Search Results - "Dal Forno, Giovanna"

Discovery Process and Characterization of Novel Carbohydrazide Derivatives as Potent and Selective GHSR1a Antagonists by Sabbatini, Fabio Maria, Di Fabio, Romano, Corsi, Mauro, Cavanni, Paolo, Bromidge, Steve M., St-Denis, Yves, D'Adamo, Lucilla, Contini, Stefania, Rinaldi, Marilisa, Guery, Sebastien, Savoia, Chiara, Mundi, Claudia, Perini, Benedetta, Carpenter, Andrew J., Dal Forno, Giovanna, Faggioni, Federico, Tessari, Michela, Pavone, Francesca, Di Francesco, Carla, Buson, Alberto, Mattioli, Mario, Perdona', Elisabetta, Melotto, Sergio

“…Ghrelins: don't feed them after dark! A novel class of highly potent and selective growth hormone secretagogue receptor 1a (GHSR1a) antagonists has been…”
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Enantiomerically pure tetrahydroquinoline derivatives as in vivo potent antagonists of the glycine binding site associated to the NMDA receptor by DI FABIO, Romano, TRANQUILLINI, Elvira, DONATI, Daniele, RATTI, Emiliangelo, ARBAN, Roberto, DAL FORNO, Giovanna, REGGIANI, Angelo, BARNABY, Robert J, BERTANI, Barbara, ALVARO, Giuseppe, MICHELI, Fabrizio, SABBATINI, Fabio, PIZZI, Maria Domenica, PENTASSUGLIA, Giorgio, PASQUARELLO, Alessandra, MESSERI, Tommaso

“…To identify neuroprotective agents after stroke, new substituted tetrahydroquinoline derivatives were designed as antagonists of the glycine binding site…”
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Novel carbazole derivatives as NPY Y1 antagonists by Leslie, Colin P., Fabio, Romano Di, Bonetti, Francesca, Borriello, Manuela, Braggio, Simone, Forno, Giovanna Dal, Donati, Daniele, Falchi, Alessandro, Ghirlanda, Damiano, Giovannini, Riccardo, Pavone, Francesca, Pecunioso, Angelo, Pentassuglia, Giorgio, Pizzi, Domenica A., Rumboldt, Giovanna, Stasi, Luigi

“…A series of carbazoles showing antagonist activity at the NPY Y1 receptor were prepared and characterised. Compound 13 combines potent activity with good brain…”
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Design and Synthesis of Novel Tricyclic Benzoxazines as Potent 5-HT1A/B/D Receptor Antagonists Leading to the Discovery of 6-{2-[4-(2-methyl-5-quinolinyl)-1-piperazinyl]ethyl}-4H-imidazo[5,1-c][1,4]benzoxazine-3-carboxamide (GSK588045) by Bromidge, Steven M, Arban, Roberto, Bertani, Barbara, Bison, Silvia, Borriello, Manuela, Cavanni, Paolo, Dal Forno, Giovanna, Di-Fabio, Romano, Donati, Daniele, Fontana, Stefano, Gianotti, Massimo, Gordon, Laurie J, Granci, Enrica, Leslie, Colin P, Moccia, Luca, Pasquarello, Alessandra, Sartori, Ilaria, Sava, Anna, Watson, Jeannette M, Worby, Angela, Zonzini, Laura, Zucchelli, Valeria

“…Bioisoteric replacement of the metabolically labile N-methyl amide group of a series of benzoxazinones with small heterocyclic rings has led to novel series of…”
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Design and Synthesis of Novel Tricyclic Benzoxazines as Potent 5-HT 1A/B/D Receptor Antagonists Leading to the Discovery of 6-{2-[4-(2-methyl-5-quinolinyl)-1-piperazinyl]ethyl}-4 H -imidazo[5,1- c ][1,4]benzoxazine-3-carboxamide (GSK588045) by Bromidge, Steven M., Arban, Roberto, Bertani, Barbara, Bison, Silvia, Borriello, Manuela, Cavanni, Paolo, Dal Forno, Giovanna, Di-Fabio, Romano, Donati, Daniele, Fontana, Stefano, Gianotti, Massimo, Gordon, Laurie J., Granci, Enrica, Leslie, Colin P., Moccia, Luca, Pasquarello, Alessandra, Sartori, Ilaria, Sava, Anna, Watson, Jeannette M., Worby, Angela, Zonzini, Laura, Zucchelli, Valeria

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Design and synthesis of novel tricyclic benzoxazines as potent 5-HT(1A/B/D) receptor antagonists leading to the discovery of 6-{2-[4-(2-methyl-5-quinolinyl)-1-piperazinyl]ethyl}-4H-imidazo[5,1-c][1,4]benzoxazine-3-carboxamide (GSK588045) by Bromidge, Steven M, Arban, Roberto, Bertani, Barbara, Bison, Silvia, Borriello, Manuela, Cavanni, Paolo, Dal Forno, Giovanna, Di-Fabio, Romano, Donati, Daniele, Fontana, Stefano, Gianotti, Massimo, Gordon, Laurie J, Granci, Enrica, Leslie, Colin P, Moccia, Luca, Pasquarello, Alessandra, Sartori, Ilaria, Sava, Anna, Watson, Jeannette M, Worby, Angela, Zonzini, Laura, Zucchelli, Valeria

“…Bioisoteric replacement of the metabolically labile N-methyl amide group of a series of benzoxazinones with small heterocyclic rings has led to novel series of…”
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Receptor binding characteristics of the novel NMDA receptor glycine site antagonist [ 3H]GV150526A in rat cerebral cortical membranes by Mugnaini, Manolo, Dal Forno, Giovanna, Corsi, Mauro, Bunnemann, Bernd

“…Binding of the glycine site antagonist 3-[2-(Phenylamino-carbonyl)ethenyl]-4,6-dichloro-indole-2-carboxylic acid sodium salt ([ 3H]GV150526A) was characterised…”
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Benzoazepine derivative as potent antagonists of the glycine binding site associated to the NMDA receptor by Di Fabio, Romano, Micheli, Fabrizio, Baraldi, Davide, Bertani, Barbara, Conti, Nadia, Dal Forno, Giovanna, Feriani, Aldo, Donati, Daniele, Marchioro, Carla, Messeri, Tommaso, Missio, Andrea, Pasquarello, Alessandra, Pentassuglia, Giorgio, Pizzi, Domenica A., Provera, Stefano, Quaglia, Anna M., Sabbatini, Fabio M.

“…A series of benzoazepine derivatives, bearing suitable substituents at the C-3 position, was designed and evaluated by superimposition with the pharmacophore…”
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