Search Results - "Cadoni, Roberta"

Carbonic anhydrases from Trypanosoma cruzi and Leishmania donovani chagasi are inhibited by benzoxaboroles by Nocentini, Alessio, Cadoni, Roberta, Dumy, Pascal, Supuran, Claudiu T., Winum, Jean-Yves

“…A series of 6-substituted ureido- and thioureido-benzoxaboroles were investigated as inhibitors of carbonic anhydrases from Trypanosoma cruzi (TcCA), and…”
Get full text

Exploring benzoxaborole derivatives as carbonic anhydrase inhibitors: a structural and computational analysis reveals their conformational variability as a tool to increase enzyme selectivity by Langella, Emma, Alterio, Vincenzo, D'Ambrosio, Katia, Cadoni, Roberta, Winum, Jean-Yves, Supuran, Claudiu T., Monti, Simona Maria, De Simone, Giuseppina, Di Fiore, Anna

“…Recent studies identified the benzoxaborole moiety as a new zinc-binding group able to interact with carbonic anhydrase (CA) active site. Here, we report a…”
Get full text

One-Pot Synthesis of Amides from Aldehydes and Amines via C–H Bond Activation by Cadoni, Roberta, Porcheddu, Andrea, Giacomelli, Giampaolo, De Luca, Lidia

“…A one-pot synthesis of amides from aldheydes with N-chloroamines, prepared in situ from amines, has been developed. Both aliphatic and aromatic aldehydes and…”
Get full text

A fast and efficient one-pot microwave assisted synthesis of variously di-substituted 1,2,4-oxadiazoles by Porcheddu, Andrea, Cadoni, Roberta, De Luca, Lidia

“…A one-pot two-step microwave assisted synthesis of variously disubstituted 1,2,4-oxadiazoles from carboxylic acids and amidoximes is reported. This methodology…”
Get more information

Benzoxaborole as a new chemotype for carbonic anhydrase inhibition by Alterio, Vincenzo, Cadoni, Roberta, Esposito, Davide, Vullo, Daniela, Fiore, Anna Di, Monti, Simona Maria, Caporale, Andrea, Ruvo, Menotti, Sechi, Mario, Dumy, Pascal, Supuran, Claudiu T, De Simone, Giuseppina, Winum, Jean-Yves

“…In this paper we report the synthesis of a series of benzoxaborole derivatives, their inhibition properties against some carbonic anhydrases (CAs), recognized…”
Get more information

Benzoxaboroles as Efficient Inhibitors of the β‑Carbonic Anhydrases from Pathogenic Fungi: Activity and Modeling Study by Nocentini, Alessio, Cadoni, Roberta, del Prete, Sonia, Capasso, Clemente, Dumy, Pascal, Gratteri, Paola, Supuran, Claudiu T, Winum, Jean-Yves

“…A series of 6-substituted benzoxaboroles were investigated as inhibitors of the β-class carbonic anhydrase from three pathogenic fungi (Cryptococcus…”
Get full text

Benzoxaboroles: New Potent Inhibitors of the Carbonic Anhydrases of the Pathogenic Bacterium Vibrio cholerae by Bonardi, Alessandro, Nocentini, Alessio, Cadoni, Roberta, del Prete, Sonia, Dumy, Pascal, Capasso, Clemente, Gratteri, Paola, Supuran, Claudiu T, Winum, Jean-Yves

“…A series of urea/thiourea substituted benzoxaboroles was investigated for the inhibition of the three carbonic anhydrases encoded by Vibrio cholerae (VchCAα,…”
Get full text

Exploring Heteroaryl-pyrazole Carboxylic Acids as Human Carbonic Anhydrase XII Inhibitors by Cadoni, Roberta, Pala, Nicolino, Lomelino, Carrie, Mahon, Brian P, McKenna, Robert, Dallocchio, Roberto, Dessì, Alessandro, Carcelli, Mauro, Rogolino, Dominga, Sanna, Vanna, Rassu, Mauro, Iaccarino, Ciro, Vullo, Daniela, Supuran, Claudiu T, Sechi, Mario

“…We report the synthesis, biological evaluation, and structural study of a series of substituted heteroaryl-pyrazole carboxylic acid derivatives. These…”
Get full text