Search Results - "Chikhalia, Kishor"

Innovative cascade reaction for 2H-indazole derivative synthesis by Choudhary, Annu, Patel, Rohit, Goswami, Dweipayan, Chikhalia, Kishor H

“…In the realm of synthetic organic chemistry, by using a one-pot sequential combination of MCR, it is possible to manufacture chemical commodities (fine…”
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Iron-catalyzed intermolecular cross-dehydrogenative C(sp3)–H/C(sp)–H coupling of pyrimidine bearing 4-thiazolidinones with terminal alkynes by Morja, Mayur I., Chikhalia, Kishor H.

“…A novel, simple and efficient protocol for the Fe-catalyzed, intermolecular cross-dehydrogenative coupling of pyrimidine bearing 4-thiazolidinones systems and…”
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Palladium(0)-catalyzed aryne annulation: a powerful strategy for the synthesis of thio-bridged compounds by Morja, Mayur I., Chikhalia, Kishor H.

“…A method for the construction of various thio-bridged compounds is developed using readily available o-(trimethylsilyl)aryl triflates as a source of aryne…”
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Synthesis of benzimidazolyl-1,3,4-oxadiazol-2ylthio-N-phenyl (benzothiazolyl) acetamides as antibacterial, antifungal and antituberculosis agents by Patel, Rahul V., Patel, Paresh K., Kumari, Premlata, Rajani, Dhanji P., Chikhalia, Kishor H.

“…To affiliate multiple bioactivities in a compact heteronuclei, two series of benzimidazole based 1,3,4-oxadiazoles were synthesized and assessed in vitro for…”
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First-row transition metal for isocyanide-involving multicomponent reactions (IMCR) by Morja, Mayur I., Moradiya, Riddhi B., Chikhalia, Kishor H.

“…First-row transition metal catalyzed transformations that are able to construct complex molecules from simple, readily obtainable feedstocks have become a…”
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Multicomponent Approaches Involving Carbon Disulfide by Morja, Mayur I., Viradiya, Riddhi H., Chikhalia, Kishor H.

“…In present scenario, innovative carbon disulfide‐involving multicomponent protocols are extremely advantageous for practical and efficient construction of…”
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Cu‐catalyzed dehydrogenative CO arylation for the synthesis of 6‐methyl benzofuro[3,2‐c] quinoline derivatives by Makwana, Bhavik S., Morja, Mayur I., Chauhan, Prakashsingh M., Chikhalia, Kishor H.

“…A novel strategy for the synthesis of 6‐methyl benzofuro[3,2‐c] quinoline derivatives via copper‐catalyzed dehydrogenative CO arylation has been presented…”
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An efficient synthesis of designed 4‐thiazolidinone fused pyrimidine derivatives as potent antimicrobial agents by Patel, Janki J., Morja, Mayur I., Chikhalia, Kishor H.

“…A novel series of hybrid 2‐substituted ((pyrimidin‐2‐yl)hydrazinyl)thiazolidin‐4‐one derivatives were synthesized by means of aromatic nucleophilic…”
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Facile synthesis of benzonitrile/nicotinonitrile based s-triazines as new potential antimycobacterial agents by Patel, Amit B., Chikhalia, Kishor H., Kumari, Premlata

“…A common strategy to synthesize…”
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An efficient Pd-catalyzed intramolecular cyclization reaction followed by formation of benzimidazole derivatives: Synthesis of novel quinolin-fused benzo[d] azeto[1,2-a]benzimidazole analogues by Patel, Janki J., Patel, Anuj P., Chikhalia, Kishor H.

