Search Results - "Cooper, Robin D. G"

Azetidinones as vasopressin V1a antagonists by Guillon, Christophe D., Koppel, Gary A., Brownstein, Michael J., Chaney, Michael O., Ferris, Craig F., Lu, Shi-fang, Fabio, Karine M., Miller, Marvin J., Heindel, Ned D., Hunden, David C., Cooper, Robin D.G., Kaldor, Stephen W., Skelton, Jeffrey J., Dressman, Bruce A., Clay, Michael P., Steinberg, Mitchell I., Bruns, Robert F., Simon, Neal G.

“…The azetidinone LY307174 ( 1) was identified as a screening lead for the vasopressin V1a receptor (IC 50 45 nM at the human V1a receptor) based on molecular…”
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Glycopeptide carboxamides active against vancomycin-resistant enterococci by Zweifel, Mark J, Snyder, Nancy J, Cooper, Robin D G, Nicas, Thalia I, Mullen, Deborah L, Butler, Thomas F, Rodriguez, Michael J

“…Glycopeptide antibiotics were synthesized via the PyBOP mediated condensation of aliphatic, heterocyclic and aromatic amines with the C-terminus of vancomycin,…”
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Reductive alkylation of glycopeptide antibiotics: synthesis and antibacterial activity by Cooper, R D, Snyder, N J, Zweifel, M J, Staszak, M A, Wilkie, S C, Nicas, T I, Mullen, D L, Butler, T F, Rodriguez, M J, Huff, B E, Thompson, R C

“…Reductive alkylation of the A82846 family of glycopeptide antibiotics has the potential of producing seven products. N-Alkylation of the disaccharide amino…”
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Enzymatic deacylation of teicoplanin followed by reductive alkylation: synthesis and antibacterial activity of new glycopeptides by Snyder, N J, Cooper, R D, Briggs, B S, Zmijewski, M, Mullen, D L, Kaiser, R E, Nicas, T I

“…Novel glycopeptides derived from teicoplanin were prepared and evaluated for activity against antibiotic-resistant gram-positive pathogens. Removal of the…”
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Orally absorbable cephalosporin antibiotics. 2. Structure-activity studies of bicyclic glycine derivatives of 7-aminodeacetoxycephalosporanic acid by Kukolja, Stjepan, Draheim, Susan E, Graves, Bernard J, Hunden, David C, Pfeil, Janice L, Cooper, Robin D. G, Ott, John L, Counter, Fred T

“…Three positional analogues (4-, 5-, and 7-) of benzothienylglycine and (N-acetylindolinyl)-5-glycine were prepared and coupled to…”
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Chemistry of cephalosporin antibiotics. XXI. Conversion of penicillins to cephalexin by Chauvette, Robert R, Pennington, Pamela A, Ryan, Charles W, Cooper, Robin D. G, Jose, Felicitas L, Wright, Ian Glaiby, Van Heyningen, Earle M, Huffman, George W

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Structural studies on penicillin derivatives. I. Configuration of phenoxymethylpenicillin sulfoxide by Cooper, Robin D. G, DeMarco, Paul V, Cheng, James C, Jones, Noel D

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Carotenoids and related compounds. Part XXXII. Synthesis of astaxanthin, phoenicoxanthin, hydroxyechinenone, and the corresponding diosphenols by Cooper, R D, Davis, J B, Leftwick, A P, Price, C, Weedon, B C

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Chemical interconversion of the .beta.-lactam antibiotics by Cooper, Robin D. G, Hatfield, Lowell D, Spry, Douglas O

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Structural studies on penicillin derivatives. V. Penicillin sulfoxide-sulfenic acid equilibrium by Cooper, Robin D. G

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Orally absorbable cephalosporin antibiotics. 1. Structure-activity relationships of benzothienyl- and naphthylglycine derivatives of 7-aminodeacetoxycephalosporanic acid by Kukolja, Stjepan, Draheim, Susan E, Pfeil, Janice L, Cooper, Robin D. G, Graves, Bernard J, Holmes, Richard E, Neel, David A, Huffman, George W, Webber, J. Alan

“…A structure-activity relationship study of a number of orally absorbed cephalosporins together with their syntheses is described. These new cephalosporins are…”
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Wherefore art thou Romeo? by Cooper, Robin D G

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Chiral synthesis of protected 3-amino-4-(alkoxycarbonyl)-2-azetidinones from .beta.-hydroxyaspartic acid by Mattingly, Philip G, Miller, Marvin J, Cooper, Robin D. G, Daughtery, B. W

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Structural studies on penicillin derivatives. II. Configuration of phthalimidopenicillin and epiphthalimidopenicillin sulfoxides by Cooper, Robin D. G, DeMarco, Paul V, Spry, Douglas O

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Chemistry of cephalosporin antibiotics. XIX. Transformation of .DELTA.2-cephem to .DELTA.3-cephem by oxidation-reduction at sulfur by Kaiser, G. V, Cooper, Robin D. G, Koehler, R. E, Murphy, C. F, Webber, J. A, Wright, Ian Glaisby, Van Heyningen, E. M

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Novel glycopeptide antibiotics: N-alkylated derivatives active against vancomycin-resistant enterococci by Rodriguez, M J, Snyder, N J, Zweifel, M J, Wilkie, S C, Stack, D R, Cooper, R D, Nicas, T I, Mullen, D L, Butler, T F, Thompson, R C

“…LY264826 (A82846B) is a naturally-occurring glycopeptide antibiotic, differing from vancomycin in the stereochemistry of the amino-sugar of the disaccharide…”
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The carbacephems: a new beta-lactam antibiotic class by Copper, R D

“…The carbacephems are a new class of beta-lactam antibiotics that are similar in structure to the cephalosporins. Carbacephems differ from cephalosporins,…”
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A Class of Small Molecules that Inhibit TNFα-Induced Survival and Death Pathways via Prevention of Interactions between TNFαRI, TRADD, and RIP1 by Gururaja, Tarikere L., Yung, Stephanie, Ding, Rongxian, Huang, Jianing, Zhou, Xiulan, McLaughlin, John, Daniel-Issakani, Sarkiz, Singh, Rajinder, Cooper, Robin D.G., Payan, Donald G., Masuda, Esteban S., Kinoshita, Taisei

“…Small-molecule library screening to find compounds that inhibit TNFα-induced, but not interleukin 1β (IL-1β)-induced, intercellular adhesion molecule 1…”
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A class of small molecules that inhibit TNFalpha-induced survival and death pathways via prevention of interactions between TNFalphaRI, TRADD, and RIP1 by Gururaja, Tarikere L, Yung, Stephanie, Ding, Rongxian, Huang, Jianing, Zhou, Xiulan, McLaughlin, John, Daniel-Issakani, Sarkiz, Singh, Rajinder, Cooper, Robin D G, Payan, Donald G, Masuda, Esteban S, Kinoshita, Taisei

“…Small-molecule library screening to find compounds that inhibit TNFalpha-induced, but not interleukin 1beta (IL-1beta)-induced, intercellular adhesion molecule…”
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Structural studies on penicillin derivatives. IV. Novel rearrangement of penicillin V sulfoxide by Cooper, Robin D. G., Jose, F. L.

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