Search Results - "DUNAISKIS, A. R"

Synthesis and Oral Efficacy of a 4-(Butylethylamino)pyrrolo[2,3-d]pyrimidine:  A Centrally Active Corticotropin-Releasing Factor1 Receptor Antagonist by Chen, Yuhpyng L, Mansbach, Robert S, Winter, Steven M, Brooks, Elizabeth, Collins, Judith, Corman, Michael L, Dunaiskis, Audrey R, Faraci, W. Stephen, Gallaschun, Randall J, Schmidt, Anne, Schulz, David W

“…The syntheses of a centrally active nonpeptide CRF1 receptor antagonist 2,…”
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Synthesis, sar and pharmacology of CP-293,019 : A potent, selective dopamine D4 receptor antagonist by SANNER, M. A, CHAPPIE, T. A, MAJCHRZAK, M. J, FARACI, W. S, COLLINS, J. L, DUIGNAN, D. B, DI PRETE, C. C, LEE, J. S, TROZZI, A, DUNAISKIS, A. R, FLIRI, A. F, DESAI, K. A, ZORN, S. H, JACKSON, E. R, JOHNSON, C. G, MORRONE, J. M, SEYMOUR, P. A

“…A series of novel, potent and selective pyrido[1,2-a]pyrazine dopamine D4 receptor antagonists are reported including CP-293,019 (D4 Ki = 3.4 nM, D2 Ki > 3,310…”
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Synthesis, sar and pharmacology of CP-293,019: A potent, selective dopamine D 4 receptor antagonist by Sanner, Mark A., Chappie, Thomas A., Dunaiskis, Audrey R., Fliri, Anton F., Desai, Kishor A., Zorn, Stevin H., Jackson, Elisa R., Johnson, Celeste G., Morrone, Jean M., Seymour, Patricia A., Majchrzak, Mark J., Stephen Faraci, W., Collins, Judith L., Duignan, David B., Di Prete, Cecilia C., Lee, Jae S., Trozzi, Angela

“…A series of novel, potent and selective pyrido[1,2- a]pyrazine dopamine D 4 receptor antagonists are reported including CP-293,019 (D 4 K i = 3.4 nM, D 2 K i >…”
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