Search Results - "Chernoburova, Elena I."

Secosteroid–quinoline hybrids as new anticancer agents by Ilovaisky, Alexey I., Scherbakov, Alexander M., Merkulova, Valentina M., Chernoburova, Elena I., Shchetinina, Marina A., Andreeva, Olga E., Salnikova, Diana I., Zavarzin, Igor V., Terent’ev, Alexander O.

“…An elegant approach to unknown secosteroid–quinoline hybrids is disclosed. A series of 13,17-secoestra-1,3,5(10)-trien-17-oic acid…”
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Secosteroid diacylhydrazines as novel effective agents against hormone-dependent breast cancer cells by Ilovaisky, Alexey I., Scherbakov, Alexander M., Chernoburova, Elena I., Shchetinina, Marina A., Merkulova, Valentina M., Bogdanov, Fedor B., Sorokin, Danila V., Salnikova, Diana I., Bozhenko, Eugene I., Zavarzin, Igor V., Terent’ev, Alexander O.

“…This research aimed to develop novel selective secosteroids that are highly active against hormone-dependent breast cancer. A simple and convenient approach to…”
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Secosteroid thiosemicarbazides and secosteroid–1,2,4-triazoles as antiproliferative agents targeting breast cancer cells: Synthesis and biological evaluation by Ilovaisky, Alexey I., Scherbakov, Alexander M., Chernoburova, Elena I., Povarov, Andrey A., Shchetinina, Marina A., Merkulova, Valentina M., Salnikova, Diana I., Sorokin, Danila V., Bozhenko, Eugene I., Zavarzin, Igor V., Terent’ev, Alexander O.

“…A convenient and selective approach to 13,17-secoestra-1,3,5(10)-trien-17-oic acid [N’-arylcarbothioamido]hydrazides and hybrid molecules containing…”
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Secosteroidal hydrazides: Promising scaffolds for anti-breast cancer agents by Ilovaisky, Alexey I., Merkulova, Valentina M., Chernoburova, Elena I., Shchetinina, Marina A., Salnikova, Diana I., Scherbakov, Alexander M., Zavarzin, Igor V., Terent’ev, Alexander O.

“…[Display omitted] •A selective approach to antitumor agents based on the opening of ring D in steroidal lactones by hydrazines was developed.•Secosteroidal…”
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Regioselective Baeyer–Villiger Oxidation of Steroidal Ketones to Lactones Using BF3/H2O2 by Ilovaisky, Alexey I., Merkulova, Valentina M., Vil', Vera A., Chernoburova, Elena I., Shchetinina, Marina A., Loguzov, Sergey D., Dmitrenok, Andrey S., Zavarzin, Igor V., Terent'ev, Alexander O.

“…A regioselective Baeyer–Villiger oxidation of estrone and androstane derivatives into 17a‐oxa‐D‐homosteroids was developed. An important feature of this…”
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A Straightforward Approach toward Multifunctionalized Pyridazines via Imination/Electrocyclization by Komkov, Alexander V, Komendantova, Anna S, Menchikov, Leonid G, Chernoburova, Elena I, Volkova, Yulia A, Zavarzin, Igor V

“…A facile synthesis of functionalized 3-carbamide pyridazines starting from readily available chlorovinyl aldehydes and oxamic acid thiohydrazides via cascade…”
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Novel steroidal 1,3,4-thiadiazines: Synthesis and biological evaluation in androgen receptor-positive prostate cancer 22Rv1 cells by Komendantova, Anna S., Scherbakov, Alexander M., Komkov, Alexander V., Chertkova, Viktoriya V., Gudovanniy, Alexey O., Chernoburova, Elena I., Sorokin, Danila V., Dzichenka, Yaraslau U., Shirinian, Valerii Z., Volkova, Yulia A., Zavarzin, Igor V.

“…[Display omitted] •A series of novel steroidal 1,3,4-thiadiazines were synthesized.•Their antiproliferative activity against androgen receptor-positive…”
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Synthesis and evaluation of avermectin–imidazo[1,2-a]pyridine hybrids as potent GABAA receptor modulators by Volkova, Yulia A., Rassokhina, Irina V., Kondrakhin, Eugeny A., Rossokhin, Alexey V., Kolbaev, Sergey N., Tihonova, Tatiana B., Kh. Dzhafarov, Mamedsalim, Schetinina, Marina A., Chernoburova, Elena I., Vasileva, Ekaterina V., Dmitrenok, Andrey S., Kovalev, Georgy I., Sharonova, Irina N., Zavarzin, Igor V.

“…[Display omitted] •A series of hybrid molecules based on Avermectin and imidazopyridine pharmacophores acting as GABAARs PAMs were designed.•In each of these…”
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Reactions of hydrazones derived from oxamic acid thiohydrazides by Volkova, Yulia A., Chernoburova, Elena I., Petrova, Albina S., Shtil, Alexander A., Zavarzin, Igor V.

“…This brief review describe the recent advances in using oxamic acid thiohydrazides as precursors for the formation of hydrazones intermediates from natural and…”
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Synthesis of 1'-arylcarbamoylthiocarbonyl-3'-methyl-3-oxo-androst-4-eno[16α,17α-d]pyrazolines by Zavarzin, Igor V., Kamernitsky, Aleksey. V., Chertkova, Viktoriya. V., Chernoburova, Elena. I., Yarovenko, Vladimir. N., Kraushkin, Michael. M., Kachala, Vadim V.

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(XantPhos)AgBr as a cheap and readily available catalyst for the bromofluorocyclopropanation of electron-rich alkenes by Novikov, Maxim A., Bobrova, Angelina Yu, Servetnik, Anton A., Chernoburova, Elena I., Zavarzin, Igor V., Tomilov, Yury V.

“…[Display omitted] A silver phosphine complex (XantPhos)AgBr proved to be a cheap and readily accessible catalyst for bromofluoro- cyclopropanation of…”
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Regioselective Baeyer–Villiger Oxidation of Steroidal Ketones to Lactones Using BF 3 /H 2 O 2 by Ilovaisky, Alexey I., Merkulova, Valentina M., Vil', Vera A., Chernoburova, Elena I., Shchetinina, Marina A., Loguzov, Sergey D., Dmitrenok, Andrey S., Zavarzin, Igor V., Terent'ev, Alexander O.

“…A regioselective Baeyer–Villiger oxidation of estrone and androstane derivatives into 17a‐oxa‐ D ‐homosteroids was developed. An important feature of this…”
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Thiooxamide chiral stationary phase for liquid chromatography by Shamshurin, Dmitri V., Zavarzin, Igor V., Yarovenko, Vladimir N., Chernoburova, Elena I., Krayushkin, Mikhail M., Volgin, Yuri V., Shapovalova, Elena N., Nesterenko, Pavel N., Shpigun, Oleg A.

“…A new chiral stationary phase was prepared by reaction of aminopropylsilica with N-(α-phenylethyl)chloroacetamide in the presence of sulfur and used for the…”
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