Search Results - "ERKER, T"

Simulation model of quarter milk flowrates to estimate quarter and cow milking duration and automated milking system's box duration by Silva Boloña, P., Upton, J., Cabrera, V., Erker, T., Reinemann, D.J.

“…The aims of this research were (1) to develop a model to simulate a herd of cows and quarter milk flowrates for a milking and derive quarter and udder milking…”
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The third-generation P-glycoprotein inhibitor tariquidar may overcome bacterial multidrug resistance by increasing intracellular drug concentration by LEITNER, I, NEMETH, J, FEURSTEIN, T, ABRAHIM, A, MATZNELLER, P, LAGLER, H, ERKER, T, LANGER, O, ZEITLINGER, M

“…The use of efflux pump inhibitors may be a powerful strategy to overcome transporter-mediated bacterial multidrug resistance. In the present study, we set out…”
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Trapping and dissociation of propafenone derivatives in HERG channels by Windisch, A, Timin, EN, Schwarz, T, Stork‐Riedler, D, Erker, T, Ecker, GF, Hering, S

“…BACKGROUND AND PURPOSE Human ether‐a‐go‐go related gene (HERG) channel inhibitors may be subdivided into compounds that are trapped in the closed channel…”
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Valerenic acid derivatives as novel subunit‐selective GABA A receptor ligands – in vitro and in vivo characterization by Khom, S, Strommer, B, Ramharter, J, Schwarz, T, Schwarzer, C, Erker, T, Ecker, GF, Mulzer, J, Hering, S

“…BACKGROUND AND PURPOSE Subunit‐specific modulators of γ‐aminobutyric acid (GABA) type A (GABA A ) receptors can help to assess the physiological function of…”
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Interaction of diltiazem with an intracellularly accessible binding site on Ca(V)1.2 by Shabbir, W, Beyl, S, Timin, E N, Schellmann, D, Erker, T, Hohaus, A, Hockerman, G H, Hering, S

“…Diltiazem inhibits Ca(V)1.2 channels and is widely used in clinical practice to treat cardiovascular diseases. Binding determinants for diltiazem are located…”
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Antitumor Effects of 3,3′,4,4′,5,5′-Hexahydroxystilbene in hl-60 Human Promyelocytic Leukemia Cells by Saiko, P., Horvath, Z., Murias, M., Handler, N., Jaeger, W., Erker, T., Fritzer-Szekeres, M., Szekeres, T.

“…Resveratrol (3,4′,5-trihydroxystilbene, RV) exerts remarkable cytostatic and cytotoxic effects against a multitude of human cancer cell lines. Since the…”
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Resveratrol, an Ingredient of Wine, Acts Synergistically with Ara-C and Tiazofurin in HL-60 Human Promyelocytic Leukemia Cells by Horvath, Z., Saiko, P., Illmer, C., Madlener, S., Hoechtl, T., Bauer, W., Erker, T., Jaeger, W., Fritzer-Szekeres, M., Szekeres, T.

“…Resveratrol (RV), a naturally occurring stilbene derivative, is a potent free radical scavenger causing a number of biochemical and antineoplastic effects. It…”
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Disposal of Arsenic-Laden Adsorptive Media: Economic Analysis for California by Chen, Wei-Hsiang, Erker, Benjamin T, Kanematsu, Masakazu, Darby, Jeannie L

“…Due to California’s stringent hazardous waste (HW) classification regulations, high-capacity adsorptive media (AM) used for the removal of arsenic from potable…”
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Antioxidant, prooxidant and cytotoxic activity of hydroxylated resveratrol analogues: structure–activity relationship by Murias, Marek, Jäger, Walter, Handler, Norbert, Erker, Thomas, Horvath, Zsuzsanna, Szekeres, Thomas, Nohl, Hans, Gille, Lars

“…Resveratrol ( trans-3,4′,5-trihydroxystilbene), a naturally occurring hydroxystilbene, is considered an essential antioxidative constituent of red wine…”
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Resveratrol analogues as selective cyclooxygenase-2 inhibitors: synthesis and structure–activity relationship by Murias, Marek, Handler, Norbert, Erker, Thomas, Pleban, Karin, Ecker, Gerhard, Saiko, Philipp, Szekeres, Thomas, Jäger, Walter

“…A series of hydroxylated and methoxylated trans-stilbenes were synthesized and evaluated for their ability to inhibit COX-1 and COX-2. Some of the hydroxylated…”
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Pros and cons of using resazurin staining for quantification of viable Staphylococcus aureus biofilms in a screening assay by Sandberg, Malena E., Schellmann, Denise, Brunhofer, Gerda, Erker, Thomas, Busygin, Igor, Leino, Reko, Vuorela, Pia M., Fallarero, Adyary

