Search Results - "Chabane, Hadjila"

Microwave-assisted synthesis of novel thiazolocarbazoles and evaluation as potential anticancer agents. Part III by Testard, Alexandra, Picot, Laurent, Fruitier-Arnaudin, Ingrid, Piot, Jean-Marie, Chabane, Hadjila, Domon, Lisianne, Thiery, Valerie, Besson, Thierry

“…Novel 6-substituted thiazolocarbazole derivatives have been synthesized under microwave irradiation via the corresponding imino-1,2,3-dithiazoles. In vitro…”
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Simple and efficient solid-phase synthesis of unprotected peptide aldehyde for peptide segment ligation by Lelièvre, Dominique, Chabane, Hadjila, Delmas, Agnès

“…We describe an efficient solid-phase synthesis of C-terminal peptide aldehyde. Making use of the stability of the PAM linker towards both acid and base…”
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Identification and pharmacological properties of E339-3D6, the first nonpeptidic apelin receptor agonist by Iturrioz, Xavier, Alvear-Perez, Rodrigo, De Mota, Nadia, Franchet, Christel, Guillier, Fabrice, Leroux, Vincent, Dabire, Hubert, Le Jouan, Melissande, Chabane, Hadjila, Gerbier, Romain, Bonnet, Dominique, Berdeaux, Alain, Maigret, Bernard, Galzi, Jean-Luc, Hibert, Marcel, Llorens-Cortes, Catherine

“…Apelin plays a prominent role in body fluid and cardiovascular homeostasis. To explore further upstream the role played by this peptide, nonpeptidic agonists…”
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Structure–Activity Relationship Studies toward the Discovery of Selective Apelin Receptor Agonists by Margathe, Jean-François, Iturrioz, Xavier, Alvear-Perez, Rodrigo, Marsol, Claire, Riché, Stéphanie, Chabane, Hadjila, Tounsi, Nassera, Kuhry, Maxime, Heissler, Denis, Hibert, Marcel, Llorens-Cortes, Catherine, Bonnet, Dominique

“…Apelin is the endogenous ligand for the previously orphaned G protein-coupled receptor APJ. Apelin and its receptor are widely distributed in the brain, heart,…”
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Synthesis of original thiazoloindolo[3,2-c]quinoline and novel 8-N-substituted-11H-indolo[3,2-c]quinoline derivatives from benzotriazoles. Part I by Beauchard, Anne, Chabane, Hadjila, Sinbandhit, Sourisak, Guenot, Pierre, Thiéry, Valérie, Besson, Thierry

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Synthesis of novel 2-cyanothiazolocarbazoles analogues of ellipticine by Chabane, Hadjila, Lamazzi, Christelle, Thiéry, Valérie, Guillaumet, Gérald, Besson, Thierry

“…Novel linear thiazolocarbazoles, which are structurally very close to the natural alkaloid ellipticine, have been rapidly synthesised via…”
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Synthesis of original thiazoloindolo[3,2- c]quinoline and novel 8- N-substituted-11 H-indolo[3,2- c]quinoline derivatives from benzotriazoles. Part I by Beauchard, Anne, Chabane, Hadjila, Sinbandhit, Sourisak, Guenot, Pierre, Thiéry, Valérie, Besson, Thierry

“…Synthesis of novel thiazoloindolo[3,2- c]quinoline and 8-substituted-11 H-indolo[3,2- c]quinolines was performed via Graebe–Ullmann thermal cyclization from…”
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Synthesis and cytotoxic activity of thiazolofluorenone derivatives by Chabane, Hadjila, Pierre, Alain, Leonce, Stephane, Pfeiffer, Bruno, Renard, Pierre, Thiery, Valerie, Guillaumet, Gerald, Besson, Thierry

“…The synthesis and biological evaluation of some novel thiazolofluorenones, thiazolofluorenes and thiazoloanthraquinones, substituted with amino side-chains are…”
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Cycloadditions of NS functions to cyclopentadienones by Chabane, Hadjila, Meth-Cohn, Otto, Rees, Charles W., White, Andrew J.P., Williams, David J.

“…Cyclopentadienones react with EtO 2CNSO and related NS reagents to provide ready syntheses of 1,2,5-thiadiazolidines ( 8 , 12 , 17 ), diaminosulfanes ( 11 ,…”
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Synthesis and cytotoxic evaluation of novel thiazolocarbazoles. Part III by Chabane, Hadjila, Lamazzi, Christelle, Thiery, Valerie, Pierre, Alain, Leonce, Stephane, Pfeiffer, Bruno, Renard, Pierre, Guillaumet, Gérald, Besson, Thierry

“…Novel thiazolocarbazole derivatives have been synthesized via the corresponding imino-1,2,3-dithiazoles. In vitro antitumor activity of these polyheterocyclic…”
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Synthesis and cytotoxic evaluation of novel thiazolocarbazoles by Lamazzi, Christelle, Chabane, Hadjila, Thiery, Valerie, Pierre, Alain, Leonce, Stephane, Pfeiffer, Bruno, Renard, Pierre, Guillaumet, Gérald, Besson, Thierry

“…Novel thiazolocarbazole derivatives 4 and 5 have been synthesized via the corresponding imino-1,2,3-dithiazoles 3. In vitro antitumor activity of these…”
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