Search Results - "DANHO, Waleed"

Editorial: The boulder peptide symposium 2021 scientific update by Angell, Yvonne, Mayer, John, Nofsinger, Rebecca, Danho, Waleed

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A Selective Phosphatase of Regenerating Liver Phosphatase Inhibitor Suppresses Tumor Cell Anchorage-Independent Growth by a Novel Mechanism Involving p130Cas Cleavage by DAOUTI, Sherif, LI, Wen-Hui, HONGJIN BIAN, REIDHAAR-OLSON, John F, BLISS, Sarah A, OLIVIER, Andree R, SERGI, Joseph A, FRY, David, DANHO, Waleed, RITLAND, Steve, FOTOUHI, Nader, HEIMBROOK, David, HONG QIAN, HUIFENG NIU, HUANG, Kuo-Sen, HOLMGREN, Janna, LEVIN, Wayne, REIK, Linda, MCGADY, Debra Lucas, GILLESPIE, Paul, PERROTTA, Agostino

“…The phosphatase of regenerating liver (PRL) family, a unique class of oncogenic phosphatases, consists of three members: PRL-1, PRL-2, and PRL-3. Aberrant…”
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The N-terminal Domain of RGS4 Confers Receptor-selective Inhibition of G Protein Signaling by Zeng, W, Xu, X, Popov, S, Mukhopadhyay, S, Chidiac, P, Swistok, J, Danho, W, Yagaloff, K A, Fisher, S L, Ross, E M, Muallem, S, Wilkie, T M

“…Regulators of heterotrimeric G protein signaling (RGS) proteins are GTPase-activating proteins (GAPs) that accelerate GTP hydrolysis by G q and G i α…”
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Structure-activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH2 at the human melanocortin-1 and -4 receptors: Arginine substitution by CHEUNG, Adrian Wai-Hing, DANHO, Waleed, SWISTOK, Joseph, QI, Lida, KURYLKO, Grazyna, FRANCO, Lucia, YAGALOFF, Keith, LI CHEN

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A predictive pharmacophore model of human melanocortin-4 receptor as derived from the solution structures of cyclic peptides by Sun, Hongmao, Greeley, David N., Chu, Xin-Jie, Cheung, Adrian, Danho, Waleed, Swistok, Joseph, Wang, Yao, Zhao, Chunlin, Chen, Li, Fry, David C.

“…A predictive pharmacophore model of human melanocortin-4 receptor (hMC4R) was derived from the NMR structures of a series of rigidified MT-II related cyclic…”
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Discovery of 1-amino-4-phenylcyclohexane-1-carboxylic acid and its influence on agonist selectivity between human melanocortin-4 and -1 receptors in linear pentapeptides by Chu, Xin-Jie, Bartkovitz, David, Danho, Waleed, Swistok, Joseph, Cheung, Adrian Wai-Hing, Kurylko, Grazyna, Rowan, Karen, Yeon, Mitch, Franco, Lucia, Qi, Lida, Chen, Li, Yagaloff, Keith

“…A design and synthesis of cis-Apc as new histidine surrogate and its incorporation into linear pentapeptides (Penta- cis-Apc-DPhe-Arg-Trp-Gly-NH 2) and related…”
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Structure-activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH2 at the human melanocortin-1 and -4 receptors: Histidine substitution by CHEUNG, Adrian Wai-Hing, DANHO, Waleed, YAGALOFF, Keith, SWISTOK, Joseph, LIDA QI, KURYLKO, Grazyna, ROWAN, Karen, YEON, Mitch, FRANCO, Lucia, CHU, Xin-Jie, LI CHEN

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Camstatins Are Peptide Antagonists of Calmodulin Based Upon a Conserved Structural Motif in PEP-19, Neurogranin, and Neuromodulin by Slemmon, J. Randall, Morgan, James I., Fullerton, Stephanie M., Danho, Waleed, Hilbush, Brian S., Wengenack, Thomas M.

“…Unbridled increases in intracellular ionized calcium can result in neuronal damage and death. Since many of the deleterious effects of calcium are mediated by…”
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Preparation of human Melanocortin-4 receptor agonist libraries : Linear peptides X-Y-DPhe7-Arg8-Trp(or 2-Nal)9-Z-NH2 by CHEUNG, Adrian Wai-Hing, LIDA QI, GORE, Vijay, CHU, Xin-Jie, BARTKOVITZ, David, KURYLKO, Grazyna, SWISTOK, Joseph, DANHO, Waleed, LI CHEN, YAGALOFF, Keith

“…Two libraries of hMC4R agonists, X-Y-DPhe(7)-Arg(8)-2-Nal(9)-Z-NH(2) and X-Y-DPhe(7)-Arg(8)-Trp(9)-Z-NH(2), totaling 185 peptides were prepared using Irori…”
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Lipidation and PEGylation strategies to prolong the in vivo half-life of a nanomolar EphA4 receptor antagonist by Gomez-Soler, Maricel, Olson, Erika J., Rubio de la Torre, Elena, Zhao, Chunxia, Lamberto, Ilaria, Flood, Dillon T., Danho, Waleed, Lechtenberg, Bernhard C., Riedl, Stefan J., Dawson, Philip E., Pasquale, Elena B.

