Search Results - "Chulakov, E. N."

Synthesis of novel biotin-based carborane amides by Telegina, A. A., Gruzdev, D. A., Chulakov, E. N., Levit, G. L., Koryakova, O. V., Krasnov, V. P.

“…A series of novel derivatives of d -biotin containing closo - and nido -carborane residues bound to the biotin carbonyl group either directly or via a linker…”
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Kinetic resolution of racemic 6-substituted 3-methyl-3,4-dihydro-2H-[1,4]benzoxazines with chiral acyl chlorides by Chulakov, E. N., Korolyova, M. A., Tumashov, A. A., Kodess, M. I., Levit, G. L., Krasnov, V. P.

“…A comparative study of the kinetic resolution of racemic 6-methoxy-, 6-nitro-, and 6-chloro-3-methyl-3,4-dihydro-2 H -[1,4]benzoxazines with ( S )-naproxen…”
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Synthesis of Glycyl-(S)-5-hydroxynorvaline by Chulakov, E. N., Tumashov, A. A., Gruzdev, D. A., Levit, G. L., Krasnov, V. P.

“…The dipeptide glycyl-( S )-5-hydroxynorvaline was obtained from 1- tert -butyl 5-methyl N -Boc-glycyl-( S )-glutamate via saponification, reduction of the…”
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Synthesis of enantiomers of 6-substituted 3-methyl-3,4-dihydro-2H-[1,4]benzoxazines by Chulakov, E. N., Gruzdev, D. A., Korolyova, M. A., Tumashov, A. A., Kodess, M. I., Levit, G. L., Krasnov, V. P.

“…Individual ( S )-enantiomers of 6-methoxy-, 6-chloro-, and 6-nitro-3-methyl-3,4-di-hydro-2 H -[1,4]benzoxazines were synthesized via an acylative kinetic…”
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Kinetic resolution of racemic 6-substituted 1,2,3,4-tetrahydroquinaldines with chiral acyl chlorides. Experiment and quantum chemical simulation by Chulakov, E. N., Korolyova, M. A., Sadretdinova, L. Sh, Tumashov, A. A., Kodess, M. I., Levit, G. L., Krasnov, V. P.

“…A comparative study of the kinetic resolution (KR) of racemic 6-substituted 2-methyl-1,2,3,4-tetrahydroquinolines with acyl chlorides of ( S )-naproxen, N…”
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HPLC separation of 2-aryloxycarboxylic acid enantiomers on chiral stationary phases by Tumashov, A. A., Vakarov, S. A., Sadretdinova, L. Sh, Chulakov, E. N., Levit, G. L., Krasnov, V. P., Charushin, V. N.

“…The possibility for separating enantiomers of a number of practically significant 2-aryloxycarboxylic acids was studied by normal- and reversed-phase HPLC on…”
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Kinetic resolution of racemic 3-tert-butyl-3,4-dihydro-2H-[1,4]benzoxazine via acylation with chiral acyl chlorides by Vakarov, S. A., Gruzdev, D. A., Chulakov, E. N., Levit, G. L., Krasnov, V. P.

“…A comparative study of the kinetic resolution of racemic 3- tert -butyl-3,4-dihydro-2 H -[1,4]-benzoxazine through the acylation by various chiral acyl…”
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Effectiveness of Repeated Administration of Praziquantel with Disodium Glycyrrhizinate and Two Enantiomers of Praziquantel on Opisthorchis felineus (Rivolta, 1884) by Avgustinovich, D. F., Tsyganov, M. A., Pakharukova, M. Y., Chulakov, E. N., Dushkin, A. V., Krasnov, V. P., Mordvinov, V. A.

“…Background Nowadays, it is still important to develop effective anti-opisthorchiasis agents. In this work, we tested a complex of praziquantel (PZQ) with a…”
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Analysis of racemic conjugates of purine with heterocyclic amines by chiral high-performance liquid chromatography by Tumashov, A. A., Gruzdev, D. A., Vigorov, A. Yu, Musiyak, V. V., Chulakov, E. N., Levit, G. L., Krasnov, V. P., Charushin, V. N.

