Search Results - "CHIARELOTTO, G"

Novel Pyrrolo[3,2- f]quinolines: Synthesis and Antiproliferative Activity by Ferlin, M.G, Gatto, B, Chiarelotto, G, Palumbo, M

“…Novel pyrrolo[3,2, f]quinoline derivatives have been synthesized and tested as antiproliferative agents. They are characterized by an angular aromatic…”
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Pyrrolo-quinoline derivatives as potential antineoplastic drugs by FERLIN, M. G, GATTO, B, CHIARELOTTO, G, PALUMBO, M

“…Some novel pyrrolo-quinoline derivatives have been synthesized as potential antineoplastic agents. They contain an angular aromatic tricyclic or tetracyclic…”
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Synthesis and in Vitro and in Vivo Antitumor Activity of 2-Phenylpyrroloquinolin-4-ones by Ferlin, Maria Grazia, Chiarelotto, Gianfranco, Gasparotto, Venusia, Dalla Via, Lisa, Pezzi, Vincenzo, Barzon, Luisa, Palù, Giorgio, Castagliuolo, Ignazio

“…In our search for potential new anticancer drugs, we designed and synthesized a series of tricyclic compounds containing the antimitotic 2-phenylazaflavone…”
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Synthesis and biological properties of a new series of N-pyrido substituted tetrahydrocarbazoles by Ferlin, M.G., Chiarelotto, G., Marzano, C., Severin, E., Baccichetti, F., Carlassare, F., Simonato, M., Bordin, F.

“…A series of methyl and ethyl quaternary pyridiniumtetrahydrocarbazoles was synthesized and studied in comparison with ellipticine, chosen as a reference. In…”
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Synthesis and Biological Activity of 7-Phenyl-6,9-dihydro-3H-pyrrolo[3,2-f]quinolin-9-ones:  A New Class of Antimitotic Agents Devoid of Aromatase Activity by Gasparotto, Venusia, Castagliuolo, Ignazio, Chiarelotto, Gianfranco, Pezzi, Vincenzo, Montanaro, Daniela, Brun, Paola, Palù, Giorgio, Viola, Giampietro, Ferlin, Maria Grazia

“…The newly synthesized 7-phenyl-3H-pyrrolo[3,2-f]quinolinones 16 − 26 and previously 27 and 28 were assayed for their in vitro antiproliferative activity on…”
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A mass spectrometric investigation on some 4,7-dioxo-4,5,6,7-tetrahydroindole derivatives by Bertazzo, A., Ferlin, M. G., Chiarelotto, G., Catinella, S., Traldi, P.

“…The mass spectrometric behaviour of a series of 2‐aryl substituted 4,7‐dioxo‐4,5,6,7‐tetrahydroindoles has been studied in different ionization conditions…”
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Novel anellated pyrazoloquinolin-3-ones: synthesis and in vitro BZR activity by Ferlin, Maria Grazia, Chiarelotto, Gianfranco, Dall’Acqua, Stefano, Maciocco, Elisabetta, Mascia, Maria Paola, Pisu, Maria Giuseppina, Biggio, Giovanni

“…New pyrazolopyrroloquinolinones were synthesized and showed high affinity for central BZRs acting as antagonists. None turned out to be active in inhibiting…”
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New mono- and bis-intercalating compounds between DNA base pairs by Chiarelotto, G, Ferlin, M G, Vedaldi, D, Dall'Acqua, F, Rodighiero, G

“…With the aim to obtain new bis-intercalating agents in DNA a series of compounds was prepared linking two identical tricyclic moieties (two…”
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Mannich bases of 3H-pyrrolo[3,2-f]quinoline having vasorelaxing activity by FERLIN, Maria Grazia, CHIARELOTTO, Gianfranco, ANTONUCCI, Francesca, CAPARROTTA, Laura, FROLDI, Guglielmina

“…Mannich bases obtained by aminoalkylation of 3H-pyrrolo[3,2-f]quinoline were designed and prepared as potential vasorelaxing agents. Compounds Ia-Va were…”
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2-substituted 1H-pyrrolo [3,2-h] quinoline derivatives: synthesis and aspects of their biological activity by Ferlin, M G, Chiarelotto, G, Baccichetti, F, Carlassare, F, Toniolo, L, Bordin, F

