Search Results - "Enguix, M J"
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New Serotonin 5-HT2A, 5-HT2B, and 5-HT2C Receptor Antagonists: Synthesis, Pharmacology, 3D-QSAR, and Molecular Modeling of (Aminoalkyl)benzo and Heterocycloalkanones
Published in Journal of medicinal chemistry (03-01-2002)“…A series of 52 conformationally constrained butyrophenones have been synthesized and pharmacologically tested as antagonists at 5-HT2A, 5-HT2B, and 5-HT2C…”
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Differential regulation of rat peripheral 5-HT(2A) and 5-HT(2B) receptor systems: influence of drug treatment
Published in Naunyn-Schmiedeberg's archives of pharmacology (01-08-2003)“…Most studies of 5-HT(2) receptor regulation have been carried out on the central nervous system (CNS) (which expresses 5-HT(2A) and 5-HT(2C) receptors); very…”
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Differential regulation of rat peripheral 5-HT 2A and 5-HT 2B receptor systems: influence of drug treatment
Published in Naunyn-Schmiedeberg's archives of pharmacology (01-08-2003)Get full text
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Conformationally constrained butyrophenones with affinity for dopamine (D(1), D(2), D(4)) and serotonin (5-HT(2A), 5-HT(2B), 5-HT(2C)) receptors: synthesis of aminomethylbenzo[b]furanones and their evaluation as antipsychotics
Published in Journal of medicinal chemistry (30-11-2000)“…A series of novel conformationally restricted butyrophenones (6-aminomethyl-4,5,6,7-tetrahydrobenzo[b]furan-4-ones bearing…”
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Different pharmacological properties of two equipotent antagonists (Clozapine and Rauwolscine) for 5-HT2B receptors in rat stomach fundus
Published in Biochemical pharmacology (15-09-2003)“…On the basis of the previously demonstrated constitutive activity in natural systems and the possibility of specific ligand-induced conformations, the aims of…”
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Conformationally Constrained Butyrophenones with Affinity for Dopamine (D1, D2, D4) and Serotonin (5-HT2A, 5-HT2B, 5-HT2C) Receptors: Synthesis of Aminomethylbenzo[b]furanones and Their Evaluation as Antipsychotics
Published in Journal of medicinal chemistry (30-11-2000)“…A series of novel conformationally restricted butyrophenones (6-aminomethyl-4,5,6,7-tetrahydrobenzo[b]furan-4-ones bearing…”
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Functional Characterization of Serotonin Receptors in Rat Isolated Aorta
Published in Biological & pharmaceutical bulletin (01-05-2002)“…Interactions of serotonin (5-HT) with different specific 5-HT receptors that can coexist in the same blood vessel sometimes generate opposite effects. The aim…”
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