Search Results - "Elkanzi, Nadia A. A."

Pumice as a Novel Natural Heterogeneous Catalyst for the Designation of 3,4-Dihydropyrimidine-2-(1H)-ones/thiones under Solvent-Free Conditions by El-Lateef, Hany M. Abd, Gouda, Mohamed, Khalaf, Mai M., Shaaban, Saad, Elkanzi, Nadia A. A., Saber, El Sayed A., Abdelhamid, Antar A., Ali, Ali M.

“…In this study, pumice is used as a novel natural heterogeneous catalyst for the synthesis of 3,4-dihydropyrimidine-2-(1H)-ones/thiones via the one-pot…”
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Facile One-Pot Multicomponent Synthesis of Pyrazolo-Thiazole Substituted Pyridines with Potential Anti-Proliferative Activity: Synthesis, In Vitro and In Silico Studies by El Azab, Islam H., Bakr, Rania B., Elkanzi, Nadia A. A.

“…Pyrazolothiazole-substituted pyridine conjugates are an important class of heterocyclic compounds with an extensive variety of potential applications in the…”
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New 1,2,3-Triazole-Containing Hybrids as Antitumor Candidates: Design, Click Reaction Synthesis, DFT Calculations, and Molecular Docking Study by El Azab, Islam H, El-Sheshtawy, Hamdy S, Bakr, Rania B, Elkanzi, Nadia A A

“…In an effort to improve and achieve biologically active anticancer agents, a novel series of 1,2,3-triazole-containing hybrids were designed and efficiently…”
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Design, Synthesis, and SAR Studies of Some Novel Chalcone Derivatives for Potential Insecticidal Bioefficacy Screening on Spodoptera frugiperda (Lepidoptera: Noctuidae) by Ali, Ali M., Salah, Hanan, Gad, Mohamed A., M. A. M, Youssef, Elkanzi, Nadia A. A.

“…Spodoptera frugiperda is a species of the order Lepidoptera. It is one of the species of fall armyworm moths distinguished by its larval life stage, is found…”
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Design, Synthesis, and Antimicrobial Evaluation of New Annelated Pyrimido[2,1- c ][1,2,4]triazolo[3,4- f ][1,2,4]triazines by El Azab, Islam H, Elkanzi, Nadia A A

“…A series of 34 new pyrimido[2,1- ][1,2,4]triazine-3,4-diones were synthesized and fully characterized using IR, NMR, MS, and microanalytical analysis. In vitro…”
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Efficient and Recoverable Bio-Organic Catalyst Cysteine for Synthesis, Docking Study, and Antifungal Activity of New Bio-Active 3,4-Dihydropyrimidin-2(1H)‑ones/thiones Under Microwave Irradiation by Elkanzi, Nadia A. A., Kadry, Asmaa M., Ryad, Rasha M., Bakr, Rania B., Ali El-Remaily, Mahmoud Abd El Aleem Ali, Ali, Ali M.

“…An eco-friendly green bio-organic catalyst and low-cost 3,4-dihydropyrimidin-2­(1H)-ones/thione derivatives 4–7 have been synthesized using a high-yield,…”
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An Efficient Synthetic Approach Towards Benzo[ b ]pyrano[2,3- e ][1,4]diazepines, and Their Cytotoxic Activity by El Azab, Islam H, Elkanzi, Nadia A A

“…In search of unprecedented tri and/or tetrapod pharmacophoric conjugates, a series of 32 new 4-ethyl-1 -benzo[ ][1,4]diazepin-2(3 )-ones were synthesized and…”
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New Benzimidazole‐Based Fe (III) and Cr (III) Complexes: Characterization, Bioactivity Screening, and Theoretical Implementations Using DFT and Molecular Docking Analysis by Elkanzi, Nadia A. A., Ali, Ali M., Albqmi, Mha, Abdou, Aly

“…Two new Fe (III) and Cr (III) complexes had been synthesized and structurally characterized. The new complexes were based on 2‐methyl‐benzimidazole (MB) and…”
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Synhesis, Molecular Docking Studies and in vitro Antimicrobial Evaluation of Novel Pyrimido[1,2-a]quinoxaline and Triazino[4,3-a]quinoxaline Derivatives by B. Bakr, Rania, A. A. Elkanzi, Nadia, A. Ghoneim, Amira, M. N. Moustafa, Shaima

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Synthesis of Chalcones Derivatives and Their Biological Activities: A Review by Elkanzi, Nadia A. A., Hrichi, Hajer, Alolayan, Ruba A., Derafa, Wassila, Zahou, Fatin M., Bakr, Rania B.