“…Certain 2-substituted 1H-pyrrolo [3,2-h] quinolines have been prepared and their biological activity in mammalian cells and in some microorganisms have been…”
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Preparation and antiproliferative activity of 1H-pyrrolo [2,3-f]quinolinium and isoquinolinium iodides by Ferlin, M G, Chiarelotto, G, Gia, O, Baccichetti, F, Carlassare, F

“…2-Carbomethoxy-N-methyl-1H-pyrrolo[2,3-f]quinolinium and isoquinolinium iodides were prepared. Their in vitro ability to form complexes with DNA is enhanced in…”
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1H-pyrrolo[2,3-f]quinoline and isoquinoline derivatives: synthesis and antiproliferative activity by Ferlin, M G, Chiarelotto, G, Basadonna, O, Gia, O, Mobilio, S, Baccichetti, F, Carlassare, F

“…Fischer indol synthesis is reported for the preparation of some 2-substituted 1H-pyrrolo[2,3-f]quinoline and isoquinoline derivatives having a structural…”
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Synthesis and antiproliferative activity of some variously substituted acridine and azacridine derivatives by FERLIN, M. G, MARZANO, C, CHIARELOTTO, G, BACCICHETTI, F, BORDIN, F

“…A group of 9-substituted acridine and azacridine derivatives (m-AMSA analogues) were synthesised following classical procedures as potential antitumour agents…”
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Synthesis and characterization of some N-mannich bases of [1,2,3]triazoloquinolines by Ferlin, Maria Grazia, Chiarelotto, Gianfranco, Castagliuolo, Ignazio

“…Some novel N‐Mannich bases of [1,2,3]‐triazolo[4,5‐f] and [4,5‐h]quinolines were synthesized following the classical experimental procedure for Mannich base…”
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Synthesis of novel methoxy and hydroxy derivatives of 2-phenyl-1H-ben[g]indoles by FERLIN, M. G, CHIARELOTTO, G, MALESANI, G

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Synthesis of novel methoxy and hydroxy derivatives of 2-phenyl-1H-benz[g]indoles by Ferlin, Maria Grazia, Chiarelotto, Gianfranco, Malesani, Giorgio

“…The synthesis of novel methoxy‐derivatives of 2‐phenyl‐1H‐benz[g]indole 3 by condensation of α‐naphthyl‐amines 1 with N‐phenacyl‐pyridinium salts 2 is…”
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Antiproliferative activity of some unsubstituted angular analogoues of ellipticine by Ferlin, M G, Chiarelotto, G, Marzano, C, Mobilio, S, Carlassare, F, Baccichetti, F

“…With the aim of obtaining further knowledge on the antiproliferative activity of pyrroloquinolines and isoquinolines, we prepared four unsubstituted angular…”
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Antimicrobial properties of some 3-acyl-4,7-disubstituted indoles by Malesani, G, Chiarelotto, G, Dall'Acqua, F, Vedaldi, D

“…In continuation of research on indole derivatives as potential chemotherapeutic agents, the antimicrobial properties of some 4,7-disubstituted 3-acylindoles…”
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Carboxylation and acylation of 4,7-dimethoxyindoles and a study of the corresponding dealkylated derivatives by Malesani, Giorgio, Chiarelotto, Gianfranco, Ferlin, Maria Grazia, Masiero, Sergio

“…Treatment of 4,7‐dimethoxyindoles 1 and 9 with ethylmagnesium bromide and ethyl chloroformate in refluxing dry ether gives the corresponding…”
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Bis-pyridoquinolines as new bifunctional intercalators for DNA by Malesani, G, Chiarelotto, G, Ferlin, M G, Bordin, F, Baccichetti, F, Carlassare, F, Vedaldi, D, Dall'Acqua, F

“…With the aim of obtaining new bifunctional intercalators for DNA, a new series of bis-pyridoquinolines were synthesized by joining two tricyclic planar…”
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