Search Results - "Christensen, Inge T"

Differential Interactions of Nateglinide and Repaglinide on the Human β-Cell Sulphonylurea Receptor 1 by HANSEN, Ann Maria K, CHRISTENSEN, Inge T, HANSEN, John Bondo, CARR, Richard D, ASHCROFT, Frances M, WAHL, Philip

“…Differential Interactions of Nateglinide and Repaglinide on the Human β-Cell Sulphonylurea Receptor 1 Ann Maria K. Hansen 1 , Inge T. Christensen 1 , John…”
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Human Glucagon Receptor Antagonists with Thiazole Cores. A Novel Series with Superior Pharmacokinetic Properties by Madsen, Peter, Kodra, János T, Behrens, Carsten, Nishimura, Erica, Jeppesen, Claus B, Pridal, Lone, Andersen, Birgitte, Knudsen, Lotte B, Valcarce-Aspegren, Carmen, Guldbrandt, Mette, Christensen, Inge T, Jørgensen, Anker S, Ynddal, Lars, Brand, Christian L, Bagger, Morten Aa, Lau, Jesper

“…The aim of the work presented here was to design and synthesize potent human glucagon receptor antagonists with improved pharmacokinetic (PK) properties for…”
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Homology building as a means to define antigenic epitopes on dihydrofolate reductase (DHFR) from Plasmodium falciparum by Alifrangis, Michael, Christensen, Inge T, Jørgensen, Flemming S, Rønn, Anita M, Weng, Jimmy E, Chen, Ming, Bygbjerg, Ib C, Sirawaraporn, Worachart, Palarasah, Yaseelan, Koch, Claus

“…The aim of this study was to develop site-specific antibodies as a tool to capture Plasmodium falciparum-dihydrofolate reductase (Pf-DHFR) from blood samples…”
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Computational prediction of solubilizers’ effect on partitioning by Hoest, Jan, Christensen, Inge T., Jørgensen, Flemming S., Hovgaard, Lars, Frokjaer, Sven

“…A computational model for the prediction of solubilizers’ effect on drug partitioning has been developed. Membrane/water partitioning was evaluated by means of…”
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Structure−Property Model for Membrane Partitioning of Oligopeptides by Alifrangis, Lene Hjorth, Christensen, Inge T, Berglund, Anders, Sandberg, Maria, Hovgaard, Lars, Frokjaer, Sven

“…The aim of this study was to develop a structure−property model for membrane partitioning of oligopeptides using statistical design methods and multivariate…”
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Assessing the relative importance of the biophysical properties of amino acid substitutions associated with human genetic disease by Terp, Bent N., Cooper, David N., Christensen, Inge T., Jørgensen, Flemming S., Bross, Peter, Gregersen, Niels, Krawczak, Michael

“…The inclusion of a mutation in a pathology‐based database such as the Human Gene Mutation Database (HGMD) is a two‐stage process: first, the mutation must…”
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Excitatory Amino Acid Receptor Ligands:  Resolution, Absolute Stereochemistry, and Enantiopharmacology of 2-Amino-3-(4-butyl-3-hydroxyisoxazol-5-yl)propionic Acid by Johansen, Tommy N, Ebert, Bjarke, Bräuner-Osborne, Hans, Didriksen, Michael, Christensen, Inge T, Søby, Karina K, Madsen, Ulf, Krogsgaard-Larsen, Povl, Brehm, Lotte

“…(RS)-2-Amino-3-(4-butyl-3-hydroxyisoxazol-5-yl)propionic acid (Bu-HIBO, 6) has previously been shown to be an agonist at…”
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Synthesis and Pharmacology of Highly Selective Carboxy and Phosphono Isoxazole Amino Acid AMPA Receptor Antagonists by Madsen, Ulf, Bang-Andersen, Benny, Brehm, Lotte, Christensen, Inge T, Ebert, Bjarke, Kristoffersen, Inge T. S, Lang, Yolande, Krogsgaard-Larsen, Povl

“…(RS)-2-Amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid (AMPA, 5) and the selective AMPA receptor antagonist…”
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Excitatory amino acid receptor ligands. Synthesis and biological activity of 3-isoxazolol amino acids structurally related to homoibotenic acid by Christensen, Inge T, Ebert, Bjarke, Madsen, Ulf, Nielsen, Birgitte, Brehm, Lotte, Krogsgaard-Larsen, Povl

“…The 3-isoxazolol amino acid (RS)-2-amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic acid (AMPA, 2) and the isomeric compound…”
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Differential interactions of nateglinide and repaglinide on the human [beta]-Cell sulphonylurea receptor 1 by Hansen, Ann Maria K, Christensen, Inge T, Hansen, John Bondo, Carr, Richard D, Ashcroft, Frances M, Wahl, Philip

“…Repaglinide and nateglinide represent a new class of insulin secretagogues, structurally unrelated to sulphonylureas, that were developed for the treatment of…”
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Assessing the relative importance of the biophysical properties of amino acid substitutions associated with human genetic disease: EFFECTS OF AMINO ACID SUBSTITUTIONS by Terp, Bent N., Cooper, David N., Christensen, Inge T., Jørgensen, Flemming S., Bross, Peter, Gregersen, Niels, Krawczak, Michael

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Homology modelling of dihydrofolate reductase from the malaria parasite by Lemcke, Thomas, Christensen, Inge T., Jergensen, Flemming S.

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