalobos‐Molina, Rafael, Moreno‐Fierros, Leticia, Hernández‐Pando, Rogelio, García‐Jiménez, Sara, Rivera‐Leyva, Julio César

“…Previously, we described tracheal rat rings relaxation by several flavonoids, being 6‐hydroxyflavone (6‐HOF) the most active derivative of the series. Thus,…”
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Methyl jasmonate and salicylic acid enhanced the production of ursolic and oleanolic acid in callus cultures of Lepechinia Caulescens by Vergara Martínez, Víctor, Estrada-Soto, Samuel, Arellano-García, José, Rivera-Leyva, Julio, Castillo-España, Patricia, Flores, Angélica, Cardoso-Taketa, Alexandre, Perea-Arango, Irene

“…Background: The production of triterpenes from plants for pharmacological purposes varies in concentration, due to genetic and environmental factors. In vitro…”
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Methyl jasmonate enhances ursolic, oleanolic and rosmarinic acid production and sucrose induced biomass accumulation, in hairy roots of Lepechinia caulescens by Vergara-Martínez, Victor M, Estrada-Soto, Samuel E, Valencia-Díaz, Susana, Garcia-Sosa, Karlina, Peña-Rodríguez, Luis Manuel, Arellano-García, José de Jesús, Perea-Arango, Irene

“…Ursolic (UA), oleanolic (OA) and rosmarinic (RA) acids are bioactive metabolites found in that have generated interest for their health benefits, which include…”
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Vasorelaxant activity of extracts obtained from Apium graveolens:Possible source for vasorelaxant molecules isolation with potential antihypertensive effect by Vergara-Galicia Jorge Jimenez-Ramirez Luis Angel Tun-Suarez Adrian Aguirre-Crespo Francisco Salazar-Gomez Anuar Estrada-Soto Samuel Sierra-Ovando Angel Hernandez-Nunez Emmanuel

“…Objective:To investigate the vasorelaxant effect of organic extracts from Apium graveolens(A.graveolens)which is a part of a group of plants subjected to…”
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Tracheal relaxation of five medicinal plants used in Mexico for the treatment of several diseases by Sánchez-Recillas, Amanda, Mantecón-Reyes, Paul, Castillo-España, Patricia, Villalobos-Molina, Rafael, Ibarra-Barajas, Maximiliano, Estrada-Soto, Samuel

“…To assess the relaxant effect of several organic extracts obtained from Agastache mexicana (A. mexicana), Cochlospermum vitifolium (C. vitifolium), Cordia…”
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Regulation of Myosin Light-Chain Phosphatase Activity to Generate Airway Smooth Muscle Hypercontractility by Álvarez-Santos, Mayra D., Álvarez-González, Marisol, Estrada-Soto, Samuel, Bazán-Perkins, Blanca

“…Smooth muscle is a central structure involved in the regulation of airway tone. In addition, it plays an important role in the development of some pathologies…”
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Novel mucoadhesive PLGA-PVM/MA micro-nanocomposites loaded with felodipine intended for pulmonary administration by nebulization by Isabel, Cruz-Zazueta, Luis, Arias-Durán, Samuel, Estrada-Soto, Elizabeth, Piñón-Segundo, Dea, Herrera-Ruiz, Sergio, Alcalá-Alcalá

“…[Display omitted] Poly(latic-co-glycolic) acid (PLGA) nanoparticles loaded with felodipine (FEL) were embedded in a mucoadhesive matrix of poly (methyl vinyl…”
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Chrysin Induces Antidiabetic, Antidyslipidemic and Anti-Inflammatory Effects in Athymic Nude Diabetic Mice by Ramírez-Espinosa, Juan José, Saldaña-Ríos, Johann, García-Jiménez, Sara, Villalobos-Molina, Rafael, Ávila-Villarreal, Gabriela, Rodríguez-Ocampo, Angélica Nallelhy, Bernal-Fernández, Germán, Estrada-Soto, Samuel

“…Extensive knowledge of diabetes and its complications is helpful to find new drugs for proper treatment to stop degenerative changes derived from this disease…”
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Semisynthesis, ex vivo evaluation, and SAR studies of coumarin derivatives as potential antiasthmatic drugs by Sánchez-Recillas, Amanda, Navarrete-Vázquez, Gabriel, Hidalgo-Figueroa, Sergio, Rios, María Yolanda, Ibarra-Barajas, Maximiliano, Estrada-Soto, Samuel