“…Staining of Staphylococcus aureus biofilms with 20 µM resazurin during 20 min was shown to provide a good screening assay in 96-well micro titer plates…”
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Synthesis of Novel Curcumin Analogues and Their Evaluation as Selective Cyclooxygenase-1 (COX-1) Inhibitors by Handler, Norbert, Jaeger, Walter, Puschacher, Helmut, Leisser, Klaus, Erker, Thomas

“…Curcumin, a major yellow pigment and active component of turmeric, has been shown to possess anti-inflammatory and anti-cancer activities. Recent studies have…”
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Antioxidant activity of resveratrol, piceatannol and 3,3',4,4',5,5'-hexahydroxy-trans-stilbene in three leukemia cell lines by OVESNA, Zdenka, KOZICS, Katarina, BADER, Yvonne, SAIKO, Philipp, HANDLER, Norbert, ERKER, Thomas, SZEKERES, Thomas

“…trans-Resveratrol (t-RES) is one of the most relevant and extensively investigated stilbenes with a broad spectrum of biological activities. In contrast to the…”
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Interaction of diltiazem with an intracellularly accessible binding site on Ca V 1.2 by Shabbir, W, Beyl, S, Timin, EN, Schellmann, D, Erker, T, Hohaus, A, Hockerman, GH, Hering, S

“…BACKGROUND AND PURPOSE Diltiazem inhibits Ca V 1.2 channels and is widely used in clinical practice to treat cardiovascular diseases. Binding determinants for…”
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The third-generation P-glycoprotein inhibitor tariquidar may overcome bacterial multidrug resistance by increasing intracellular drug concentration by Leitner, I, Nemeth, J, Feurstein, T, Abrahim, A, Matzneller, P, Lagler, H, Erker, T, Langer, O, Zeitlinger, M

“…The use of efflux pump inhibitors may be a powerful strategy to overcome transporter-mediated bacterial multidrug resistance. In the present study, we set out…”
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Interaction of diltiazem with an intracellularly accessible binding site on CaV1.2 by Shabbir, W, Beyl, S, Timin, EN, Schellmann, D, Erker, T, Hohaus, A, Hockerman, GH, Hering, S

“…BACKGROUND AND PURPOSE Diltiazem inhibits CaV1.2 channels and is widely used in clinical practice to treat cardiovascular diseases. Binding determinants for…”
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Valerenic acid derivatives as novel subunit‐selective GABAA receptor ligands –in vitro and in vivo characterization by Khom, S, Strommer, B, Ramharter, J, Schwarz, T, Schwarzer, C, Erker, T, Ecker, GF, Mulzer, J, Hering, S

“…BACKGROUND AND PURPOSE Subunit‐specific modulators of γ‐aminobutyric acid (GABA) type A (GABAA) receptors can help to assess the physiological function of…”
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Novel Resveratrol Derivatives Induce Apoptosis and Cause Cell Cycle Arrest in Prostate Cancer Cell Lines by Horvath, Z, Marihart-Fazekas, S, Saiko, P, Grusch, M, Oezsuey, M, Harik, M, Handler, N, Erker, T, Jaeger, W, Fritzer-Szekeres, M, Djavan, B, Szekeres, T

“…Background: Resveratrol (RV), a naturally occurring phytoalexin, exerts manifold biological effects against a variety of human tumor cell lines. In this study,…”
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Synergistic action of resveratrol, an ingredient of wine, with Ara-C and tiazofurin in HL-60 human promyelocytic leukemia cells by Horvath, Zsuzsanna, Saiko, Philipp, Illmer, Christoph, Madlener, Sibylle, Hoechtl, Thomas, Bauer, Wolfgang, Erker, Thomas, Jaeger, Walter, Fritzer-Szekeres, Monika, Szekeres, Thomas

“…Resveratrol, a naturally occurring stilbene derivative, is a potent free-radical scavenger causing a number of biochemical and antineoplastic effects. It was…”
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Studies on the chemistry of thienoanellated O, N- and S, N-containing heterocycles. Part 30: Synthesis and pharmacological properties of thieno[2,3- b][1,4]thiazines with potential vasopressin receptor antagonistic activity by Galanski, Maria E., Erker, Thomas, Handler, Norbert, Lemmens-Gruber, Rosa, Kamyar, Majidreza, Studenik, Christian R.

“…A series of new nonpeptide vasopressin antagonists with a 6-ethyl-thieno[2,3- b][1,4]thiazine or 6-benzyl-thieno[2,3- b][1,4]thiazine skeleton and structural…”
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