Search Results - "Enguix, M. J."

New Serotonin 5-HT2A, 5-HT2B, and 5-HT2C Receptor Antagonists:  Synthesis, Pharmacology, 3D-QSAR, and Molecular Modeling of (Aminoalkyl)benzo and Heterocycloalkanones by Brea, José, Rodrigo, Jordi, Carrieri, Antonio, Sanz, Ferran, Cadavid, M. Isabel, Enguix, María J, Villazón, María, Mengod, Guadalupe, Caro, Yolanda, Masaguer, Christian F, Raviña, Enrique, Centeno, Nuria B, Carotti, Angelo, Loza, M. Isabel

“…A series of 52 conformationally constrained butyrophenones have been synthesized and pharmacologically tested as antagonists at 5-HT2A, 5-HT2B, and 5-HT2C…”
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Differential regulation of rat peripheral 5-HT(2A) and 5-HT(2B) receptor systems: influence of drug treatment by Enguix, M J, Sánchez, L, Villazón, M, Brea, J, Tristán, H, Caruncho, H J, Cadavid, M I, Loza, M I

“…Most studies of 5-HT(2) receptor regulation have been carried out on the central nervous system (CNS) (which expresses 5-HT(2A) and 5-HT(2C) receptors); very…”
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Differential regulation of rat peripheral 5-HT 2A and 5-HT 2B receptor systems: influence of drug treatment by Enguix, M. J., S nchez, L., Villaz n, M., Brea, J., Trist n, H., Caruncho, H. J., Cadavid, M. I., Loza, M. I.

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Conformationally constrained butyrophenones with affinity for dopamine (D(1), D(2), D(4)) and serotonin (5-HT(2A), 5-HT(2B), 5-HT(2C)) receptors: synthesis of aminomethylbenzo[b]furanones and their evaluation as antipsychotics by Raviña, E, Casariego, I, Masaguer, C F, Fontenla, J A, Montenegro, G Y, Rivas, M E, Loza, M I, Enguix, M J, Villazon, M, Cadavid, M I, Demontis, G C

“…A series of novel conformationally restricted butyrophenones (6-aminomethyl-4,5,6,7-tetrahydrobenzo[b]furan-4-ones bearing…”
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Different pharmacological properties of two equipotent antagonists (Clozapine and Rauwolscine) for 5-HT2B receptors in rat stomach fundus by VILLAZON, Maria, ENGUIX, Maria José, TRISTAN, Helena, HONRUBIA, Maria Angeles, BREA, José, MAAYANI, Saul, CADAVID, Maria Isabel, LOZA, Maria Isabel

“…On the basis of the previously demonstrated constitutive activity in natural systems and the possibility of specific ligand-induced conformations, the aims of…”
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Conformationally Constrained Butyrophenones with Affinity for Dopamine (D1, D2, D4) and Serotonin (5-HT2A, 5-HT2B, 5-HT2C) Receptors:  Synthesis of Aminomethylbenzo[b]furanones and Their Evaluation as Antipsychotics by Raviña, Enrique, Casariego, Isabel, Masaguer, Christian F, Fontenla, José A, Montenegro, Gisela Y, Rivas, María E, Loza, M. Isabel, Enguix, Maria J, Villazon, Maria, Cadavid, M. Isabel, Demontis, Gian C

“…A series of novel conformationally restricted butyrophenones (6-aminomethyl-4,5,6,7-tetrahydrobenzo[b]furan-4-ones bearing…”
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Functional Characterization of Serotonin Receptors in Rat Isolated Aorta by Villazón, María, Padín, Juan Fernando, Cadavid, María Isabel, Enguix, María José, Tristán, Helena, Orallo, Francisco, Loza, María Isabel

“…Interactions of serotonin (5-HT) with different specific 5-HT receptors that can coexist in the same blood vessel sometimes generate opposite effects. The aim…”
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