Search Results - "Devillers, Ingrid"

The Mechanism of Catalytic Enantioselective Fluorination: Computational and Experimental Studies by Piana, Stefano, Devillers, Ingrid, Togni, Antonio, Rothlisberger, Ursula

“…A parallel orientation between the coordinated substrate enolate and a face‐on naphthyl group of the TADDOL ligand (see picture; Ti dark gray, O red, Cl green,…”
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A biomimetic synthesis of coelenterazine analogs by Devillers, Ingrid, Arrault, Axelle, Olive, Gilles, Marchand-Brynaert, Jacqueline

“…N-(Trifluoroacetyl)dehydrodipeptides 2– 3 were coupled to aminomethylene dimethylacetal derivatives 4– 5 . The resulting pseudo-tripeptides 6 were stepwise…”
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Developing Catalytic Enantioselective Fluorination by Antonio Togni, Antonio Mezzetti, Peter Barthazy, Claus Becker, Ingrid Devillers, Richard Frantz, Lukas Hintermann, Mauro Perseghini, Maria Sanna

“…The background that led to the development ofthe first catalytic and enantioselective carbon-fluorine bond-forming reaction is presented. Two different…”
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Constrained Cyclic β,γ‐Diamino Acids from Glutamic Acid: Synthesis of Both Diastereomers and Unexpected Kinetic Resolution by Wan, Yang, Auberger, Nicolas, Thétiot‐Laurent, Sophie, Bouillère, Francelin, Zulauf, Anaïs, He, Jiefang, Courtiol‐Legourd, Stéphanie, Guillot, Régis, Kouklovsky, Cyrille, Cote des Combes, Sylvain, Pacaud, Christophe, Devillers, Ingrid, Alezra, Valérie

“…We describe here an efficient synthesis of both diastereomers of cyclic β,γ‐diamino acids starting from l‐glutamic acid, based on the Blaise reaction. We show…”
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The Mechanism of Catalytic Enantioselective Fluorination: Computational and Experimental Studies by Piana, Stefano, Devillers, Ingrid, Togni, Antonio, Rothlisberger, Ursula

“…Parallel zum Face‐on‐Naphthylrest des TADDOLs (siehe Bild; Ti dunkelgrau, O rot, Cl grün, F orange, N blauviolett) ausgerichtet ist die Enolatgruppe bei der…”
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Constrained Cyclic [beta],[gamma]-Diamino Acids from Glutamic Acid: Synthesis of Both Diastereomers and Unexpected Kinetic Resolution by Wan, Yang, Auberger, Nicolas, Thetiot-Laurent, Sophie, Bouillere, Francelin, Zulauf, Anaïs, He, Jiefang, Courtiol-Legourd, Stéphanie, Guillot, Régis, Kouklovsky, Cyrille, Cote des Combes, Sylvain, Pacaud, Christophe, Devillers, Ingrid, Alezra, Valérie

“…We describe here an efficient synthesis of both diastereomers of cyclic [beta],[gamma]-diamino acids starting from l-glutamic acid, based on the Blaise…”
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Efficient synthesis of both diastereomers of [beta],[gamma]-diamino acids from phenylalanine and tryptophan by Auberger, Nicolas, Stanovych, Andrii, Thétiot-laurent, Sophie, Guillot, Régis, Kouklovsky, Cyrille, Cote Des Combes, Sylvain, Pacaud, Christophe, Devillers, Ingrid, Alezra, Valérie

“…We synthesized in a few steps both diastereomers of orthogonally protected [beta],γ-diamino acids starting from l-phenylalanine or l-tryptophan. These final…”
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Efficient synthesis of both diastereomers of β,γ-diamino acids from phenylalanine and tryptophan by Auberger, Nicolas, Stanovych, Andrii, Thétiot-Laurent, Sophie, Guillot, Régis, Kouklovsky, Cyrille, Cote des Combes, Sylvain, Pacaud, Christophe, Devillers, Ingrid, Alezra, Valérie

“…We synthesized in a few steps both diastereomers of orthogonally protected β,γ-diamino acids starting from l -phenylalanine or l -tryptophan. These final…”
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The Crocacins: Novel Natural Products as Leads for Agricultural Fungicides by Patrick J. Crowley, Paul A. Worthington, Joe Swanborough, Olivia-Anabelle Sageot, Gordon R. Munns, Ingrid M. Devillers, Christopher R.A. Godfrey, Kevin Gillen, Ian H. Aspinall, John Williams

“…A short route to the synthesis of analogues of the antifungal but unstable natural product crocacin D was developed. A wide range of compounds were made in…”
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Preparation of azaindolines and benzoyl substituted azaindolines: precursors of triazabenzo[cd]azulen-9-one PDE4 inhibitors by Badland, Matthew, Devillers, Ingrid, Durand, Corinne, Fasquelle, Véronique, Gaudillière, Bernard, Jacobelli, Henry, Manage, Ajith C., Pevet, Isabelle, Puaud, Jocelyne, Shorter, Anthony J., Wrigglesworth, Roger

“…The syntheses of various substituted azaindolines are described. Azaindolines were identified as potential key intermediates towards new PDE4 inhibitors…”
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Relative Electrophilic Fluorinating Power as Assayed by Competitive Catalytic Halogenation Reactions by Toullec, Patrick Y., Devillers, Ingrid, Frantz, Richard, Togni, Antonio

“…Catalytic fluorination/chlorination competition experiments of β‐keto ester 5 were used to assess the relative fluorinating activity of various electrophilic…”
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Imidazolopyrazinones as potential antioxidants by Devillers, Ingrid, Dive, Georges, De Tollenaere, Catherine, Falmagne, Bénédicte, de Wergifosse, Bertrand, Rees, Jean-François, Marchand-Brynaert, Jacqueline

“…A series of imidazolopyrazinones 3, substituted at C-2, and C-2/C-6, has been prepared. The compounds behaved as quenchers of superoxide anion. The more active…”
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New substituted triaza-benzo[ cd]azulen-9-ones as promising phosphodiesterase-4 inhibitors by Devillers, Ingrid, Pevet, Isabelle, Jacobelli, Henry, Durand, Corinne, Fasquelle, Véronique, Puaud, Jocelyne, Gaudillière, Bernard, Idrissi, Moulay, Moreau, François, Wrigglesworth, Roger

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Developing Catalytic Enantioselective Fluorination by Antonio Togni, Antonio Mezzetti, Peter Barthazy, Claus Becker, Ingrid Devillers, Richard Frantz, Lukas Hintermann, Mauro Perseghini, Maria Sanna

“…The background that led to the development ofthe first catalytic and enantioselective carbon-fluorine bond-forming reaction is presented. Two different…”
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The Mechanism of Catalytic Enantioselective Fluorination: Computational and Experimental Studies by Piana, Stefano, Devillers, Ingrid, Togni, Antonio, Rothlisberger, Ursula

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Imidazolopyrazinones as potential antioxydants by Devillers, Ingrid, Dive, Georges, De Tollenaere, Catherine, Falmagne, Bénédicte, De Wergifosse, Bertrand, Rees, Jean-François, Marchand-Brynaert, Jacqueline

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