Search Results - "Caldirola, Patrizia"

Novel 2-Aminotetralin and 3-AminoChroman Derivatives as Selective Serotonin 5-HT7 Receptor Agonists and Antagonists by Holmberg, Pär, Sohn, Daniel, Leideborg, Robert, Caldirola, Patrizia, Zlatoidsky, Pavel, Hanson, Sverker, Mohell, Nina, Rosqvist, Susanne, Nordvall, Gunnar, Johansson, Anette M, Johansson, Rolf

“…The understanding of the physiological role of the G-protein coupled serotonin 5-HT7 receptor is largely rudimentary. Therefore, selective and potent…”
Get full text

Integrin α5β1 Inhibition by CLT-28643 Reduces Postoperative Wound Healing in a Mouse Model of Glaucoma Filtration Surgery by Van Bergen, Tine, Zahn, Grit, Caldirola, Patrizia, Fsadni, Mario, Caram-Lelham, Ninus, Vandewalle, Evelien, Moons, Lieve, Stalmans, Ingeborg

“…To evaluate the therapeutic potential of the small molecule integrin α5β1 inhibitor, CLT-28643, to improve the filtering surgery outcome in a mouse model…”
Get full text

[alpha]5[beta]1-Integrin inhibitor (CLT-28643) effective in rabbit trabeculectomy model by Schultheiss, Maximilian, Schnichels, Sven, Konrad, Eva-Maria, Bartz-Schmidt, Karl U, Zahn, Grit, Caldirola, Patrizia, Fsadni, Mario G, Caram-Lelham, Ninus, Spitzer, Martin S

“…Purpose Glaucoma filtration surgery (GFS) fails due to fibrosis. The [alpha]5[beta]1-integrin plays a pivotal role in fibrosis, angiogenesis and inflammation…”
Get full text

α 5 β 1‐Integrin inhibitor ( CLT ‐28643) effective in rabbit trabeculectomy model by Schultheiss, Maximilian, Schnichels, Sven, Konrad, Eva‐Maria, Bartz‐Schmidt, Karl U., Zahn, Grit, Caldirola, Patrizia, Fsadni, Mario G., Caram‐Lelham, Ninus, Spitzer, Martin S.

“…Purpose Glaucoma filtration surgery (GFS) fails due to fibrosis. The alpha 5 beta 1-integrin plays a pivotal role in fibrosis, angiogenesis and inflammation…”
Get full text

α5β1‐Integrin inhibitor (CLT‐28643) effective in rabbit trabeculectomy model by Schultheiss, Maximilian, Schnichels, Sven, Konrad, Eva‐Maria, Bartz‐Schmidt, Karl U., Zahn, Grit, Caldirola, Patrizia, Fsadni, Mario G., Caram‐Lelham, Ninus, Spitzer, Martin S.

“…Purpose Glaucoma filtration surgery (GFS) fails due to fibrosis. The α5β1‐integrin plays a pivotal role in fibrosis, angiogenesis and inflammation. This is the…”
Get full text

Novel 2-Aminotetralin and 3-AminoChroman Derivatives as Selective Serotonin 5-HT 7 Receptor Agonists and Antagonists by Holmberg, Pär, Sohn, Daniel, Leideborg, Robert, Caldirola, Patrizia, Zlatoidsky, Pavel, Hanson, Sverker, Mohell, Nina, Rosqvist, Susanne, Nordvall, Gunnar, Johansson, Anette M., Johansson, Rolf

Get full text

trans-3,4-Disubstituted pyrrolidines by 1,3-dipolar cycloaddition: enantioselective approaches and their limitations by Karlsson, Staffan, Han, Fusen, Högberg, Hans-Erik, Caldirola, Patrizia

“…In the presence of a chiral Lewis acid as co-catalyst, the acid-catalysed 1,3-dipolar cycloaddition reaction yielding trans-3,4-disubstituted pyrrolidines from…”
Get full text

Intramolecular Transfer of CO from (.eta.6-arene)Cr(CO)3 Complexes in Stille-Type Palladium-Catalyzed Cross-Coupling Reactions by Caldirola, Patrizia, Chowdhury, Ratan, Johansson, Anette M, Hacksell, Uli

Get full text

Alkylation of Tricarbonylchromium-Stabilized Benzylic Anions of 3-(Dipropylamino)chroman by Brisander, Magnus, Caldirola, Patrizia, Johansson, Anette M, Hacksell, Uli

“…Tricarbonylchromium complexes of racemic and resolved 3-(dipropylamino)chromans were prepared. Benzylic alkylation of the complexes provided access to…”
Get full text

Novel derivatives of 3-(dipropylamino)chroman. Interactions with 5-HT 1A and D 2A receptors by Caldirola, Patrizia, Chowdhury, Ratan, Unelius, Lena, Mohell, Nina, Hacksell, Uli, Johansson, Anette M.

“…Novel 8-aryl and 8-aroyl substituted derivatives of 3-(dipropylamino)chroman are described. The compounds have been prepared by a palladium catalyzed reaction…”
Get full text

Novel derivatives of 3-(dipropylamino)chroman. Interactions with 5-HT1A and D2A receptors by CALDIROLA, P, CHOWDHURY, R, UNELIUS, L, MOHELL, N, HACKSELL, U, JOHANSSON, A. M

“…Novel 8-aryl and 8-aroyl substituted derivatives of 3-(dipropylamino)chroman are described. The compounds have been prepared by a palladium catalyzed reaction…”
Get full text

Resolved pyrrolidine, piperidine, and perhydroazepine analogs of the muscarinic agent N-methyl-N-(1-methyl-4-pyrrolidino-2-butynyl)acetamide by Lundkvist, J. R. Michael, Vargas, Hugo M, Caldirola, Patrizia, Ringdahl, Bjoern, Hacksell, Uli

“…A series of conformationally restricted analogues of the partial muscarinic agonist N-methyl-N-(1-methyl-4-pyrrolidino-2-butynyl)acetamide (BM 5; 1) was…”
Get full text

A New synthesis of 4,5,6,7-tetrahydrofuro[2,3-c]pyridines and furo[2,3-c]pyrrolidines by Arnoldi, Anna, Bregante, Giovanna, Caldirola, Patrizia, Merlini, Lucio, Tamburini, Bruno

“…New syntheses of 4,5,6,7‐tetrahydrofuro[2,3‐c]pyridines and furo[2,3‐c]pyrrolidine derivatives, starting from furan‐3‐carboxaldehyde, are reported…”
Get full text

An efficient synthesis of isoxazoles and isoxazolines by CALDIROLA, P, DE AMICI, M, DE MICHELI, C

Get full text

In vitro and in vivo characterization of a calcium modulator of the diphenylalkylamine type with selective coronary dilatory properties by Caldirola, P, Monteil, A, Zandberg, P, Mannhold, R, Timmerman, H

“…VUF 8929 (N-¿2-[bis(p-fluorophenyl)methoxy]ethyl¿-(2-phenyl)ethylamine maleate, CAS 140890-71-7) is a diphenylalkylamine derivative structurally related to…”
Get more information