“…Chalcone derivatives are considered valuable species because they possess a ketoethylenic moiety, CO–CHCH–. Due to the presence of a reactive α,β-unsaturated…”
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New mononuclear Fe(III), Co(II), Ni(II), Cu(II), and Zn(II) complexes incorporating 4‐{[(2 hydroxyphenyl)imino]methyl}phenyl‐4‐methylbenzenesulfonate (HL): Synthesis, characterization, theoretical, anti‐inflammatory, and molecular docking investigation by Elkanzi, Nadia A. A., Ali, Ali M., Hrichi, Hajer, Abdou, Aly

“…Herein, new Fe(III), Co(II), Ni(II), Cu(II), and Zn(II) complexes incorporating 4‐{[(2‐hydroxyphenyl)imino]methyl}phenyl 4‐methylbenzenesulfonate Schiff‐base…”
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A novel colorimetric chemosensor based on 2-[(carbamothioylhydrazono) methyl]phenyl 4-methylbenzenesulfonate (CHMPMBS) for the detection of Cu(II) in aqueous medium by Hrichi, Hajer, Elkanzi, Nadia A. A., Ali, Ali M., Abdou, Aly

“…In this study, 2-[(carbamothioylhydrazono)methyl-phenyl-4-methylbenzenesulfonate (CHMPMBS) , which exhibits selective colorimetric chemosensor properties for…”
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Preparation of some novel thiazolidinones, imidazolinones, and azetidinone bearing pyridine and pyrimidine moieties with antimicrobial activity by Bakr, Rania B., Elkanzi, Nadia A. A.

“…By aiming to design new antimicrobial agents, we prepared new series of thiazolidin‐4‐ones(12a–d), imidazolin‐4‐ones(13a–d), and azetidin‐2‐ones (14a–d),…”
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A selective colorimetric chemosensor for detecting Ni(II) in aqueous solutions based on 4-[{[4-(3-chlorophenyl)-1,3-thiazol-2-yl]hydrazono}methyl]phenyl 4-methyl benzene sulfonate (CTHMBS) by Hrichi, Hajer, Ali, Ali M., Elkanzi, Nadia A. A., Abdou, Aly

“…Among the toxic heavy metals, Ni(II) can cause a variety of side effects on human health, such as allergy, cardiovascular and kidney diseases, lung fibrosis,…”
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Construction and Docking Studies of Novel Pyrimido[4,5‐b]quinolines as Antimicrobial Agents by Bakr, Rania B., El Azab, Islam H., Elkanzi, Nadia A. A.

“…In order to develop novel antimicrobial agents, we prepared quinoline bearing pyrimidine analogues 2–7, 8 a–d and 9 a–d and their structures were elucidated by…”
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Review of the recent advances of pyrazole derivatives as selective COX-2 inhibitors for treating inflammation by Ghoneim, Mohammed M, Abdelgawad, Mohamed A, Elkanzi, Nadia A A, Bakr, Rania B

“…Pyrazole heterocycle is regarded as an extremely significant agent for the therapy of inflammation. Celecoxib, lonazolac, deracoxib, and phenylbutazone are…”
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Antioxidant and Antimicrobial Potential of 1,8‐Naphthyridine Based Scaffolds: Design, Synthesis and in Silico Simulation Studies within Topoisomerase II by Elkanzi, Nadia A. A., Hrichi, Hajer, Muqbil Alsirhani, Alaa, Bakr, Rania B.

“…A series of spiro β‐Lactams (4 a–c, 7 a–c) and thiazolidinones (5 a–c, 8 a–c) possessing 1,8‐naphthyridine moiety were synthesized in this study. The structure…”
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A literature review on pharmacological aspects, docking studies, and synthetic approaches of quinazoline and quinazolinone derivatives by Ghoneim, Mohammed M., Abdelgawad, Mohamed A., Elkanzi, Nadia A. A., Parambi, Della Grace Thomas, Alsalahat, Izzeddin, Farouk, Amr, Bakr, Rania B.

“…Quinazoline and quinazolinone derivatives piqued medicinal chemistry interest in developing novel drug candidates owing to their pharmacological potential…”
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Design and Synthesis of Pyridine and Thiazole Derivatives as Eco‐friendly Insecticidal to Control Olive Pests by Elkanzi, Nadia A. A., Al‐Hazmi, Aryam Khaled Ghayad, Bakr, Rania B., Gad, Mohamed A., Abd El‐Lateef, Hany M., Ali, Ali M.

“…Treatment of p‐tosyloxybenzaldehyde (1) with ethyl cyanoacetate afforded ethyl 2‐cyano‐3‐(4‐{[(4‐methylphenyl)sulfonyl]oxy}phenyl)acrylate (2) which reacted…”
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Design, Synthesis, Molecular Modeling Study, and Antimicrobial Activity of Some Novel Pyrano[2,3‐b]pyridine and Pyrrolo[2,3‐b]pyrano[2.3‐d]pyridine Derivatives by Elkanzi, Nadia A. A., Bakr, Rania B., Ghoneim, Amira A.

“…Novel derivatives of pyrano[2,3‐b]pyridine and pyrrolo[2,3‐b]pyrano[2.3‐d]pyridine were prepared, and their structures were elucidated by spectral and…”
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