Search Results - "Casara, P J"

Cure of Trypanosoma brucei brucei and Trypanosoma brucei rhodesiense infections in mice with an irreversible inhibitor of S-adenosylmethionine decarboxylase by Bitonti, A J, Byers, T L, Bush, T L, Casara, P J, Bacchi, C J, Clarkson, Jr, A B, McCann, P P, Sjoerdsma, A

“…Classifications Services AAC Citing Articles Google Scholar PubMed Related Content Social Bookmarking CiteULike Delicious Digg Facebook Google+ Mendeley Reddit…”
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General synthesis of 3-substituted alkenyl gaba as potential anticonvulsants by Serfass, Lucile, Casara, Patrick J.

“…stereospecific synthesis of cis and trans 3-substituted vinyl-γ-aminobutyric acid analogs were obtained by either a Claisen rearrangement or a Wittig reaction…”
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Catalytic irreversible inhibition of bacterial and plant arginine decarboxylase activities by novel substrate and product analogues by Bitonti, A J, Casara, P J, McCann, P P, Bey, P

“…Arginine decarboxylase (ADC) activity from Escherichia coli and two plant species (oats and barley) was inhibited by five new substrate (arginine) and product…”
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Synthesis of N, N′-disubstituted 3-aminobenzo[ c] and [ d]azepin-2-ones as potent and specific farnesyl transferase inhibitors by Le Diguarher, Thierry, Ortuno, Jean-Claude, Shanks, David, Guilbaud, Nicolas, Pierré, Alain, Raimbaud, Eric, Fauchère, Jean-Luc, Hickman, John A, Tucker, Gordon C, Casara, Patrick J

“…A structure–activity study was performed by synthesis on N, N′-disubstitution of 3-aminobenzo[ c] and [ d]azepin-2-one 2 and 3 to afford potent and specific…”
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Decrease in survival threshold of quiescent colon carcinoma cells in the presence of a small molecule integrin antagonist by Burbridge, Mike F, Venot, Virginie, Casara, Patrick J, Perron-Sierra, Françoise, Hickman, John A, Tucker, Gordon C

“…The role of adhesion molecules, such as alphav integrins, in the control of the survival of quiescent tumor cells is unclear. We used S 34961, a novel small…”
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Parallel liquid synthesis of N, N′-Disubstituted 3-amino azepin-2-ones as potent and specific farnesyl transferase inhibitors by Le Diguarher, Thierry, Ortuno, Jean-Claude, Dorey, Gilbert, Shanks, David, Guilbaud, Nicolas, Pierré, Alain, Fauchère, Jean-Luc, Hickman, John A., Tucker, Gordon C., Casara, Patrick J.

“…A rapid structure–activity study was performed by parallel liquid synthesis on N, N′-disubstitution of 3-amino azepin-2-one to afford potent and specific…”
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Cure of Trypanosoma brucei brucei and Trypanosoma brucei rhodesiense infectious in mice with an irreversible inhibitor of S-adenosylmethionine decarboxylase by BITONTI, A. J, BYERS, T. L, BUSH, T. L, CASARA, P. J, BACCHI, C. J, CLARKSON, A. B. JR, MCCANN, P. P, SJOERDSMA, A

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Synthesis and antiviral activity of rigid acyclonucleotide analogs by Casara, Patrick J., Altenburger, Jean-Michel, Taylor, Debra L., Stanley Tyms, A., Kenny, Michael, Navé, Jean-François

“…The synthesis, anti-HIV-1 and anti-herpesvirus activities of new rigid acyclonucleotide analogs are described…”
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Synthesis, enzymatic phosphorylation and antiviral activity of acyclic dienyl phosphonate derivatives of guanine by Navé, Jean-François, Casara, Patrick J., Taylor, Debra L., Stanley Tyms, A., Kenny, Michael, HalazyS, Serge

“…The synthesis, phosphorylation by guanylate kinase, anti HIV-1 and anti-herpesvirus activity of two acyclic dienyl phosphonate derivatives of guanine are…”
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