Search Results - "COUSSY, L"
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Up‐regulation of [3H]‐des‐Arg10‐kallidin binding to the bradykinin B1 receptor by interleukin‐1β in isolated smooth muscle cells: correlation with B1 agonist‐induced PGI2 production
Published in British journal of pharmacology (01-10-1994)“…1 Binding of the specific bradykinin B1 receptor agonist, [3H]‐des‐Arg10‐kallidin (‐KD) was investigated in smooth muscle cells (SMC) isolated from rabbit…”
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G-Protein-Coupled Receptor Affinity Prediction Based on the Use of a Profiling Dataset: QSAR Design, Synthesis, and Experimental Validation
Published in Journal of medicinal chemistry (20-10-2005)“…A QSAR model accounting for “average” G-protein-coupled receptor (GPCR) binding was built from a large set of experimental standardized binding data (1939…”
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QSAR Strategy and Experimental Validation for the Development of a GPCR Focused Library
Published in QSAR & combinatorial science (01-06-2005)“…An innovative approach has been developed in order to construct new GPCR focused libraries. Experimental binding data generated in house from 1939 diverse drug…”
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Journal Article