Search Results - "Delgado, Pete"

Structural analysis of inhibitor binding to human carbonic anhydrase II by Boriack‐Sjodin, P. Ann, Zeitlin, Samantha, Christianson, David W., Chen, Huang‐Hsing, Crenshaw, Lori, Gross, Sharon, Dantanarayana, Anura, Delgado, Pete, May, Jesse A., Dean, Tom

“…X‐ray crystal structures of carbonic anhydrase II (CAII) complexed with sulfonamide inhibitors illuminate the structural determinants of high affinity binding…”
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Use of Green Solvents in Metallaphotoredox Cross-Electrophile Coupling Reactions Utilizing a Lipophilic Modified Dual Ir/Ni Catalyst System by Delgado, Pete, Glass, Raoul J, Geraci, Gina, Duvadie, Rohit, Majumdar, Dyuti, Robinson, Richard I, Elmaarouf, Imran, Mikus, Malte, Tan, Kian L

“…Facilitating photoredox coupling reactions in process-friendly green solvents was achieved by the successful application of a dual Ir/Ni catalyst system with…”
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Merging Biocatalysis, Flow, and Surfactant Chemistry: Innovative Synthesis of an FXI (Factor XI) Inhibitor by Wu, Bin, Zhang, Sisi, Hong, Tao, Zhou, Yizong, Wang, Hui, Shi, Min, Yang, Hongwei, Tian, Xiangguang, Guo, Jing, Bian, Jianwei, Roache, James, Delgado, Pete, Mo, Ruowei, Fridrich, Cary, Gao, Feng, Wang, Jianhua

“…The scalable synthesis of an FXI (Factor XI) inhibitor employing multiple emerging technologies is described. The reduction of ketone to chiral alcohol was…”
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Two-step N-acylindazole to N-alkylindazole reduction. Further synthetic studies on the serotonergic agonist AL-34662 by Conrow, Raymond E., Delgado, Pete, Dean, W. Dennis, Callen, Gary R., Plummer, Scott V.

“…The two-step method avoids C–N bond cleavage, which predominates under typical metal hydride reduction conditions. This opens a new route to regiocontrolled…”
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AL-12182, a novel 11-oxa prostaglandin analog with topical ocular hypotensive activity in the monkey by Selliah, Robert D, Hellberg, Mark R, Sharif, Najam A, McLaughlin, Marsha A, Williams, Gary W, Scott, Daniel A, Earnest, David, Haggard, Karen S, Dennis Dean, W, Delgado, Pete, Gaines, Michael S, Conrow, Raymond E, Klimko, Peter G

“…Graphic A series of 11-oxa prostaglandin analogs was evaluated for FP receptor binding and activation. Several compounds having aryloxy-terminated lower chains…”
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Novel Esters and Amides of Nonsteroidal Antiinflammatory Carboxylic Acids as Antioxidants and Antiproliferative Agents by Hellberg, Mark R, Namil, Abdelmoula, Delgado, Pete, David, Karen C, Kessler, Timothy L, Graff, Gustav, Haggard, Karen S, Nixon, Jon C

“…A series of phenolic antioxidant ester and amide derivatives of the nonsteroidal antiinflammatory drug naproxen was designed to have both antiinflammatory and…”
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