“…Reversed-phase HPLC on chiral stationary phases was used to study the influence of the structure of purine and 2-aminopurine conjugates with chiral…”
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Synthesis of Purine and 2-Aminopurine Conjugates with N-(4-Aminobenzoyl)-(S)-glutamic Acid by Krasnov, V. P., Vigorov, A. Yu, Chulakov, E. N., Nizova, I. A., Levit, G. L., Kravchenko, M. A., Charushin, V. N.

“…Purine and 2-aminopurine conjugates with N -(4-aminobenzoyl)-( S )-glutamic acid connected to C 6 of the purine system either directly or through an aminoethyl…”
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Diastereoselective Acylation of Racemic Heterocyclic Amines with N-Phthaloyl and N-Naphthaloyl (S)-Amino Acyl Chlorides: Possibility of Parallel Kinetic Resolution by Gruzdev, D. A., Chulakov, E. N., Sadretdinova, L. Sh, Levit, G. L., Krasnov, V. P., Charushin, V. N.

“…The acylative kinetic resolution of racemic 2-methyl-1,2,3,4-tetrahydroquinoline and 3,4-dihydro-3-methyl-2 H -[1,4]benzoxazines with acyl chlorides of N…”
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Synthesis and piezoelectric properties of N-phthaloylglutamic acid derivatives by Ustinova, V. O., Vigorov, A. Yu, Gruzdev, D. A., Nuraeva, A. S., Nizova, I. A., Chulakov, E. N., Sadretdinova, L. Sh, Slepukhin, P. A., Zelenovsky, P. S., Shur, V. Ya, Krasnov, V. P.

“…The ( S , S )- and ( R , R )-enantiomers of dimethyl 2,4-diphthalimidoglutarate were synthesized by nucleophilic substitution of bromine in dimethyl (2 S ,4 RS…”
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Diastereoselective Acylation of Racemic Heterocyclic Amines with N-Tosyl-(S)-Prolyl Chloride and its Structural Analogs by Vakarov, S. A., Gruzdev, D. A., Chulakov, E. N., Sadretdinova, L. Sh, Ezhikova, M. A., Kodess, M. I., Levit, G. L., Krasnov, V. P.

“…A comparative study on the kinetic resolution of racemic amines (2,3-dihydro-4H-1,4-benzoxazine and 1,2,3,4-tetrahydroquinoline derivatives) via…”
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Enantioselective microbial synthesis of (S)-7,8-difluoro-3,4-dihydro-3-methyl-2H-[1,4]benzoxazine by Chulakov, E. N., Levit, G. L., Tumashov, A. A., Lugovskaya, N. P., Remezovskaya, N. B., Maksimov, A. Yu, Demakov, V. A., Krasnov, V. P.

“…New strains of Rhodococcus erythropolis 25 and Microbacterium paraoxydans 20-11c actinobacteria were used to obtain ( S )-7,8-difluoro-3,4-dihydro-3-methyl-2 H…”
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2-Arylpropionyl chlorides in kinetic resolution of racemic 3-methyl-2,3-dihydro-4H-[1,4]benzoxazines by Chulakov, E. N., Gruzdev, D. A., Levit, G. L., Sadretdinova, L. Sh, Krasnov, V. P., Charushin, V. N.

“…Kinetic resolution of racemic 3-methyl-2,3-dihydro-4 H -[1,4]benzoxazines in the reaction with chiral 2-arylpropionyl chloride predominantly yielded R *, R…”
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Structures of the racemate and (S)-enantiomer of 7,8-difluoro-3-methyl-2,3-dihydro-4H-[1,4]benzoxazine by Slepukhin, P. A., Gruzdev, D. A., Chulakov, E. N., Levit, G. L., Krasnov, V. P., Charushin, V. N.

“…The comparative X-ray diffraction study of racemic and ( S )-enantiomer of 7,8-difluoro-3-methyl-2,3-dihydro-4 H -[1,4]benzoxazine was carried out. The both…”
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Kinetic resolution of racemic 2-methyl-1,2,3,4-tetrahydroquinoline and its structural analogs by using 2-arylpropionyl chlorides by Chulakov, E. N., Levit, G. L., Tumashov, A. A., Sadretdinova, L. Sh, Krasnov, V. P.

“…Acylation of 2-methyl-1,2,3,4-tetrahydroquinoline and 2-methylindoline with the acyl chlorides of naproxen, ibuprofen, and 2-phenylpropionic acid has been…”
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