“…Novel quinolin-fused benzo[d]azeto[1,2-a]benzimidazole analogues have been synthesized from o-phenylene diamine and various substituted…”
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Privileged s-triazines: structure and pharmacological applications by Shah, Dhruvin R, Modh, Rahul P, Chikhalia, Kishor H

“…This review summarizes recent reports on s-triazine and its respective analogs from the medicinal chemistry angle. Due to its high reactivity and binding…”
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Comparative biological study between quinazolinyl–triazinyl semicarbazide and thiosemicarbazide hybrid derivatives by Patel, Janki J., Modh, Rahul P., Asamdi, Manjoorahmed, Chikhalia, Kishor H.

“…Practical synthesis and biological activities of quinazolinyl–triazinyl semicarbazides ( 10a – j ) and quinazolinyl–triazinyl thiosemicarbazides ( 11a – j )…”
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Iron‐catalyzed construction of cyanomethylated thiohydantoins by cross‐dehydrogenative C(sp3)‐C(sp3) coupling by Morja, Mayur I., Moradiya, Riddhi B., Makwana, Bhavik S., Chikhalia, Kishor H.

“…The efficient and novel approach for synthesizing cyanomethylated thiohydantoin from readily obtainable acetonitrile and 1,3‐dibenzyl‐2‐thiohydantoin through…”
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Synthesis and studies of novel 2-(4-cyano-3-trifluoromethylphenyl amino)-4-(quinoline-4-yloxy)-6-(piperazinyl/piperidinyl)- s-triazines as potential antimicrobial, antimycobacterial and anticancer agents by Patel, Rahul V., Kumari, Premlata, Rajani, Dhanji P., Chikhalia, Kishor H.

“…A series of novel s-triazine analogs were synthesized and characterized by IR, 1H NMR, 13C NMR, 19F NMR spectroscopy and elemental analysis. Preliminary…”
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Design, synthesis, antimicrobial activity and anti-HIV activity evaluation of novel hybrid quinazoline-triazine derivatives by Modh, Rahul P, De Clercq, Erik, Pannecouque, Christophe, Chikhalia, Kishor H

“…A series of novel hybrid quinazoline-triazine derivatives was designed and synthesized from cyanuric chloride and anthranilic acid through sequential…”
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Palladium-catalyzed acid-free Fujiwara–Moritani alkenylation of 4-thiazolidinones by Patel, Anuj, Patel, Janki, Chikhalia, Kishor H.

“…Herein, we report a facile method for the alkenylation of a 4-thiazolidinone motif without using external acid and high-pressure gas, which are required in…”
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Palladium(II)-catalyzed direct annulation of 2-chloronicotinaldehyde with 2-bromothiophenol via novel C(formyl)-C(aryl) coupling strategy by Morja, Mayur I., Chauhan, Prakashsingh M., Chikhalia, Kishor H.

“…An efficient and unprecedented method to the synthesis of 1-azathioxanthone derivatives has been developed by means of palladium-catalyzed C(formyl)-C(aryl)…”
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Design, synthesis, bioactivity, and computational studies of some morpholine-clubbed coumarinyl acetamide and cinnamide derivatives by Chauhan, Prakashsingh M., Thummar, Sandeep N., Chikhalia, Kishor H.

“…The novel derivatives of morpholine-clubbed 3-substituted coumarinyl acetamide and cinnamide derivatives 5a–5j and 6a–6j have been synthesized via various…”
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Recent Scenario for the Synthesis of Benzimidazole Moiety(2020–2022) by Choudhary, Annu, Viradiya, Riddhi H., Ghoghari, Rajnikant N., Chikhalia, Kishor H.

“…The benzene ring is fused to the 4 and 5 positions of the imidazole ring in the bicyclic heterocyclic aromatic compound known as benzimidazole. Benzimidazole…”
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Potent biological investigation into a new class of sulfone derivatives endowed with quinolinyl–cyclopropane analogue by Patel, Janki J., Morja, Mayur I., Chauhan, Prakashsingh M., Chikhalia, Kishor H.

“…Novel series of quinoline derivatives incorporating cyclopropyl ring and sulfone linkage as substituents have been synthesized, and oxidation of…”
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