Search Results - "Elkin, Pavel K"

Rapid Access to 2,2-Disubstituted Indolines via Dearomative Indolic-Claisen Rearrangement: Concise, Enantioselective Total Synthesis of (+)-Hinckdentine A by Baidilov, Daler, Elkin, Pavel K., Athe, Sudhakar, Rawal, Viresh H.

“…The construction of 2,2-disubstituted indolines has long presented a synthetic challenge without any general solutions. Herein, we report a robust protocol for…”
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Diels–Alder Reactions of 1‑Alkoxy-1-amino-1,3-butadienes: Direct Synthesis of 6‑Substituted and 6,6-Disubstituted 2‑Cyclohexenones and 6‑Substituted 5,6-Dihydropyran-2-ones by Elkin, Pavel K, Durfee, Nathaniel D, Rawal, Viresh H

“…We report the cycloaddition reactions of 1-alkoxy-1-amino-1,3-butadienes. These doubly activated dienes are prepared on a multigram scale from crotonic acid…”
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Three-component reactions of CF3-substituted boranes, ethyl diazoacetate and imines by Elkin, Pavel K., Levin, Vitalij V., Dilman, Alexander D., Struchkova, Marina I., Arkhipov, Dmitry E., Korlyukov, Alexander A.

“…Reactions of boranes, ethyl diazoacetate, and N-(4-methoxyphenyl)imines lead to Mannich-type products with good syn selectivity…”
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Diels-Alder reactions of fused 5-, 6- and 7-membered ring 2-vinylindoles: Synthesis of annulated tetrahydrocarbazoles by Noland, Wayland E., Herzig, Ryan J., Kumar, Honnaiah Vijay, Narina, Venkata Srinivasarao, Elkin, Pavel K., Valverde, Karen I., Kim, Briana L.

“…Scaffolds of tetrahydrocarbazoles are an important class of biologically active compounds found abundant in nature. In the present investigation,…”
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Nucleophilic fluoroalkylation of (bromomethyl)pinacolborane using silicon reagents by Levin, Vitalij V., Elkin, Pavel K., Struchkova, Marina I., Dilman, Alexander D.

“…A method for the synthesis of pinacol boronic esters bearing a fluorinated group is described. •Nucleophilic fluoroalkylation of…”
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Reactions of CF3-substituted boranes with α-diazocarbonyl compounds by Elkin, Pavel K., Levin, Vitalij V., Dilman, Alexander D., Struchkova, Marina I., Belyakov, Pavel A., Arkhipov, Dmitry E., Korlyukov, Alexander A., Tartakovsky, Vladimir A.

“…Trifluoromethylation of methyl boronic esters followed by reaction with α-diazocarbonyl compounds is described. Boranes substituted with a CF3-group can be…”
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Reactions of CF sub(3-substituted boranes with [alpha]-diazocarbonyl compounds) by Elkin, Pavel K, Levin, Vitalij V, Dilman, Alexander D, Struchkova, Marina I, Belyakov, Pavel A, Arkhipov, Dmitry E, Korlyukov, Alexander A, Tartakovsky, Vladimir A

“…Boranes substituted with a CF sub(3-group can be generated from methyl boronic esters RB(OMe)) sub(2) and Me sub(3SiCF) sub(3)/KF followed by treatment with Me…”
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Reactions of CF3-substituted boranes with α-diazocarbonyl compounds by ELKIN, Pavel K, LEVIN, Vitalij V, DILMAN, Alexander D, STRUCHKOVA, Marina I, BELYAKOV, Pavel A, ARKHIPOV, Dmitry E, KORLYUKOV, Alexander A, TARTAKOVSKY, Vladimir A

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