“…Asthma is a chronic inflammatory disorder that causes contraction in the smooth muscle of the airway and blocking of airflow. Reversal the contractile process…”
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Vasorelaxant Activity of Salvia hispanica L.: Involvement of the Nitric Oxide Pathway in Its Pharmacological Mechanism by Herbert-Doctor, Luis A., Sánchez-Recillas, Amanda, Ortiz-Andrade, Rolffy, Hernández-Núñez, Emanuel, Araujo-León, Jesús Alfredo, Coral-Martínez, Tania Isolina, Cob-Calan, Nubia Noemi, Segura Campos, Maira Rubi, Estrada-Soto, Samuel

“…Salvia hispanica L., commonly known as chía, and its seeds have been used since ancient times to prepare different beverages. Due to its nutritional content,…”
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Design, Synthesis and in Combo Antidiabetic Bioevaluation of Multitarget Phenylpropanoic Acids by Colín-Lozano, Blanca, Estrada-Soto, Samuel, Chávez-Silva, Fabiola, Gutiérrez-Hernández, Abraham, Cerón-Romero, Litzia, Giacoman-Martínez, Abraham, Almanza-Pérez, Julio Cesar, Hernández-Núñez, Emanuel, Wang, Zhilong, Xie, Xin, Cappiello, Mario, Balestri, Francesco, Mura, Umberto, Navarrete-Vazquez, Gabriel

“…We have synthesized a small series of five 3-[4-arylmethoxy)phenyl]propanoic acids employing an easy and short synthetic pathway. The compounds were tested in…”
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Metronidazole and Secnidazole Carbamates: Synthesis, Antiprotozoal Activity, and Molecular Dynamics Studies by Rocha-Garduño, Genaro, Hernández-Martínez, Norma Angélica, Colín-Lozano, Blanca, Estrada-Soto, Samuel, Hernández-Núñez, Emanuel, Prieto-Martínez, Fernando Daniel, Medina-Franco, José L, Chale-Dzul, Juan Bautista, Moo-Puc, Rosa, Navarrete-Vázquez, Gabriel

“…We prepared a series of 10 carbamates derivatives based on two common antiprotozoal drugs: metronidazole ( - ) and secnidazole ( - ). The compounds were tested…”
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Spasmolytic effect of Mentha pulegium L. involves ionic flux regulation in rat ileum strips by Estrada-Soto, Samuel, González-Maldonado, Dalia, Castillo-España, Patricia, Aguirre-Crespo, Francisco, Sánchez-Salgado, Juan Carlos

“…Mentha pulegium is common known as “poleo” and used for the treatment of diarrhea, headache and cough in Mexican traditional medicine. Organic extracts from…”
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The α1D-adrenoreceptor antagonist BMY 7378 reverses cardiac hypertrophy in spontaneously hypertensive rats by Rodríguez, Jessica E., Saucedo-Campos, Alberto D., Vega, Ana V., Ramírez-Hernández, Diana, Martínez-Aguilar, Luisa, Jiménez-Flores, J. Rafael, Andrade-Jorge, Erik, Estrada-Soto, Samuel E., Villalobos-Molina, Rafael, Touyz, Rhian M., Gallardo-Ortíz, Itzell A.

“…OBJECTIVE:The α1D-adrenoreceptor (α1D-AR) is involved in angiotensin II-induced vascular remodeling and hypertension. Whether α1D-AR plays a role in…”
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Relaxant Activity of 4H-Pyran and 1,6-Dihydropyridine Derivatives on Isolated Rat Trachea by Estrada-Soto, Samuel, Alemán-Pantitlán, Soledad, Gaona-Tovar, Emmanuel, Hernández-Borja, Fernando, Alcaraz, Yolanda, Villalobos-Molina, Rafael, Vázquez, Miguel A.

“…Derivatives of 4H-pyrans and 1,6-dihydropyridines have generated considerable attention due to their interesting biological and therapeutic values. Their…”
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Synthesis, In Vitro, In Vivo and In Silico Antidiabetic Bioassays of 4-Nitro(thio)phenoxyisobutyric Acids Acting as Unexpected PPARγ Modulators: An In Combo Study by Colin-Lozano, Blanca, Torres-Gomez, Héctor, Hidalgo-Figueroa, Sergio, Chávez-Silva, Fabiola, Estrada-Soto, Samuel, Almanza-Pérez, Julio Cesar, Navarrete-Vazquez, Gabriel

“…Four isobutyric acids (two nitro and two acetamido derivatives) were prepared in two steps and characterized using spectral analysis. The mRNA concentrations…”
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