Search Results - "Didier, Agnès"

Cyclosporins:  Structure−Activity Relationships for the Inhibition of the Human MDR1 P-Glycoprotein ABC Transporter by Loor, Francis, Tiberghien, Françoise, Wenandy, Tom, Didier, Agnès, Traber, René

“…Cyclic undecapeptide cyclo-[MeBmt-Abu-MeGly-MeLeu-Val-MeLeu-Ala-d-Ala-MeLeu-MeLeu-MeVal], the immunosuppressive and antifungal antibiotic cyclosporin A (CsA),…”
Get full text

Cyclosporins:  Structure−Activity Relationships for the Inhibition of the Human FPR1 Formylpeptide Receptor by Loor, Francis, Tiberghien, Françoise, Wenandy, Tom, Didier, Agnès, Traber, Rene

“…The human formylpeptide receptor (FPR) is a seven-transmembranous G-protein-coupled receptor (7TM-GPCR) for chemotactic peptides of bacterial origins, possibly…”
Get full text

Decreased biotolerability for ivermectin and cyclosporin A in mice exposed to potent P-glycoprotein inhibitors by Didier, A D, Loor, F

“…SDZ PSC 833 or SDZ 280-446 are strong blockers of the function of class I mdr gene-encoded P-glycoprotein molecules, which were developed for the reversal of…”
Get more information

Aureobasidins:  Structure−Activity Relationships for the Inhibition of the Human MDR1 P-Glycoprotein ABC-Transporter by Tiberghien, Françoise, Kurome, Toru, Takesako, Kazutoh, Didier, Agnès, Wenandy, Tom, Loor, Francis

“…Cyclic depsipeptide cyclo-[d-Hmp-l-MeVal-l-Phe-l-MePhe-l-Pro-l-aIle-l-MeVal-l-Leu-l-βHOMeVal], the antifungal antibiotic aureobasidin A (AbA), was reported to…”
Get full text

The MultiScreen® filtration system to measure chemoattractant-induced release of leukocyte granule enzymes by differentiated HL-60 cells or normal human monocytes by Tiberghien, Françoise, Didier, Agnès, Bohbot, Alain, Loor, Francis

“…A variety of chemoattractants initiate chemotaxis by selective binding to chemoattractant receptors (CARs), a subfamily of seven transmembranous G-protein…”
Get full text

The abamectin derivative ivermectin is a potent P-glycoprotein inhibitor by Didier, A, Loor, F

“…Among the compounds endowed with the capacity to reverse the P-glycoprotein (Pgp)-mediated multidrug resistance of cancer cells, a powerful agent was found to…”
Get more information