“…The EphA4 receptor tyrosine kinase plays a role in neurodegenerative diseases, inhibition of nerve regeneration, cancer progression and other diseases…”
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Structure-activity relationship of cyclic peptide Penta-c[Asp-His6-DPhe7-Arg8-Trp9-Lys]-NH2 at the human melanocortin-1 and -4 receptors: His6 substitution by WAI-HING CHEUNG, Adrian, DANHO, Waleed, YAGALOFF, Keith, SWISTOK, Joseph, QI, Lida, KURYLKO, Grazyna, ROWAN, Karen, YEON, Mitch, FRANCO, Lucia, CHU, Xin-Jie, LI CHEN

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Structure-activity relationship of linear peptide Bu-His6-DPhe7-Arg8-Trp9-Gly10-NH2 at the human melanocortin-1 and -4 receptors : DPhe7 and Trp9 substitution by DANHO, Waleed, SWISTOK, Joseph, CHEUNG, Adrian Wai-Hing, KURYLKO, Grazyna, FRANCO, Lucia, CHU, Xin-Jie, LI CHEN, YAGALOFF, Keith

“…A series of pentapeptides, based on hMC4R pentapeptide agonist (Bu-His(6)-DPhe(7)-Arg(8)-Trp(9)-Gly(10)-NH(2)), was prepared in which either DPhe(7) or Trp(9)…”
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Molecular cloning of G proteins and phosphodiesterases from rat taste cells by McLaughlin, S K, McKinnon, P J, Spickofsky, N, Danho, W, Margolskee, R F

“…To identify and characterize those proteins involved in taste transduction, we cloned G proteins and phosphodiesterases from rat taste tissue. Using degenerate…”
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Preparation and Characterization of Albumin Conjugates of a Truncated Peptide YY Analogue for Half-Life Extension by Ehrlich, George K, Michel, Hanspeter, Truitt, Theresa, Riboulet, William, Pop-Damkov, Petar, Goelzer, Petra, Hainzl, Dominik, Qureshi, Farooq, Lueckel, Barbara, Danho, Waleed, Conde-Knape, Karin, Konkar, Anish

“…Recombinant human serum albumin (HSA) conjugates of a 15-amino-acid truncated peptide YY (PYY) analogue were prepared using three heterobifunctional linkers…”
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The structure of XIAP BIR2: understanding the selectivity of the BIR domains by Lukacs, Christine, Belunis, Charles, Crowther, Robert, Danho, Waleed, Gao, Lin, Goggin, Barry, Janson, Cheryl A., Li, Shirley, Remiszewski, Stacy, Schutt, Andrew, Thakur, Manish K., Singh, Saroj K., Swaminathan, Srinivasan, Pandey, Rajat, Tyagi, Rajiv, Gosu, Ramachandraiah, Kamath, Ajith V., Kuglstatter, Andreas

“…XIAP, a member of the inhibitor of apoptosis family of proteins, is a critical regulator of apoptosis. Inhibition of the BIR domain–caspase interaction is a…”
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Vomeromodulin, a putative pheromone transporter: cloning, characterization, and cellular localization of a novel glycoprotein of lateral nasal gland by Khew-Goodall, Y, Grillo, M, Getchell, M L, Danho, W, Getchell, T V, Margolis, F L

“…Vomeromodulin, a novel glycoprotein of lateral nasal gland, has been cloned by differential hybridization from nasal/olfactory tissue. The 2.2-kb mRNA directs…”
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Opportunities and challenges of developing peptide drugs in the pharmaceutical industry by Danho, Waleed, Swistok, Joseph, Khan, Wajiha, Chu, Xin-Jie, Cheung, Adrian, Fry, David, Sun, Hongmao, Kurylko, Grazyna, Rumennik, Leonid, Cefalu, Joseph, Cefalu, Gretchen, Nunn, Philip

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Carboxylic acids and tetrazoles as isosteric replacements for sulfate in cholecystokinin analogs by Tilley, Jefferson W, Danho, Waleed, Lovey, Kathleen, Wagner, Rolf, Swistok, Joseph, Makofske, Raymond, Michalewsky, Joseph, Triscari, Joseph, Nelson, David, Weatherford, Sally

“…A series of analogues of the satiety-inducing peptide cholecystokinin (CCK-8) was prepared in which the sulfated tyrosine required for activation of peripheral…”
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Isolation and Sequencing of Two Cerebellum-Specific Peptides by Slemmon, J. Randall, Blacher, Russell, Danho, Waleed, Hempstead, James L., Morgan, James I.

“…By comparing the HPLC elution profiles of peptides isolated from different brain regions, two cerebellum-specific species have been identified. The peptides…”
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T cells recognize both conformational and cryptic determinants on the insulin molecule by Thomas, J W, George-Gattner, H, Danho, W

“…T lymphocytes from strain 2 guinea pigs were studied for recognition of isolated insulin A and B chains. Insulin-immune T cells require intact conformation of…”
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